Substrate | Species | Linear Range | Conditions for Kinetic Study | |||||
---|---|---|---|---|---|---|---|---|
Incubation Time | Protein Concentration | Incubation Time | Protein Concentration | MNTX Concentration | ||||
M4 | M5 | M4 | M5 | |||||
min | min | mg/ml | mg/ml | min | mg/ml | μM | ||
MNTX | Mouse | N.A. | 0–120 | 0–6.0 | 0–6.0 | 120 | 4.0 | 5–2000 |
Rat | N.A. | 0–120 | N.A. | 0–6.0 | 120 | 4.0 | 5–5000 | |
Monkey | 0–60 | 0–60 | 0–6.0 | 0–6.0 | 60 | 4.0 | 5–2000 | |
Human | 0–120 | 0–120 | 0–4.0 | 0–4.0 | 120 | 1.0 | 0.5–5000 | |
Naltrexone | Human | 0–120 | 0–0.5 | 30 | 0.5 | 5–1000 |
N.A., not applicable.