Compound | Relative Vmax | Km | Ki |
---|---|---|---|
peak area of glucuronide/mg protein/min | μM | ||
Alprazolam | 169 | 261 | N.A. |
Fluconazole | 158 | 1667 | N.A. |
Itraconazole | No data | No data | No data |
Voriconazole | 436 | 1130 | N.A. |
Tioconazole | 31445 | 124 | 245 |
Ketoconazole | 541 (n = 2) | 7 (n = 2) | 941 (n = 2) |
Econazole | 6532 | 115 | 192 |
Miconazole | 7513 | 58.7 | 475 |
Bifonazole | 13268 | 28 | 47 |
Sulconazole | 4902 | 35 | 290 |
N.A., not applicable.