TABLE 2
Inhibitory conditions of fluorescence bioassay
Enzyme
Inhibitor
Concentrations (μM)
Microsomes
THLE Cells
CYP1A2
α-NF
5
0.1
CYP3A4
TAO
50
50
CYP2D6
Quinidine
20
10
COMT
Ro 41-0960
10
GST
BSO
50