Reference Compounds | Papp | Faa | Model Compounds | Papp |
---|---|---|---|---|
(×10−6 cm/s) | (×10−6 cm/s) | |||
Acetaminophen | 2.8 | 0.80 | Alprazolam | 7.0 |
Acyclovir | 0.0 | 0.21 | Amlodipine | 19.5 |
Alprenolol | 37.2 | 0.94 | Clonazepam | 18.6 |
Amphotericin B | 0.0 | 0.05 | Midazolam | 30.8 |
Antipyrine | 2.6 | 1.00 | Nifedipine | 13.4 |
Atenolol | 0.1 | 0.52 | Nicardipine | 31.5 |
Caffeine | 2.0 | 1.00 | Quinidine | 17.9 |
Carbamazepine | 27.7 | 1.00 | Tacrolimus | 34.3 |
Diclofenac | 32.9 | 1.00 | Verapamil | 35.8 |
Furosemide | 0.2 | 0.60 | ||
Hydrochlorothiazide | 0.1 | 0.70 | ||
Indomethacin | 22.4 | 1.00 | ||
Ketoprofen | 12.7 | 1.00 | ||
Ketorolac | 4.0 | 1.00 | ||
Metoprolol | 11.3 | 0.95 | ||
Nadolol | 0.0 | 0.32 | ||
Naproxen | 11.1 | 0.98 | ||
Piroxicam | 16.1 | 1.00 | ||
Prednisone | 14.3 | 0.99 | ||
Propranolol | 37.4 | 0.93 | ||
Ranitidine | 0.1 | 0.55 | ||
Sulpiride | 0.0 | 0.36 | ||
Terbutaline | 0.7 | 0.68 | ||
Theophylline | 1.8 | 0.97 | ||
Warfarin | 12.9 | 0.97 |
↵a Quoted from Zhu et al. (2002).