Parameter | Unit | cTfRMAb-TNFR |
---|---|---|
A1 | %ID/ml | 14.8 ± 1.3 |
A2 | %ID/ml | 16.1 ± 0.7 |
k1 | min−1 | 0.38 ± 0.06 |
k2 | min−1 | 0.0094 ± 0.0011 |
MRT | min | 105 ± 12 |
Vc | ml/kg | 130 ± 5 |
Vss | ml/kg | 238 ± 10 |
AUC (60 min) | %ID · min/ml | 778 ± 13 |
AUCss | %ID · min/ml | 1761 ± 144 |
CL | ml/(min · kg) | 2.3 ± 0.2 |
MRT, mean residence time; Vc, plasma volume; Vss, steady-state volume of distribution; AUC (60 min), AUC first 60 min; AUCss, steady-state AUC; CL, clearance from plasma.