Sample | Time Point | Day 1 | Day 14 | Day 34 (Recovery Phase) |
---|---|---|---|---|
h | μg Eq casopitant free base/g | |||
Plasma | 2 | 20.8 | 69.5 ± 4.1a | |
24 | 9.68 | 49.2 ± 5.0a | 11.6 | |
Blood | 2 | 11.3 | 47.4 ± 2.5a | |
24 | 9.40 | 35.3 ± 3.4a | 9.95 | |
Myocardium | 24 | N.D. | 243 | 96.2 |
Lungs | 24 | N.D. | 905 | 345 |
Kidneys | 24 | N.D. | 308 | 102 |
Liver | 24 | N.D. | 1050 | 612 |
Skeletal muscle | 24 | N.D. | 99.2 | 21.3 |
N.D., not determined.
↵a n = 4.