Glucuronide | UGT Isoform | Vmax | Km | Ksi | Vmax/Km | kcat | kcat/Km |
---|---|---|---|---|---|---|---|
pmol · min−1 · mg protein−1 | μM | μM | μl · min−1 · mg protein−1 | s−1 | M−1 · s−1 | ||
G2 | 1A1 | 664 ± 410 | 7.91 ± 5.89 | 1.54 ± 1.11 | 83.9 | 7.20 × 10−3 | 903 |
1A3 | 112 ± 27 | 7.21 ± 2.64 | 13.5 ± 5.0 | 15.5 | 1.82 × 10−3 | 252 | |
G3 | 1A1 | 146 ± 73 | 5.56 ± 3.85 | 4.67 ± 3.12 | 26.2 | 1.58 × 10−3 | 284 |
1A3 | 849 ± 485 | 17.9 ± 11.8 | 2.55 ± 1.67 | 47.5 | 1.38 × 10−2 | 774 | |
1A8 | 206 ± 88 | 6.05 ± 3.44 | 3.64 ± 2.00 | 34.0 | 1.84 × 10−3 | 303 |