Metabolites | 001F 1 h after Dose | 002F 1 h after Dose | 003F 4 h after Dose | 004F 4 h after Dose |
---|---|---|---|---|
Ticagrelor | 73.3 | 78.9 | 70.7 | 60.0 |
M5 (AR-C133913) | 13.0 | 7.8 | 1.4 | 2.8 |
M7a + M10aa | ND | ND | 2.9 | 3.6 |
M8 (AR-C124910) | 9.3 | 9.1 | 11.6 | 12.5 |
M10b | ND | ND | 3.0 | 1.9 |
M13 | ND | ND | 0.9 | 1.7 |
M14 | ND | ND | 1.2 | 0.9 |
Total radioactivityb | 95.6 | 95.8 | 91.7 | 83.4 |
ND, not detected.
a Coeluting metabolites.
b Sum of radioactivity of all integrated peaks.