TABLE 1

Kinetic data for CYP3A-catalyzed oxidation of proluciferin acetal 1 based on analysis of Fig. 3, D and L

ReactionKmkcatkcat/Km
μM
CYP3A42.88 ± 0.185.87 ± 0.142.04
CYP3A54.21 ± 0.310.94 ± 0.020.22
CYP3A78.85 ± 0.530.17 ± 0.0040.02