N+-Glucuronidation | HLMs | Recombinant UGT1A9 | ||||
---|---|---|---|---|---|---|
Km | Vmax | Vmax/Km | Km | Vmax | Vmax/Km | |
mM | pmol · min−1 · mg protein−1 | ml · min−1 · mg protein−1 | mM | pmol · min−1 · mg protein−1 | ml · min−1 · mg protein−1 | |
S-Morinidazole | 11.3 | 111 | 0.010 | 3.29 | 144 | 0.044 |
R-Morinidazole | 15.1 | 1660 | 0.110 | 2.95 | 2358 | 0.799 |