Transporter | Substrate | Jmax | Km | Transport Efficiency |
---|---|---|---|---|
pmol · min−1 · mg protein−1 | μM | μl · min−1 · mg protein−1 | ||
OAT2 | Acyclovir | 561 ± 65 | 94 ± 8 | 6 |
OAT2 | Ganciclovir | 1838 ± 374 | 264 ± 24 | 7 |
OAT2 | Penciclovir | 6675 ± 576 | 284 ± 10 | 23 |
OAT1 | PAH | 230 ± 34 | 20 ± 3 | 11 |
OAT3 | ES | 436 ± 262 | 17 ± 10 | 26 |
OCT2 | MPP | 141 ± 19 | 2.7 ± 0.2 | 52 |