Isoform | Parameters | (−)PAN | (+)PAN |
---|---|---|---|
Mean (±S.E.) | |||
rAbcg2 | TMax, nmol/h · cm2 | 2.49 ± 0.41 | 7.86 ± 2.20 |
KM, μM | 0.25 ± 0.06 | 1.85 ± 0.66 | |
r2 | 0.983 | 0.933 | |
PSAE,Eff, (μ/h)/cm2 | 9960 | 4250 | |
ABCG2 | TMax, nmol/h · cm2 | 3.29 ± 0.48 | 10.2 ± 2.43 |
KM, μM | 0.59 ± 0.12 | 5.32 ± 1.62 | |
r2 | 0.984 | 0.932 | |
PSAE,Eff, (μ/h)/cm2 | 5480 | 1920 |