Compound | CLactive | Pdiff | Kpua | fucella | Metabolism |
---|---|---|---|---|---|
μl · min−1 · 106 cells−1 | |||||
Atorvastatin | 1500 | 5.35 | 494 | 0.056 | Extensive |
Clarithromycin | 50.7 | 10.9 | 6.05 | 0.024 | Moderate |
Erythromycin | 11.4 | 12.2 | 2.00 | 0.05 | Moderate |
Fexofenadine | 167 | 6.75 | 25.5 | 0.10 | Minor |
Pitavastatin | 197 | 18.8 | 22.9 | 0.028 | Minor |
Repaglinide | 299 | 58.2 | 7.94 | 0.036 | Extensive |
Rosuvastatin | 418 | 7.08 | 58.2 | 0.48 | Minor |
Saquinavir | 239 | 191 | 2.34 | 0.0075 | Extensive |
↵a Calculated from eqs. 5 and 6.