Drug | fu,p | AUC0-∞p,u | Cmax,p,u | Tmax,p,u | AUC0-∞eECF | Cmax,ECF | Tmax,ECF |
---|---|---|---|---|---|---|---|
% | nM min | nM | min | nM min | nM | min | |
Escitalopram | 50* | 13,888 (12) | 131 (27) | 26 (29) | 11815 (10) | 62 (23) | 120 (35) |
Clozapine | 6.1 (4) | 19,732 (49) | 77 (41) | 60 (41) | 2659 (49) | 6 (33) | 240 (18) |
N-desmethylclozapine | 11 (8) | 32,296 (34) | 90 (77) | 63 (157) | 805 (55) | 2 (64) | 278 (47) |
Risperidone | 16 (7) | 24,022 (18) | 181 (32) | 53 (29) | 3543 (17) | 20 (23) | 75 (23) |
↵* Escitalopram fu,p estimate is from Bundgaard et al., 2007a.