Enzyme | Substrate | Concentration (ยตM) | Time (min) | Metabolite |
---|---|---|---|---|
CYP1A2 | Phenacetin | 50 | 15 | Acetaminophen |
CYP2C9 | Tolbutamide | 100 | 15 | 4-Hydroxytolbutamide |
CYP2C19 | S-mephenytoin | 100 | 40 | 4'-Hydroxymephenytoin |
CYP2D6 | Dextromethorphan | 5 | 15 | Dextrorphan |
CYP2E1 | Chlorzoxazone | 50 | 15 | 6-Hydroxychlorzoxazone |
CYP3A4 | Midazolam | 5 | 15 | 1-Hydroxymidazolam |
CYP, cytochrome P450.