Parameters | NBP | M2 | M3-1 | M3-2 | M5-2 |
---|---|---|---|---|---|
Cmax (ng/ml) | 514 ± 124 | 516 ± 141 | 1370 ± 750 | 1681 ± 187 | 1568 ± 108 |
Tmax (hours) | 0.75 ± 0.29 | 1.00 ± 0.00 | 0.75 ± 0.29 | 1.50 ± 0.41 | 1.00 ± 0.00 |
AUC0-t (ng·h/ml) | 831 ± 258 | 1336 ± 349 | 2478 ± 1165 | 8879 ± 2300 | 3510 ± 867 |
AUC0-∞ (ng·h/ml) | 864 ± 274 | 1370 ± 354 | 2525 ± 1164 | 8902 ± 2292 | 3529 ± 878 |
t1/2 (hours) | 5.33 ± 4.27 | 2.29 ± 0.26 | 9.09 ± 2.57 | 3.93 ± 0.31 | 3.25 ± 2.10 |
AUC, area under the curve; S.D., standard deviation.