List of transporters, specific substrates, and inhibitors for particular transporters and inhibition mechanism
| Transporter | Specific Substrate | Specific Inhibitor | Inhibition Mechanism |
|---|---|---|---|
| PEPT | Gly-Sar | H-Pro-Phe-OH | Competitive inhibition |
| OCT | MPP+ | Metformin | Competitive inhibition |
| ATB0,+ | l-Tryptophan | α-Methyl tryptophan | Specific inhibition (not a substrate) |
| MCT | Phenylacetic acid | Nicotinic acid | Competitive inhibition |
ATB0,+, neutral and basic amino acid transporter; MCT, monocarboxylate transporter; MPP+, 1-methyl-4-phenylpyridinium; OCT, organic cation transporter.