| | µM | µM | | | | |
BOC (800 mg, three times daily) | 18 ± 2.4 | 0.79 | 8.92 | 1.5 | Atorvastatin | 2.3 | Hulskotte EG et al., 2011 |
CsA (100 mg) | 0.3 ± 0.1 | 0.06 | 0.23 | 1.8 | Pitavastatin | 4.5 | Shitara and Sugiyama, 2006 |
Rifampin (600 mg) | 1.4 ± 0.2 | 0.87 | 2.47 | 2.8 | Atorvastatin | 8 | He et al., 2009 |
Lopinavir (400 mg) | 0.4 ± 0.1 | 0.3 | 0.49 | 2.4 | Rosuvastatin | 2 | Kiser et al., 2008 |
Telaprevir (750 mg) | 3.4 ± 0.1 | 1.01 | 9.84 | 3.9 | Atorvastatin | 7.9 | Lee et al., 2011 |
Amprenavir (600 mg)a | 10.0 ± 1.6 | 1.2 | 3.57 | 1.4 | Rosuvastatin | 1.1 | Karlgren et al., 2012 |
Ritonavir (100 mg, twice daily)b | 0.8 ± 0.2 | 0.03 | 0.09 | 1.1 | Rosuvastatin | No | Busti et al., 2008 |