TABLE 2

Ki values of dioscin uptake in the presence of cyclosporin A, rifampicin, EGCG, and telmisartan in OATP1B3-HEK293 cells

InhibitorKi
μM
Cyclosporin A1.43 ± 0.12
Rifampicin4.55 ± 0.78
(–)-Epigallocatechin gallate8.29 ± 0.76
Telmisartan1.03 ± 0.07
  • EGCG, (–)-Epigallocatechin gallate.