TABLE 2

Mean percentage of cumulative radioactivity recovered from six healthy male subjects after a single 1500 mg i.v. infusion dose of [14C]GSK2251052

Time PeriodUrineFecesTotal
h% dose% dose% dose
0–2451.20.151.3
0–4869.21.370.5
0–7276.94.381.2
0–9681.16.487.5
0–12083.47.390.7
0–14485.17.592.6
0–16886.47.694.0
0–19287.47.695.0
0–21688.27.695.8
0–24088.87.696.4
0–26489.37.697.0
0–28889.87.697.4
0–31290.27.697.8
0–33690.57.698.2