| mg/day | | | AUC or Cmax Ratio | µM | µM | |
Amiodaronea | 800 | 1.68 | 1.84 | 1.84 | 2.2 | 4693 | (Robinson et al., 1989) |
Amiodaronea | 400 | 1.63 | 1.72 | 1.72 | 2.5 | 2347 | (Robinson et al., 1989) |
Captopril | 37.5 | 1.39 | 1.59 | 1.59 | 0.23 | 230 | (Kirimli et al., 2001) |
Carvedilol (female) | 12.5 | 1.24 | 1 | 1.24 | 0.044 | 64 | (Baris et al., 2006) |
Carvedilol (male) | 12.5 | 1.56 | 1.38 | 1.56 | 0.044 | 64 | (Baris et al., 2006) |
Diltiazem | 90 | 1.4 | 1.38 | 1.4 | 0.489 | 1596 | (Mahgoub et al., 2002) |
Diltiazem | 180 | 1.24 | 1.24 | 1.24 | 0.196 | 798 | (Rameis et al., 1984) |
Felodipine | 2.5 | 1.43 | 1.35 | 1.43 | 0.0071 | 26 | (Rehnqvist et al., 1987) |
Felodipine | 5 | 0.76 | 1.14 | 1.14 | 0.0132 | 52 | (Rehnqvist et al., 1987) |
Felodipine | 10 | 1.18 | 1.35 | 1.35 | 0.0256 | 104 | (Rehnqvist et al., 1987) |
Felodipine | 10 | Not available | 1.18 | 1.18 | 0.0315 | 104 | (Dunselman et al., 1988) |
Isradipine | 15 | 1.11 | 1.26 | 1.26 | 0.03 | 56 | (Rodin et al., 1988) |
Mibefradilb | 150 | 1.31 | 1.41 | 1.41 | 2.77 | 1212 | (Siepmann et al., 1995) |
Nicardipine | 20 | 1.06 | 1.06 | 1.06 | 0.046 | 167 | (Lessem and Bellinetto, 1983) |
Nifedipine | 15 | 1.21 | 1.01 | 1.21 | 0.110 | 173 | (Kirch et al., 1986a) |
Nifedipine | 30 | 1.23 | 1.06 | 1.23 | 0.230 | 347 | (Kirch et al., 1986a) |
Nifedipine | 60 | 1.18 | 1.08 | 1.18 | 0.460 | 693 | (Kirch et al., 1986a) |
Nitrendipine | 20 | 1.15 | 1.57 | 1.57 | 0.115 | 222 | (Kirch et al., 1986b) |
Nitrendipine | 10 | 1.09 | 1.22 | 1.22 | 0.030 | 111 | (Kirch et al., 1986b) |
Quinidine | 600 | 1.76 | 1.75 | 1.76 | 8.83 | 8152 | (Wanwimolruk et al., 2002) |
Quinidine | 1200 | 2.65 | 2.11 | 2.65 | 11.2 | 16,305 | (Hager et al., 1979) |
Quinidine | 750 | Not available | 2.65 | 2.65 | 3.5 | 10,191 | (Belz et al., 1983) |
Ranolazine | 2000 | 1.6 | 1.46 | 1.6 | 8.4 | 18,712 | (Jerling et al., 2005) |
Sertraline | 200 | 1.1 | 1.05 | 1.1 | 0.39 | 2612 | (Rapeport et al., 1996). |
Telmisartan | 120 | 1.22 | 1.58 | 1.58 | 1.1 | 933 | (Stangier et al., 2000). |
Troglitazone | 400 | 1.04 | 1.05 | 1.05 | 3.17 | 3624 | (Loi et al., 1998) |
Verapamil | 240 | 1.51 | 1.44 | 1.51 | 1.2 | 652 | (Rodin et al., 1988) |
Verapamil | 360 | Not available | 1.61 | 1.61 | 0.0577 | 2932 | (Belz et al., 1983) |
Verapamil | 240 | Not available | 1.77 | 1.77 | 0.0332 | 1955 | (Belz et al., 1983) |
Verapamil | 240 | Not available | 1.53 | 1.53 | 0.0258 | 1955 | (Doering, 1983) |