TABLE 2

Inhibition constants for inhibition of trandolapril hydrolase activity in recombinant CES1 by diltiazem and verapamil

InhibitorKiaInhibition type
Diltiazem9.0 ± 0.5Competitive
Verapamil16.0 ± 1.1Noncompetitive
  • a Mean ± S.E.M. for two independent determinations.