Recombinant Human P450 Isoform Relative % Metabolite Formation | ||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|
Observation Time | 1A1 | 1A2 | 2A6 | 2B6 | 2C8 | 2C9 | 2C18 | 2C19 | 2D6 | 2E1 | 3A4 | 3A5 |
30 min | 4.5 | 3.4 | 1.5 | 1.5 | 1.3 | 0.9 | 1.8 | 10.6 | 4.4 | 1.3 | 29.8 | NA |
2 h | NA | 9.5 | NA | NA | NT | NT | NA | 43.9 | 8.8 | NT | 83.6 | 15.9 |
NA, not available; NT, no significant turnover detected.