Pharmacologically Active Metabolite Substrate | Km | Vmax | CLint in vitro | CLint |
---|---|---|---|---|
μM | pmol/min/mg protein | μl/min/mg protein | ml/min/kg b.wt. | |
SS form | ||||
Rat | 32.58 | 734.80 | 22.55 | 40.41 |
Dog | 155.24 | 722.79 | 4.66 | 11.62 |
Human | 26.29 | 362.01 | 13.77 | 17.28 |
SR form | ||||
Rat | 79.34 | 1665.74 | 20.99 | 37.61 |
Dog | 208.04 | 205.30 | 0.99 | 2.47 |
Human | 17.26 | 243.50 | 14.11 | 17.71 |