Tedizolid Phosphate 10 mg/kg Administered Intravenously | Tedizolid Phosphate 25 mg/kg Administered Orally | |||||||
---|---|---|---|---|---|---|---|---|
Rat | Dog | Rat | Dog | |||||
Male | Female | Male | Female | Male | Female | Male | Female | |
% | ||||||||
Desmethyl tedizolid | — | — | 2.3 | 1.3 | — | — | 2.5 | 3.4 |
Tedizolid sulfate | 100 | 87.1 | 91.3 | 97.5 | 100 | 91 | 94.7 | 77.1 |
Tedizolid | — | 12.9 | 6.4 | 1.2 | — | 9 | 2.8 | 18.8 |