TABLE 2

Protein expression levels of uptake transporters in human liver membrane fractions

TransporternProtein Expression Level
Mean ± S.D.MedianMinMaxMax/Min
fmol µg membrane protein−1
NTCP121.8 ± 1.01.50.53.97.5
OATP1B11223.2 ± 9.419.612.144.43.7
OATP1B3123.2 ± 1.93.80.26.032.0
OATP2B1121.6 ± 1.11.20.64.37.5
  • Max, maximum; Max/Min, fold range in expression; Min, minimum.