Compound | CL | Vss | ||||||||
---|---|---|---|---|---|---|---|---|---|---|
1.25-fold | 1.5-fold | 2-fold | 2.5-fold | 3-fold | 1.25-fold | 1.5-fold | 2-fold | 2.5-fold | 3-fold | |
Talinolol | 24 | 4 | 0 | 0 | 0 | NA | NA | NA | NA | NA |
Propranolol | 53 | 29 | 6 | 1 | 0 | NA | NA | NA | NA | NA |
Cisatracurium | 36 | 8 | 0 | 0 | 0 | NA | NA | NA | NA | NA |
Acetaminophen | 10 | 0 | 0 | 0 | 0 | 7 | 0 | 0 | 0 | 0 |
Lidocaine | 48 | 20 | 2 | 0 | 0 | 54 | 22 | 2 | 0 | 0 |
Propofol | 56 | 35 | 13 | 4 | 0 | NA | NA | NA | NA | NA |
Metronidazole | 50 | 27 | 5 | 1 | 1 | 22 | 3 | 0 | 0 | 0 |
Theophylline | 44 | 19 | 2 | 0 | 0 | NA | NA | NA | NA | NA |
Ciprofloxacin | 43 | 17 | 3 | 1 | 0 | 21 | 3 | 0 | 0 | 0 |
Midazolam | 56 | 32 | 11 | 4 | 2 | 73 | 48 | 22 | 11 | 5 |
Antipyrine | 54 | 26 | 2 | 0 | 0 | 18 | 0 | 0 | 0 | 0 |
Digoxin | 63 | 37 | 18 | 8 | 5 | 56 | 28 | 13 | 0 | 0 |
Furosemide | 55 | 28 | 6 | 1 | 0 | 51 | 33 | 0 | 0 | 0 |
Lorazepam | 59 | 36 | 10 | 3 | 1 | 13 | 0 | 0 | 0 | 0 |
Diazepam | 56 | 30 | 5 | 1 | 0 | 45 | 15 | 2 | 0 | 0 |
Thiopental | 34 | 7 | 0 | 0 | 0 | 50 | 26 | 4 | 0 | 0 |
Alfentanil | 68 | 45 | 16 | 8 | 3 | NA | NA | NA | NA | NA |
NA, not applicable (data were not available).