Inhibitor | AUC0–t | AUC0–∞ | CLt | Vd | Kp,liver | |
---|---|---|---|---|---|---|
Compound | Dose | |||||
mg/kg | ng·h/ml | ng·h/ml | ml/h/kg | ml/kg | 1 hour | |
— | — | 2013 ± 482 | 2025 ± 547 | 266 ± 90 | 359 ± 94 | 18 ± 10 |
Rifampicin | 20 | 16,686 ± 330 | 16,781 ± 350 | 29.8 ± 0.6 | 96.8 ± 2.5 | 0.44 ± 0.07 |
Rifampicin | 80 | 27,428 ± 6358 | 28,208 ± 6952 | 18.6 ± 5.2 | 104 ± 11 | 0.42 ± 0.06 |