Species | System | Transporter | Substrate | IC50 (μM) |
---|---|---|---|---|
Rat | Hepatocytes | Ntcp | d8-TCA | 10.9 ± 0.7 |
Hepatocytes | Oatps | d8-TCA | 2.94 ± 0.34 | |
Human | HEK293 cells | OATP1B1 | Atorvastatin | 2.28 ± 0.17 |
HEK293 cells | OATP1B3 | Atorvastatin | 3.98 ± 0.26 | |
MDCK cells | MRP2 | Vinblastine | 2.41 ± 0.50 |