TABLE 5

Summary of the transporters involved in the drug canalicular efflux

DrugTransportersReferences
AzithromycinPgP (+++)Sugie et al., 2004
MRP2 (++)
CeftriaxoneMRP2 (+++)Kato et al., 2008
BCRP (++)
DigoxinPgP (+++)Greiner et al., 1999
BuprenorphinePgP (+/−)Hassan et al., 2009
BCRP (–)Tournier et al., 2010
MRP2 (?)