IC50 Value for Thiamine Uptake | |||
---|---|---|---|
Compound | Caco-2 | THTR-1 | THTR-2 |
µM | µM | µM | |
Fedratinib | 0.940 ± 0.080 | 7.10 ± 1.26 | 1.36 ± 0.59 |
AZD1480 | 183 ± 68.9 | 22.2 ± 6.20 | 15.3 ± 2.90 |
Cerdulatinib | >300 | 276 ± 117 | >300 |
Momelotinib | >30.0 | >30.0 | >30.0 |
Trimethoprim | 154 ± 22.4 | 6.84 ± 1.68 | 5.56 ± 0.65 |
Oxythiamine | 198 ± 16.0 | 67.3 ± 7.50 | 66.4 ± 21.4 |
Amprolium | 9.40 ± 2.80 | 2.60 ± 0.93 | 0.620 ± 0.270 |