Substrate | Km (mM) | vmax (nmol·min−1·mg protein−1) | |
---|---|---|---|
vorinostat | mARC1 | 1.45 ± 0.37 | 46.3 ± 5.5 |
mARC2 | 2.73 ± 0.18 | 19.3 ± 0.8 | |
benzhydroxamic acid | mARC1 | 0.31 ± 0.11 | 73.7 ± 7.0 |
mARC2 | 2.12 ± 0.28 | 313.5 ± 22.5 | |
bufexamac | mARC1 | 1.09 ± 0.15 | 13.4 ± 1.1 |
mARC2 | 1.07 ± 0.15 | 8.2 ± 0.7 | |
CP544439 | mARC1 | 0.25 ± 0.06 | 50.2 ± 4.4 |
mARC2 | −/− | −/−a | |
N-hydroxyphenacetin | mARC1 | −/− | −/−b |
mARC2 | −/− | −/−b | |
benzamidoxime | mARC1 | 0.63 ± 0.06 | 674.8 ± 25.1 |
mARC2 | 0.54 ± 0.03 | 549.6 ± 12.1 |