Substrate Concentration (µM) | Marker Metabolite | Total Metabolite Formation (pmol per Million Hepatocytes) | |||
---|---|---|---|---|---|
CCHH | MMHH | ||||
Average | S.D. | Average | S.D. | ||
mM | |||||
100 | Acetaminophen Glutathione | 206.50 | 3.91 | 856.72 | 71.28 |
200 | Acetaminophen Glutathione | 99.81 | 7.49 | 676.70 | 54.43 |
100 | Acetaminophen Glucuronide | 572.55 | 27.12 | 1298.77 | 64.29 |
200 | Acetaminophen Glucuronide | 170.28 | 16.38 | 1361.84 | 83.36 |
100 | Acetaminophen Sulfate | 105.55 | 3.36 | 150.22 | 6.68 |
200 | Acetaminophen Sulfate | 52.58 | 1.40 | 156.36 | 11.86 |