TABLE 4

Efflux ratio values for select control compounds

CompoundMDR1 ERmBCRP ER
Prazosin21.150.8
Quinidine78.23.0
Triprolidine3.32.2
Metoprolol2.51.2
Fleroxacin3.56.4
Pitavastatin16.380.5
  • ER, efflux ratio; mBCRP, murine breast cancer resistance protein; MDR1, multidrug resistance protein 1.