VPA-985, a nonpeptide orally active and selective vasopressin V2 receptor antagonist

Adv Exp Med Biol. 1998:449:439-43. doi: 10.1007/978-1-4615-4871-3_55.
No abstract available

Publication types

  • Review

MeSH terms

  • Animals
  • Antidiuretic Hormone Receptor Antagonists
  • Arginine Vasopressin / antagonists & inhibitors*
  • Azepines / pharmacology*
  • Benzamides / pharmacology*
  • Blood Pressure / drug effects
  • Cyclic AMP / metabolism
  • Dogs
  • Heart Failure / physiopathology
  • Humans
  • Hyponatremia / etiology
  • Hyponatremia / physiopathology
  • Inappropriate ADH Syndrome / physiopathology
  • Kidney / drug effects
  • Kidney / physiology
  • Kidney / physiopathology
  • Pyrroles
  • Receptors, Vasopressin / metabolism*

Substances

  • Antidiuretic Hormone Receptor Antagonists
  • Azepines
  • Benzamides
  • Pyrroles
  • Receptors, Vasopressin
  • Arginine Vasopressin
  • lixivaptan
  • Cyclic AMP