Bufuralol, dextromethorphan, and debrisoquine as prototype substrates for human P450IID6

Methods Enzymol. 1991:206:509-17. doi: 10.1016/0076-6879(91)06120-r.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adrenergic beta-Antagonists / metabolism*
  • Chromatography, High Pressure Liquid / methods
  • Cytochrome P-450 CYP2D6
  • Cytochrome P-450 Enzyme System / metabolism*
  • Debrisoquin / metabolism*
  • Dextromethorphan / metabolism*
  • Ethanolamines / metabolism*
  • Humans
  • Microsomes, Liver / enzymology*
  • Mixed Function Oxygenases / metabolism*
  • Spectrometry, Fluorescence / methods
  • Substrate Specificity

Substances

  • Adrenergic beta-Antagonists
  • Ethanolamines
  • Dextromethorphan
  • bufuralol
  • Cytochrome P-450 Enzyme System
  • Mixed Function Oxygenases
  • Cytochrome P-450 CYP2D6
  • Debrisoquin