Gefitinib concentrations in human glioblastoma tissue

J Neurooncol. 2007 Apr;82(2):175-6. doi: 10.1007/s11060-006-9257-3. Epub 2006 Sep 29.
No abstract available

MeSH terms

  • Antineoplastic Agents / pharmacokinetics*
  • Biological Availability
  • Brain Neoplasms / drug therapy
  • Brain Neoplasms / metabolism*
  • Chromatography, High Pressure Liquid
  • Cytochrome P-450 CYP3A
  • Cytochrome P-450 Enzyme System / metabolism
  • ErbB Receptors / antagonists & inhibitors
  • Gefitinib
  • Glioblastoma / drug therapy
  • Glioblastoma / metabolism*
  • Humans
  • Quinazolines / pharmacokinetics*

Substances

  • Antineoplastic Agents
  • Quinazolines
  • Cytochrome P-450 Enzyme System
  • Cytochrome P-450 CYP3A
  • CYP3A4 protein, human
  • ErbB Receptors
  • Gefitinib