Mitigating heterocycle metabolism in drug discovery

J Med Chem. 2012 Jul 12;55(13):6002-20. doi: 10.1021/jm300343m. Epub 2012 May 7.
No abstract available

Publication types

  • Review

MeSH terms

  • Animals
  • Biotransformation
  • Databases, Factual
  • Drug Discovery / methods*
  • Drug Interactions
  • Heterocyclic Compounds, 1-Ring / chemistry
  • Heterocyclic Compounds, 1-Ring / metabolism*
  • Heterocyclic Compounds, 4 or More Rings / chemistry
  • Heterocyclic Compounds, 4 or More Rings / metabolism*
  • Humans
  • Mice
  • Pharmaceutical Preparations / chemistry
  • Pharmaceutical Preparations / metabolism*
  • Rats

Substances

  • Heterocyclic Compounds, 1-Ring
  • Heterocyclic Compounds, 4 or More Rings
  • Pharmaceutical Preparations