Metabolic pathway of paroxetine in animals and man and the comparative pharmacological properties of its metabolites

Acta Psychiatr Scand Suppl. 1989:350:24-6. doi: 10.1111/j.1600-0447.1989.tb07163.x.
No abstract available

MeSH terms

  • Animals
  • Antidepressive Agents / pharmacokinetics*
  • Antidepressive Agents / pharmacology
  • Biotransformation
  • Brain / drug effects
  • Chemical Phenomena
  • Chemistry
  • Humans
  • Hypothalamus / drug effects
  • Mice
  • Paroxetine
  • Piperidines / pharmacokinetics*
  • Rats
  • Receptors, Serotonin / drug effects
  • Serotonin Antagonists / pharmacokinetics*
  • Serotonin Antagonists / pharmacology
  • Structure-Activity Relationship
  • Synaptosomes / drug effects

Substances

  • Antidepressive Agents
  • Piperidines
  • Receptors, Serotonin
  • Serotonin Antagonists
  • Paroxetine