Mephenytoin hydroxylase activity in human liver: inhibition by steroids

Drug Metab Dispos. 1985 Nov-Dec;13(6):746-9.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aryl Hydrocarbon Hydroxylases*
  • Cytochrome P-450 CYP2C19
  • Cytochrome P-450 Enzyme System / metabolism
  • Humans
  • Hydantoins / metabolism*
  • In Vitro Techniques
  • Kinetics
  • Liver / enzymology*
  • Mephenytoin / metabolism*
  • Microsomes, Liver / metabolism
  • Mixed Function Oxygenases / antagonists & inhibitors*
  • Mixed Function Oxygenases / metabolism
  • Steroids / pharmacology*

Substances

  • Hydantoins
  • Steroids
  • Cytochrome P-450 Enzyme System
  • Mixed Function Oxygenases
  • Aryl Hydrocarbon Hydroxylases
  • CYP2C19 protein, human
  • Cytochrome P-450 CYP2C19
  • Mephenytoin