Determination of biological activity of alprazolam, triazolam and their metabolites

J Pharm Pharmacol. 1982 Feb;34(2):115-6. doi: 10.1111/j.2042-7158.1982.tb04197.x.
No abstract available

MeSH terms

  • Alprazolam
  • Animals
  • Anti-Anxiety Agents / metabolism*
  • Benzodiazepines / metabolism*
  • Binding, Competitive
  • Brain / metabolism
  • Diazepam / pharmacology
  • Flunitrazepam / metabolism
  • Kinetics
  • Male
  • Membranes / metabolism
  • Rats
  • Rats, Inbred Strains
  • Receptors, Drug / metabolism*
  • Receptors, GABA-A
  • Triazolam / metabolism*

Substances

  • Anti-Anxiety Agents
  • Receptors, Drug
  • Receptors, GABA-A
  • Benzodiazepines
  • Triazolam
  • Flunitrazepam
  • Diazepam
  • Alprazolam