Inhibition of uridinediphosphate glucuronyltransferase caused by furosemide

Experientia. 1980 Jul 15;36(7):861-3. doi: 10.1007/BF01978616.

Abstract

The diuretic agent, furosemide, inhibits liver microsomal uridinediphosphate glucuronyltransferase (EC. 2.4.1.17), in monkey and rat. Inhibition is of the non-competitive type.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Furosemide / pharmacology*
  • Glucuronosyltransferase / antagonists & inhibitors*
  • Guinea Pigs
  • Haplorhini
  • Kinetics
  • Macaca mulatta
  • Microsomes, Liver / enzymology*
  • Rats
  • Species Specificity

Substances

  • Furosemide
  • Glucuronosyltransferase