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Research ArticleArticle

Effect of Inhibitor Depletion on Inhibitory Potency: Tight Binding Inhibition of CYP3A by Clotrimazole

Megan A. Gibbs, Kent L. Kunze, William N. Howald and Kenneth E. Thummel
Drug Metabolism and Disposition May 1999, 27 (5) 596-599;
Megan A. Gibbs
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Kent L. Kunze
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William N. Howald
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Kenneth E. Thummel
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Article Information

vol. 27 no. 5 596-599
PubMed 
10220488

Published By 
American Society for Pharmacology and Experimental Therapeutics
Print ISSN 
0090-9556
Online ISSN 
1521-009X
History 
  • Received October 6, 1998
  • Accepted January 19, 1999
  • Published online May 1, 1999.

Copyright & Usage 
The American Society for Pharmacology and Experimental Therapeutics

Author Information

  1. Megan A. Gibbs2,
  2. Kent L. Kunze1,
  3. William N. Howald1 and
  4. Kenneth E. Thummel2
  1. Departments of 1Medicinal Chemistry (K.L.K., W.N.H.) and 2Pharmaceutics (M.A.G., K.E.T.), School of Pharmacy, University of Washington, Seattle, Washington
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    Drug Metabolism and Disposition: 27 (5)
    Drug Metabolism and Disposition
    Vol. 27, Issue 5
    1 May 1999
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    Research ArticleArticle

    Effect of Inhibitor Depletion on Inhibitory Potency: Tight Binding Inhibition of CYP3A by Clotrimazole

    Megan A. Gibbs, Kent L. Kunze, William N. Howald and Kenneth E. Thummel
    Drug Metabolism and Disposition May 1, 1999, 27 (5) 596-599;

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    Research ArticleArticle

    Effect of Inhibitor Depletion on Inhibitory Potency: Tight Binding Inhibition of CYP3A by Clotrimazole

    Megan A. Gibbs, Kent L. Kunze, William N. Howald and Kenneth E. Thummel
    Drug Metabolism and Disposition May 1, 1999, 27 (5) 596-599;
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