Index by author
December 01, 2002; Volume 30,Issue 12
A
Austin, Rupert P.
- You have accessThe Influence of Nonspecific Microsomal Binding on Apparent Intrinsic Clearance, and Its Prediction from Physicochemical PropertiesRupert P. Austin, Patrick Barton, Scott L. Cockroft, Mark C. Wenlock and Robert J. RileyDrug Metabolism and Disposition December 2002, 30 (12) 1497-1503; DOI: https://doi.org/10.1124/dmd.30.12.1497
Awasthi, Sanjay
- You have accessRLIP76, a Novel Transporter Catalyzing ATP-Dependent Efflux of XenobioticsSanjay Awasthi, Rajendra Sharma, Sharad S. Singhal, Piotr Zimniak and Yogesh C. AwasthiDrug Metabolism and Disposition December 2002, 30 (12) 1300-1310; DOI: https://doi.org/10.1124/dmd.30.12.1300
Awasthi, Yogesh C.
- You have accessRLIP76, a Novel Transporter Catalyzing ATP-Dependent Efflux of XenobioticsSanjay Awasthi, Rajendra Sharma, Sharad S. Singhal, Piotr Zimniak and Yogesh C. AwasthiDrug Metabolism and Disposition December 2002, 30 (12) 1300-1310; DOI: https://doi.org/10.1124/dmd.30.12.1300
B
Backman, Janne T.
- You have accessGemfibrozil Inhibits CYP2C8-Mediated Cerivastatin Metabolism in Human Liver MicrosomesJun-Sheng Wang, Mikko Neuvonen, Xia Wen, Janne T. Backman and Pertti J. NeuvonenDrug Metabolism and Disposition December 2002, 30 (12) 1352-1356; DOI: https://doi.org/10.1124/dmd.30.12.1352
Bailey, Nigel J.C.
- You have accessApplication of Directly Coupled High Performance Liquid Chromatography-NMR-Mass Spectometry and 1H NMR Spectroscopic Studies to the Investigation of 2,3-Benzofuran Metabolism in Sprague-Dawley RatsJohn C. Connelly, Susan C. Connor, Soria Monte, Nigel J.C. Bailey, Nathan Borgeaud, Elaine Holmes, Jeff Troke, Jeremy K. Nicholson and Claire L. GavaghanDrug Metabolism and Disposition December 2002, 30 (12) 1357-1363; DOI: https://doi.org/10.1124/dmd.30.12.1357
Barton, Patrick
- You have accessThe Influence of Nonspecific Microsomal Binding on Apparent Intrinsic Clearance, and Its Prediction from Physicochemical PropertiesRupert P. Austin, Patrick Barton, Scott L. Cockroft, Mark C. Wenlock and Robert J. RileyDrug Metabolism and Disposition December 2002, 30 (12) 1497-1503; DOI: https://doi.org/10.1124/dmd.30.12.1497
Berry, Loren M.
- You have accessInvolvement of CYP3A in the Metabolism of Eplerenone in Humans and Dogs: Differential Metabolism by CYP3A4 and CYP3A5Chyung S. Cook, Loren M. Berry, David H. Kim, Earl G. Burton, Jeremy D. Hribar and Liming ZhangDrug Metabolism and Disposition December 2002, 30 (12) 1344-1351; DOI: https://doi.org/10.1124/dmd.30.12.1344
Beydon, Dominique
- You have accessToxicokinetics and Metabolism ofN-[14C]Methylpyrrolidone in Male Sprague-Dawley Rats. A Saturable NMP Elimination ProcessJean-Paul Payan, Dominique Beydon, Jean-Paul Fabry, Isabelle Boudry, Benoit Cossec and Elisabeth FerrariDrug Metabolism and Disposition December 2002, 30 (12) 1418-1424; DOI: https://doi.org/10.1124/dmd.30.12.1418
Bhathena, Anahita
- You have accessSuppression of Cytochrome P450 2C11 by Aromatic Hydrocarbons: Mechanistic Insights from Studies of the 5′-Flanking Region of theCYP2C11 GeneAnahita Bhathena, Chunja Lee and David S. RiddickDrug Metabolism and Disposition December 2002, 30 (12) 1385-1392; DOI: https://doi.org/10.1124/dmd.30.12.1385
Blaschke, Terrence F.
- You have accessModel-based Analysis of the Pharmacokinetic Interactions Between Ritonavir, Nelfinavir, and Saquinavir after Simultaneous and Staggered Oral AdministrationJian-Feng Lu, Terrence F. Blaschke, Charles Flexner, Susan L. Rosenkranz, Lewis B. Sheiner and AIDS Clinical Trials Group Protocol 378 InvestigatorsDrug Metabolism and Disposition December 2002, 30 (12) 1455-1461; DOI: https://doi.org/10.1124/dmd.30.12.1455
Bonner, Heather S.
- You have accessRegional Pharmacokinetics of Amifostine in Anesthetized Dogs: Role of the Liver, Gastrointestinal Tract, Lungs, and KidneysMicha Levi, James A. Knol, William D. Ensminger, Susan J. DeRemer, Chunzhi Dou, Susan M. Lunte, Heather S. Bonner, Leslie M. Shaw and David E. SmithDrug Metabolism and Disposition December 2002, 30 (12) 1425-1430; DOI: https://doi.org/10.1124/dmd.30.12.1425
Borgeaud, Nathan
- You have accessApplication of Directly Coupled High Performance Liquid Chromatography-NMR-Mass Spectometry and 1H NMR Spectroscopic Studies to the Investigation of 2,3-Benzofuran Metabolism in Sprague-Dawley RatsJohn C. Connelly, Susan C. Connor, Soria Monte, Nigel J.C. Bailey, Nathan Borgeaud, Elaine Holmes, Jeff Troke, Jeremy K. Nicholson and Claire L. GavaghanDrug Metabolism and Disposition December 2002, 30 (12) 1357-1363; DOI: https://doi.org/10.1124/dmd.30.12.1357
Boudry, Isabelle
- You have accessToxicokinetics and Metabolism ofN-[14C]Methylpyrrolidone in Male Sprague-Dawley Rats. A Saturable NMP Elimination ProcessJean-Paul Payan, Dominique Beydon, Jean-Paul Fabry, Isabelle Boudry, Benoit Cossec and Elisabeth FerrariDrug Metabolism and Disposition December 2002, 30 (12) 1418-1424; DOI: https://doi.org/10.1124/dmd.30.12.1418
Buhler, Donald R.
- You have accessFunctional Properties of a Rainbow Trout CYP3A27 Expressed by Recombinant Baculovirus in Insect CellsSu-Jun Lee and Donald R. BuhlerDrug Metabolism and Disposition December 2002, 30 (12) 1406-1412; DOI: https://doi.org/10.1124/dmd.30.12.1406
Burton, Earl G.
- You have accessInvolvement of CYP3A in the Metabolism of Eplerenone in Humans and Dogs: Differential Metabolism by CYP3A4 and CYP3A5Chyung S. Cook, Loren M. Berry, David H. Kim, Earl G. Burton, Jeremy D. Hribar and Liming ZhangDrug Metabolism and Disposition December 2002, 30 (12) 1344-1351; DOI: https://doi.org/10.1124/dmd.30.12.1344
C
Cai, Hongbo
- You have accessRegulation of CYP2B6 and CYP3A Expression by Hydroxymethylglutaryl Coenzyme A Inhibitors in Primary Cultured Human HepatocytesThomas A. Kocarek, Michael S. Dahn, Hongbo Cai, Stephen C. Strom and Nancy A. Mercer-HainesDrug Metabolism and Disposition December 2002, 30 (12) 1400-1405; DOI: https://doi.org/10.1124/dmd.30.12.1400
Carter, K. M.
- You have accessIrreversible Inhibition of CYP2D6 by (−)-Chloroephedrine, a Possible Impurity in MethamphetamineB. Rege, K. M. Carter, M. A. Sarkar, G. E. Kellogg and W. H. SoineDrug Metabolism and Disposition December 2002, 30 (12) 1337-1343; DOI: https://doi.org/10.1124/dmd.30.12.1337
Chen, Chun-Lin
- You have accessMetabolism of Stavudine-5′-[p-Bromophenyl Methoxyalaninyl Phosphate], Stampidine, in Mice, Dogs, and CatsChun-Lin Chen, Gengli Yu, T. K. Venkatachalam and Fatih M. UckunDrug Metabolism and Disposition December 2002, 30 (12) 1523-1531; DOI: https://doi.org/10.1124/dmd.30.12.1523
Cheng, K.-C.
- You have accessDevelopment of a Novel in Vitro Model to Predict Hepatic Clearance Using Fresh, Cryopreserved, and Sandwich-Cultured HepatocytesYau Yi Lau, Elpida Sapidou, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition December 2002, 30 (12) 1446-1454; DOI: https://doi.org/10.1124/dmd.30.12.1446
Clarke, Stephen E.
- You have accessQuinidine and Haloperidol as Modifiers of CYP3A4 Activity: Multisite Kinetic Model ApproachAleksandra Galetin, Stephen E. Clarke and J. Brian HoustonDrug Metabolism and Disposition December 2002, 30 (12) 1512-1522; DOI: https://doi.org/10.1124/dmd.30.12.1512
Cockroft, Scott L.
- You have accessThe Influence of Nonspecific Microsomal Binding on Apparent Intrinsic Clearance, and Its Prediction from Physicochemical PropertiesRupert P. Austin, Patrick Barton, Scott L. Cockroft, Mark C. Wenlock and Robert J. RileyDrug Metabolism and Disposition December 2002, 30 (12) 1497-1503; DOI: https://doi.org/10.1124/dmd.30.12.1497
Connelly, John C.
- You have accessApplication of Directly Coupled High Performance Liquid Chromatography-NMR-Mass Spectometry and 1H NMR Spectroscopic Studies to the Investigation of 2,3-Benzofuran Metabolism in Sprague-Dawley RatsJohn C. Connelly, Susan C. Connor, Soria Monte, Nigel J.C. Bailey, Nathan Borgeaud, Elaine Holmes, Jeff Troke, Jeremy K. Nicholson and Claire L. GavaghanDrug Metabolism and Disposition December 2002, 30 (12) 1357-1363; DOI: https://doi.org/10.1124/dmd.30.12.1357
Connor, Susan C.
- You have accessApplication of Directly Coupled High Performance Liquid Chromatography-NMR-Mass Spectometry and 1H NMR Spectroscopic Studies to the Investigation of 2,3-Benzofuran Metabolism in Sprague-Dawley RatsJohn C. Connelly, Susan C. Connor, Soria Monte, Nigel J.C. Bailey, Nathan Borgeaud, Elaine Holmes, Jeff Troke, Jeremy K. Nicholson and Claire L. GavaghanDrug Metabolism and Disposition December 2002, 30 (12) 1357-1363; DOI: https://doi.org/10.1124/dmd.30.12.1357
Cook, Chyung S.
- You have accessInvolvement of CYP3A in the Metabolism of Eplerenone in Humans and Dogs: Differential Metabolism by CYP3A4 and CYP3A5Chyung S. Cook, Loren M. Berry, David H. Kim, Earl G. Burton, Jeremy D. Hribar and Liming ZhangDrug Metabolism and Disposition December 2002, 30 (12) 1344-1351; DOI: https://doi.org/10.1124/dmd.30.12.1344
Cook, James M.
- You have accessEnzyme Kinetics for the Formation of 3-Hydroxyquinine and Three New Metabolites of Quinine in Vitro; 3-Hydroxylation by CYP3A4 is Indeed the Major Metabolic PathwayRajaa A. Mirghani, Ümit Yasar, Tao Zheng, James M. Cook, Lars L. Gustafsson, Gunnel Tybring and Örjan EricssonDrug Metabolism and Disposition December 2002, 30 (12) 1368-1371; DOI: https://doi.org/10.1124/dmd.30.12.1368
Cossec, Benoit
- You have accessToxicokinetics and Metabolism ofN-[14C]Methylpyrrolidone in Male Sprague-Dawley Rats. A Saturable NMP Elimination ProcessJean-Paul Payan, Dominique Beydon, Jean-Paul Fabry, Isabelle Boudry, Benoit Cossec and Elisabeth FerrariDrug Metabolism and Disposition December 2002, 30 (12) 1418-1424; DOI: https://doi.org/10.1124/dmd.30.12.1418
Cui, Xiaoming
- You have accessDevelopment of a Novel in Vitro Model to Predict Hepatic Clearance Using Fresh, Cryopreserved, and Sandwich-Cultured HepatocytesYau Yi Lau, Elpida Sapidou, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition December 2002, 30 (12) 1446-1454; DOI: https://doi.org/10.1124/dmd.30.12.1446
D
Dabrowiak, James C.
- You have accessKinetic Study of the Reaction of Cisplatin with ThiolsJames C. Dabrowiak, Jerry Goodisman and Abdul-Kader SouidDrug Metabolism and Disposition December 2002, 30 (12) 1378-1384; DOI: https://doi.org/10.1124/dmd.30.12.1378
Dahn, Michael S.
- You have accessRegulation of CYP2B6 and CYP3A Expression by Hydroxymethylglutaryl Coenzyme A Inhibitors in Primary Cultured Human HepatocytesThomas A. Kocarek, Michael S. Dahn, Hongbo Cai, Stephen C. Strom and Nancy A. Mercer-HainesDrug Metabolism and Disposition December 2002, 30 (12) 1400-1405; DOI: https://doi.org/10.1124/dmd.30.12.1400
Davidson, Jeffrey N.
- You have accessDihydroorotase Catalyzes the Ring Opening of the Hydrolysis Intermediates of the Cardioprotective Drug Dexrazoxane (ICRF-187)Patricia E. Schroeder, Jeffrey N. Davidson and Brian B. HasinoffDrug Metabolism and Disposition December 2002, 30 (12) 1431-1435; DOI: https://doi.org/10.1124/dmd.30.12.1431
DeRemer, Susan J.
- You have accessRegional Pharmacokinetics of Amifostine in Anesthetized Dogs: Role of the Liver, Gastrointestinal Tract, Lungs, and KidneysMicha Levi, James A. Knol, William D. Ensminger, Susan J. DeRemer, Chunzhi Dou, Susan M. Lunte, Heather S. Bonner, Leslie M. Shaw and David E. SmithDrug Metabolism and Disposition December 2002, 30 (12) 1425-1430; DOI: https://doi.org/10.1124/dmd.30.12.1425
Dou, Chunzhi
- You have accessRegional Pharmacokinetics of Amifostine in Anesthetized Dogs: Role of the Liver, Gastrointestinal Tract, Lungs, and KidneysMicha Levi, James A. Knol, William D. Ensminger, Susan J. DeRemer, Chunzhi Dou, Susan M. Lunte, Heather S. Bonner, Leslie M. Shaw and David E. SmithDrug Metabolism and Disposition December 2002, 30 (12) 1425-1430; DOI: https://doi.org/10.1124/dmd.30.12.1425
E
Elaut, G.
- You have accessMajor Phase I Biotransformation Pathways of Trichostatin A in Rat Hepatocytes and in Rat and Human Liver MicrosomesG. Elaut, G. Török, M. Vinken, G. Laus, P. Papeleu, D. Tourwe and V. RogiersDrug Metabolism and Disposition December 2002, 30 (12) 1320-1328; DOI: https://doi.org/10.1124/dmd.30.12.1320
Ensminger, William D.
- You have accessRegional Pharmacokinetics of Amifostine in Anesthetized Dogs: Role of the Liver, Gastrointestinal Tract, Lungs, and KidneysMicha Levi, James A. Knol, William D. Ensminger, Susan J. DeRemer, Chunzhi Dou, Susan M. Lunte, Heather S. Bonner, Leslie M. Shaw and David E. SmithDrug Metabolism and Disposition December 2002, 30 (12) 1425-1430; DOI: https://doi.org/10.1124/dmd.30.12.1425
Ericsson, Örjan
- You have accessEnzyme Kinetics for the Formation of 3-Hydroxyquinine and Three New Metabolites of Quinine in Vitro; 3-Hydroxylation by CYP3A4 is Indeed the Major Metabolic PathwayRajaa A. Mirghani, Ümit Yasar, Tao Zheng, James M. Cook, Lars L. Gustafsson, Gunnel Tybring and Örjan EricssonDrug Metabolism and Disposition December 2002, 30 (12) 1368-1371; DOI: https://doi.org/10.1124/dmd.30.12.1368
F
Fabry, Jean-Paul
- You have accessToxicokinetics and Metabolism ofN-[14C]Methylpyrrolidone in Male Sprague-Dawley Rats. A Saturable NMP Elimination ProcessJean-Paul Payan, Dominique Beydon, Jean-Paul Fabry, Isabelle Boudry, Benoit Cossec and Elisabeth FerrariDrug Metabolism and Disposition December 2002, 30 (12) 1418-1424; DOI: https://doi.org/10.1124/dmd.30.12.1418
Ferrari, Elisabeth
- You have accessToxicokinetics and Metabolism ofN-[14C]Methylpyrrolidone in Male Sprague-Dawley Rats. A Saturable NMP Elimination ProcessJean-Paul Payan, Dominique Beydon, Jean-Paul Fabry, Isabelle Boudry, Benoit Cossec and Elisabeth FerrariDrug Metabolism and Disposition December 2002, 30 (12) 1418-1424; DOI: https://doi.org/10.1124/dmd.30.12.1418
Flexner, Charles
- You have accessModel-based Analysis of the Pharmacokinetic Interactions Between Ritonavir, Nelfinavir, and Saquinavir after Simultaneous and Staggered Oral AdministrationJian-Feng Lu, Terrence F. Blaschke, Charles Flexner, Susan L. Rosenkranz, Lewis B. Sheiner and AIDS Clinical Trials Group Protocol 378 InvestigatorsDrug Metabolism and Disposition December 2002, 30 (12) 1455-1461; DOI: https://doi.org/10.1124/dmd.30.12.1455
Fuse, Eiichi
- You have accessEffects of Olopatadine, a New Antiallergic Agent, on Human Liver Microsomal Cytochrome P450 ActivitiesJiro Kajita, Keiko Inano, Eiichi Fuse, Takashi Kuwabara and Hiroyuki KobayashiDrug Metabolism and Disposition December 2002, 30 (12) 1504-1511; DOI: https://doi.org/10.1124/dmd.30.12.1504
G
Galetin, Aleksandra
- You have accessQuinidine and Haloperidol as Modifiers of CYP3A4 Activity: Multisite Kinetic Model ApproachAleksandra Galetin, Stephen E. Clarke and J. Brian HoustonDrug Metabolism and Disposition December 2002, 30 (12) 1512-1522; DOI: https://doi.org/10.1124/dmd.30.12.1512
Gavaghan, Claire L.
- You have accessApplication of Directly Coupled High Performance Liquid Chromatography-NMR-Mass Spectometry and 1H NMR Spectroscopic Studies to the Investigation of 2,3-Benzofuran Metabolism in Sprague-Dawley RatsJohn C. Connelly, Susan C. Connor, Soria Monte, Nigel J.C. Bailey, Nathan Borgeaud, Elaine Holmes, Jeff Troke, Jeremy K. Nicholson and Claire L. GavaghanDrug Metabolism and Disposition December 2002, 30 (12) 1357-1363; DOI: https://doi.org/10.1124/dmd.30.12.1357
Ghosheh, Omar
- You have accessMicrosomal N-Glucuronidation of Nicotine and Cotinine: Human Hepatic Interindividual, Human Intertissue, and Interspecies Hepatic VariationOmar Ghosheh and Edward M. HawesDrug Metabolism and Disposition December 2002, 30 (12) 1478-1483; DOI: https://doi.org/10.1124/dmd.30.12.1478
Gibbs, Megan A.
- You have accessMicrosomal Protein Concentration Modifies the Apparent Inhibitory Potency of CYP3A InhibitorsThanh Huu Tran, Lisa L. von Moltke, Karthik Venkatakrishnan, Brian W. Granda, Megan A. Gibbs, R. Scott Obach, Jerold S. Harmatz and David J. GreenblattDrug Metabolism and Disposition December 2002, 30 (12) 1441-1445; DOI: https://doi.org/10.1124/dmd.30.12.1441
Goodisman, Jerry
- You have accessKinetic Study of the Reaction of Cisplatin with ThiolsJames C. Dabrowiak, Jerry Goodisman and Abdul-Kader SouidDrug Metabolism and Disposition December 2002, 30 (12) 1378-1384; DOI: https://doi.org/10.1124/dmd.30.12.1378
Granda, Brian W.
- You have accessMicrosomal Protein Concentration Modifies the Apparent Inhibitory Potency of CYP3A InhibitorsThanh Huu Tran, Lisa L. von Moltke, Karthik Venkatakrishnan, Brian W. Granda, Megan A. Gibbs, R. Scott Obach, Jerold S. Harmatz and David J. GreenblattDrug Metabolism and Disposition December 2002, 30 (12) 1441-1445; DOI: https://doi.org/10.1124/dmd.30.12.1441
Greenblatt, David J.
- You have accessMicrosomal Protein Concentration Modifies the Apparent Inhibitory Potency of CYP3A InhibitorsThanh Huu Tran, Lisa L. von Moltke, Karthik Venkatakrishnan, Brian W. Granda, Megan A. Gibbs, R. Scott Obach, Jerold S. Harmatz and David J. GreenblattDrug Metabolism and Disposition December 2002, 30 (12) 1441-1445; DOI: https://doi.org/10.1124/dmd.30.12.1441
Gustafsson, Lars L.
- You have accessEnzyme Kinetics for the Formation of 3-Hydroxyquinine and Three New Metabolites of Quinine in Vitro; 3-Hydroxylation by CYP3A4 is Indeed the Major Metabolic PathwayRajaa A. Mirghani, Ümit Yasar, Tao Zheng, James M. Cook, Lars L. Gustafsson, Gunnel Tybring and Örjan EricssonDrug Metabolism and Disposition December 2002, 30 (12) 1368-1371; DOI: https://doi.org/10.1124/dmd.30.12.1368
H
Halladay, Jason S.
- You have accessComparative Pharmacokinetic and Disposition Studies of [1-14C]1-Eicosanylcyclohexane, a Surrogate Mineral Hydrocarbon, in Female Fischer-344 and Sprague-Dawley RatsJason S. Halladay, Carl R. Mackerer, Lorraine E. Twerdok and I. Glenn SipesDrug Metabolism and Disposition December 2002, 30 (12) 1470-1477; DOI: https://doi.org/10.1124/dmd.30.12.1470
Harmatz, Jerold S.
- You have accessMicrosomal Protein Concentration Modifies the Apparent Inhibitory Potency of CYP3A InhibitorsThanh Huu Tran, Lisa L. von Moltke, Karthik Venkatakrishnan, Brian W. Granda, Megan A. Gibbs, R. Scott Obach, Jerold S. Harmatz and David J. GreenblattDrug Metabolism and Disposition December 2002, 30 (12) 1441-1445; DOI: https://doi.org/10.1124/dmd.30.12.1441
Hasegawa, Hiroshi
- You have accessKinetics of Sequential Metabolism from d-Leucine tol-Leucine via α-Ketoisocaproic Acid in RatHiroshi Hasegawa, Takehisa Matsukawa, Yoshihiko Shinohara and Takao HashimotoDrug Metabolism and Disposition December 2002, 30 (12) 1436-1440; DOI: https://doi.org/10.1124/dmd.30.12.1436
Hashimoto, Takao
- You have accessKinetics of Sequential Metabolism from d-Leucine tol-Leucine via α-Ketoisocaproic Acid in RatHiroshi Hasegawa, Takehisa Matsukawa, Yoshihiko Shinohara and Takao HashimotoDrug Metabolism and Disposition December 2002, 30 (12) 1436-1440; DOI: https://doi.org/10.1124/dmd.30.12.1436
Hasinoff, Brian B.
- You have accessDihydroorotase Catalyzes the Ring Opening of the Hydrolysis Intermediates of the Cardioprotective Drug Dexrazoxane (ICRF-187)Patricia E. Schroeder, Jeffrey N. Davidson and Brian B. HasinoffDrug Metabolism and Disposition December 2002, 30 (12) 1431-1435; DOI: https://doi.org/10.1124/dmd.30.12.1431
Hawes, Edward M.
- You have accessMicrosomal N-Glucuronidation of Nicotine and Cotinine: Human Hepatic Interindividual, Human Intertissue, and Interspecies Hepatic VariationOmar Ghosheh and Edward M. HawesDrug Metabolism and Disposition December 2002, 30 (12) 1478-1483; DOI: https://doi.org/10.1124/dmd.30.12.1478
Holmes, Elaine
- You have accessApplication of Directly Coupled High Performance Liquid Chromatography-NMR-Mass Spectometry and 1H NMR Spectroscopic Studies to the Investigation of 2,3-Benzofuran Metabolism in Sprague-Dawley RatsJohn C. Connelly, Susan C. Connor, Soria Monte, Nigel J.C. Bailey, Nathan Borgeaud, Elaine Holmes, Jeff Troke, Jeremy K. Nicholson and Claire L. GavaghanDrug Metabolism and Disposition December 2002, 30 (12) 1357-1363; DOI: https://doi.org/10.1124/dmd.30.12.1357
Houston, J. Brian
- You have accessQuinidine and Haloperidol as Modifiers of CYP3A4 Activity: Multisite Kinetic Model ApproachAleksandra Galetin, Stephen E. Clarke and J. Brian HoustonDrug Metabolism and Disposition December 2002, 30 (12) 1512-1522; DOI: https://doi.org/10.1124/dmd.30.12.1512
Hribar, Jeremy D.
- You have accessInvolvement of CYP3A in the Metabolism of Eplerenone in Humans and Dogs: Differential Metabolism by CYP3A4 and CYP3A5Chyung S. Cook, Loren M. Berry, David H. Kim, Earl G. Burton, Jeremy D. Hribar and Liming ZhangDrug Metabolism and Disposition December 2002, 30 (12) 1344-1351; DOI: https://doi.org/10.1124/dmd.30.12.1344
Hu, Yiding
- You have accessEnantioselective Metabolism of the Endocrine Disruptor Pesticide Methoxychlor by Human Cytochromes P450 (P450s): Major Differences in Selective Enantiomer Formation by Various P450 IsoformsYiding Hu and David KupferDrug Metabolism and Disposition December 2002, 30 (12) 1329-1336; DOI: https://doi.org/10.1124/dmd.30.12.1329
Huang, Jin-Ding
- You have accessPharmacokinetics of Midazolam and 1′-Hydroxymidazolam in Chinese with Different CYP3A5 GenotypesPei-Shan Shih and Jin-Ding HuangDrug Metabolism and Disposition December 2002, 30 (12) 1491-1496; DOI: https://doi.org/10.1124/dmd.30.12.1491
Huang, Shiew-Mei
- You have accessEvaluation of Cytochrome P450 Probe Substrates Commonly Used by the Pharmaceutical Industry to Study in Vitro Drug InteractionsRae Yuan, Soraya Madani, Xiao-Xiong Wei, Kellie Reynolds and Shiew-Mei HuangDrug Metabolism and Disposition December 2002, 30 (12) 1311-1319; DOI: https://doi.org/10.1124/dmd.30.12.1311
I
Inano, Keiko
- You have accessEffects of Olopatadine, a New Antiallergic Agent, on Human Liver Microsomal Cytochrome P450 ActivitiesJiro Kajita, Keiko Inano, Eiichi Fuse, Takashi Kuwabara and Hiroyuki KobayashiDrug Metabolism and Disposition December 2002, 30 (12) 1504-1511; DOI: https://doi.org/10.1124/dmd.30.12.1504
Itose, Minoru
- You have accessMechanism for the Tissue Distribution of Grepafloxacin, a Fluoroquinolone Antibiotic, in RatsTakashi Suzuki, Yukio Kato, Hiroyuki Sasabe, Minoru Itose, Gohachiro Miyamoto and Yuichi SugiyamaDrug Metabolism and Disposition December 2002, 30 (12) 1393-1399; DOI: https://doi.org/10.1124/dmd.30.12.1393
K
Kajita, Jiro
- You have accessEffects of Olopatadine, a New Antiallergic Agent, on Human Liver Microsomal Cytochrome P450 ActivitiesJiro Kajita, Keiko Inano, Eiichi Fuse, Takashi Kuwabara and Hiroyuki KobayashiDrug Metabolism and Disposition December 2002, 30 (12) 1504-1511; DOI: https://doi.org/10.1124/dmd.30.12.1504
Kato, Yukio
- You have accessMechanism for the Tissue Distribution of Grepafloxacin, a Fluoroquinolone Antibiotic, in RatsTakashi Suzuki, Yukio Kato, Hiroyuki Sasabe, Minoru Itose, Gohachiro Miyamoto and Yuichi SugiyamaDrug Metabolism and Disposition December 2002, 30 (12) 1393-1399; DOI: https://doi.org/10.1124/dmd.30.12.1393
Kellogg, G. E.
- You have accessIrreversible Inhibition of CYP2D6 by (−)-Chloroephedrine, a Possible Impurity in MethamphetamineB. Rege, K. M. Carter, M. A. Sarkar, G. E. Kellogg and W. H. SoineDrug Metabolism and Disposition December 2002, 30 (12) 1337-1343; DOI: https://doi.org/10.1124/dmd.30.12.1337
Kim, David H.
- You have accessInvolvement of CYP3A in the Metabolism of Eplerenone in Humans and Dogs: Differential Metabolism by CYP3A4 and CYP3A5Chyung S. Cook, Loren M. Berry, David H. Kim, Earl G. Burton, Jeremy D. Hribar and Liming ZhangDrug Metabolism and Disposition December 2002, 30 (12) 1344-1351; DOI: https://doi.org/10.1124/dmd.30.12.1344
Kitamura, Shigeyuki
- You have accessDeacylation of N-Arylformamides andN-Arylacetamides by Formamidase in Rat LiverOsamu Ueda, Shigeyuki Kitamura and Shigeru OhtaDrug Metabolism and Disposition December 2002, 30 (12) 1297-1299; DOI: https://doi.org/10.1124/dmd.30.12.1297
Knol, James A.
- You have accessRegional Pharmacokinetics of Amifostine in Anesthetized Dogs: Role of the Liver, Gastrointestinal Tract, Lungs, and KidneysMicha Levi, James A. Knol, William D. Ensminger, Susan J. DeRemer, Chunzhi Dou, Susan M. Lunte, Heather S. Bonner, Leslie M. Shaw and David E. SmithDrug Metabolism and Disposition December 2002, 30 (12) 1425-1430; DOI: https://doi.org/10.1124/dmd.30.12.1425
Kobayashi, Hiroyuki
- You have accessEffects of Olopatadine, a New Antiallergic Agent, on Human Liver Microsomal Cytochrome P450 ActivitiesJiro Kajita, Keiko Inano, Eiichi Fuse, Takashi Kuwabara and Hiroyuki KobayashiDrug Metabolism and Disposition December 2002, 30 (12) 1504-1511; DOI: https://doi.org/10.1124/dmd.30.12.1504
Kocarek, Thomas A.
- You have accessRegulation of CYP2B6 and CYP3A Expression by Hydroxymethylglutaryl Coenzyme A Inhibitors in Primary Cultured Human HepatocytesThomas A. Kocarek, Michael S. Dahn, Hongbo Cai, Stephen C. Strom and Nancy A. Mercer-HainesDrug Metabolism and Disposition December 2002, 30 (12) 1400-1405; DOI: https://doi.org/10.1124/dmd.30.12.1400
Kupfer, David
- You have accessEnantioselective Metabolism of the Endocrine Disruptor Pesticide Methoxychlor by Human Cytochromes P450 (P450s): Major Differences in Selective Enantiomer Formation by Various P450 IsoformsYiding Hu and David KupferDrug Metabolism and Disposition December 2002, 30 (12) 1329-1336; DOI: https://doi.org/10.1124/dmd.30.12.1329
Kuwabara, Takashi
- You have accessEffects of Olopatadine, a New Antiallergic Agent, on Human Liver Microsomal Cytochrome P450 ActivitiesJiro Kajita, Keiko Inano, Eiichi Fuse, Takashi Kuwabara and Hiroyuki KobayashiDrug Metabolism and Disposition December 2002, 30 (12) 1504-1511; DOI: https://doi.org/10.1124/dmd.30.12.1504
Kwon, Jun-Tack
- You have accessCharacterization of Nicotine and CotinineN-Glucuronidations in Human Liver MicrosomesMiki Nakajima, Eriko Tanaka, Jun-Tack Kwon and Tsuyoshi YokoiDrug Metabolism and Disposition December 2002, 30 (12) 1484-1490; DOI: https://doi.org/10.1124/dmd.30.12.1484
L
Lau, Yau Yi
- You have accessDevelopment of a Novel in Vitro Model to Predict Hepatic Clearance Using Fresh, Cryopreserved, and Sandwich-Cultured HepatocytesYau Yi Lau, Elpida Sapidou, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition December 2002, 30 (12) 1446-1454; DOI: https://doi.org/10.1124/dmd.30.12.1446
Laus, G.
- You have accessMajor Phase I Biotransformation Pathways of Trichostatin A in Rat Hepatocytes and in Rat and Human Liver MicrosomesG. Elaut, G. Török, M. Vinken, G. Laus, P. Papeleu, D. Tourwe and V. RogiersDrug Metabolism and Disposition December 2002, 30 (12) 1320-1328; DOI: https://doi.org/10.1124/dmd.30.12.1320
Lee, Chunja
- You have accessSuppression of Cytochrome P450 2C11 by Aromatic Hydrocarbons: Mechanistic Insights from Studies of the 5′-Flanking Region of theCYP2C11 GeneAnahita Bhathena, Chunja Lee and David S. RiddickDrug Metabolism and Disposition December 2002, 30 (12) 1385-1392; DOI: https://doi.org/10.1124/dmd.30.12.1385
Lee, Su-Jun
- You have accessFunctional Properties of a Rainbow Trout CYP3A27 Expressed by Recombinant Baculovirus in Insect CellsSu-Jun Lee and Donald R. BuhlerDrug Metabolism and Disposition December 2002, 30 (12) 1406-1412; DOI: https://doi.org/10.1124/dmd.30.12.1406
Levi, Micha
- You have accessRegional Pharmacokinetics of Amifostine in Anesthetized Dogs: Role of the Liver, Gastrointestinal Tract, Lungs, and KidneysMicha Levi, James A. Knol, William D. Ensminger, Susan J. DeRemer, Chunzhi Dou, Susan M. Lunte, Heather S. Bonner, Leslie M. Shaw and David E. SmithDrug Metabolism and Disposition December 2002, 30 (12) 1425-1430; DOI: https://doi.org/10.1124/dmd.30.12.1425
Lu, Jian-Feng
- You have accessModel-based Analysis of the Pharmacokinetic Interactions Between Ritonavir, Nelfinavir, and Saquinavir after Simultaneous and Staggered Oral AdministrationJian-Feng Lu, Terrence F. Blaschke, Charles Flexner, Susan L. Rosenkranz, Lewis B. Sheiner and AIDS Clinical Trials Group Protocol 378 InvestigatorsDrug Metabolism and Disposition December 2002, 30 (12) 1455-1461; DOI: https://doi.org/10.1124/dmd.30.12.1455
Lunte, Susan M.
- You have accessRegional Pharmacokinetics of Amifostine in Anesthetized Dogs: Role of the Liver, Gastrointestinal Tract, Lungs, and KidneysMicha Levi, James A. Knol, William D. Ensminger, Susan J. DeRemer, Chunzhi Dou, Susan M. Lunte, Heather S. Bonner, Leslie M. Shaw and David E. SmithDrug Metabolism and Disposition December 2002, 30 (12) 1425-1430; DOI: https://doi.org/10.1124/dmd.30.12.1425
M
Mackerer, Carl R.
- You have accessComparative Pharmacokinetic and Disposition Studies of [1-14C]1-Eicosanylcyclohexane, a Surrogate Mineral Hydrocarbon, in Female Fischer-344 and Sprague-Dawley RatsJason S. Halladay, Carl R. Mackerer, Lorraine E. Twerdok and I. Glenn SipesDrug Metabolism and Disposition December 2002, 30 (12) 1470-1477; DOI: https://doi.org/10.1124/dmd.30.12.1470
Madani, Soraya
- You have accessEvaluation of Cytochrome P450 Probe Substrates Commonly Used by the Pharmaceutical Industry to Study in Vitro Drug InteractionsRae Yuan, Soraya Madani, Xiao-Xiong Wei, Kellie Reynolds and Shiew-Mei HuangDrug Metabolism and Disposition December 2002, 30 (12) 1311-1319; DOI: https://doi.org/10.1124/dmd.30.12.1311
Matsukawa, Takehisa
- You have accessKinetics of Sequential Metabolism from d-Leucine tol-Leucine via α-Ketoisocaproic Acid in RatHiroshi Hasegawa, Takehisa Matsukawa, Yoshihiko Shinohara and Takao HashimotoDrug Metabolism and Disposition December 2002, 30 (12) 1436-1440; DOI: https://doi.org/10.1124/dmd.30.12.1436
Mercer-Haines, Nancy A.
- You have accessRegulation of CYP2B6 and CYP3A Expression by Hydroxymethylglutaryl Coenzyme A Inhibitors in Primary Cultured Human HepatocytesThomas A. Kocarek, Michael S. Dahn, Hongbo Cai, Stephen C. Strom and Nancy A. Mercer-HainesDrug Metabolism and Disposition December 2002, 30 (12) 1400-1405; DOI: https://doi.org/10.1124/dmd.30.12.1400
Mirghani, Rajaa A.
- You have accessEnzyme Kinetics for the Formation of 3-Hydroxyquinine and Three New Metabolites of Quinine in Vitro; 3-Hydroxylation by CYP3A4 is Indeed the Major Metabolic PathwayRajaa A. Mirghani, Ümit Yasar, Tao Zheng, James M. Cook, Lars L. Gustafsson, Gunnel Tybring and Örjan EricssonDrug Metabolism and Disposition December 2002, 30 (12) 1368-1371; DOI: https://doi.org/10.1124/dmd.30.12.1368
Miyamoto, Gohachiro
- You have accessMechanism for the Tissue Distribution of Grepafloxacin, a Fluoroquinolone Antibiotic, in RatsTakashi Suzuki, Yukio Kato, Hiroyuki Sasabe, Minoru Itose, Gohachiro Miyamoto and Yuichi SugiyamaDrug Metabolism and Disposition December 2002, 30 (12) 1393-1399; DOI: https://doi.org/10.1124/dmd.30.12.1393
Monte, Soria
- You have accessApplication of Directly Coupled High Performance Liquid Chromatography-NMR-Mass Spectometry and 1H NMR Spectroscopic Studies to the Investigation of 2,3-Benzofuran Metabolism in Sprague-Dawley RatsJohn C. Connelly, Susan C. Connor, Soria Monte, Nigel J.C. Bailey, Nathan Borgeaud, Elaine Holmes, Jeff Troke, Jeremy K. Nicholson and Claire L. GavaghanDrug Metabolism and Disposition December 2002, 30 (12) 1357-1363; DOI: https://doi.org/10.1124/dmd.30.12.1357
N
Nakajima, Miki
- You have accessTroglitazone Glucuronidation in Human Liver and Intestine Microsomes: High Catalytic Activity of UGT1A8 and UGT1A10Yuichiro Watanabe, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition December 2002, 30 (12) 1462-1469; DOI: https://doi.org/10.1124/dmd.30.12.1462
- You have accessCharacterization of Nicotine and CotinineN-Glucuronidations in Human Liver MicrosomesMiki Nakajima, Eriko Tanaka, Jun-Tack Kwon and Tsuyoshi YokoiDrug Metabolism and Disposition December 2002, 30 (12) 1484-1490; DOI: https://doi.org/10.1124/dmd.30.12.1484
Neuvonen, Mikko
- You have accessGemfibrozil Inhibits CYP2C8-Mediated Cerivastatin Metabolism in Human Liver MicrosomesJun-Sheng Wang, Mikko Neuvonen, Xia Wen, Janne T. Backman and Pertti J. NeuvonenDrug Metabolism and Disposition December 2002, 30 (12) 1352-1356; DOI: https://doi.org/10.1124/dmd.30.12.1352
Neuvonen, Pertti J.
- You have accessGemfibrozil Inhibits CYP2C8-Mediated Cerivastatin Metabolism in Human Liver MicrosomesJun-Sheng Wang, Mikko Neuvonen, Xia Wen, Janne T. Backman and Pertti J. NeuvonenDrug Metabolism and Disposition December 2002, 30 (12) 1352-1356; DOI: https://doi.org/10.1124/dmd.30.12.1352
Nicholson, Jeremy K.
- You have accessApplication of Directly Coupled High Performance Liquid Chromatography-NMR-Mass Spectometry and 1H NMR Spectroscopic Studies to the Investigation of 2,3-Benzofuran Metabolism in Sprague-Dawley RatsJohn C. Connelly, Susan C. Connor, Soria Monte, Nigel J.C. Bailey, Nathan Borgeaud, Elaine Holmes, Jeff Troke, Jeremy K. Nicholson and Claire L. GavaghanDrug Metabolism and Disposition December 2002, 30 (12) 1357-1363; DOI: https://doi.org/10.1124/dmd.30.12.1357
O
Obach, R. Scott
- You have accessMicrosomal Protein Concentration Modifies the Apparent Inhibitory Potency of CYP3A InhibitorsThanh Huu Tran, Lisa L. von Moltke, Karthik Venkatakrishnan, Brian W. Granda, Megan A. Gibbs, R. Scott Obach, Jerold S. Harmatz and David J. GreenblattDrug Metabolism and Disposition December 2002, 30 (12) 1441-1445; DOI: https://doi.org/10.1124/dmd.30.12.1441
Ohta, Shigeru
- You have accessDeacylation of N-Arylformamides andN-Arylacetamides by Formamidase in Rat LiverOsamu Ueda, Shigeyuki Kitamura and Shigeru OhtaDrug Metabolism and Disposition December 2002, 30 (12) 1297-1299; DOI: https://doi.org/10.1124/dmd.30.12.1297
P
Papeleu, P.
- You have accessMajor Phase I Biotransformation Pathways of Trichostatin A in Rat Hepatocytes and in Rat and Human Liver MicrosomesG. Elaut, G. Török, M. Vinken, G. Laus, P. Papeleu, D. Tourwe and V. RogiersDrug Metabolism and Disposition December 2002, 30 (12) 1320-1328; DOI: https://doi.org/10.1124/dmd.30.12.1320
Payan, Jean-Paul
- You have accessToxicokinetics and Metabolism ofN-[14C]Methylpyrrolidone in Male Sprague-Dawley Rats. A Saturable NMP Elimination ProcessJean-Paul Payan, Dominique Beydon, Jean-Paul Fabry, Isabelle Boudry, Benoit Cossec and Elisabeth FerrariDrug Metabolism and Disposition December 2002, 30 (12) 1418-1424; DOI: https://doi.org/10.1124/dmd.30.12.1418
R
Rege, B.
- You have accessIrreversible Inhibition of CYP2D6 by (−)-Chloroephedrine, a Possible Impurity in MethamphetamineB. Rege, K. M. Carter, M. A. Sarkar, G. E. Kellogg and W. H. SoineDrug Metabolism and Disposition December 2002, 30 (12) 1337-1343; DOI: https://doi.org/10.1124/dmd.30.12.1337
Reynolds, Kellie
- You have accessEvaluation of Cytochrome P450 Probe Substrates Commonly Used by the Pharmaceutical Industry to Study in Vitro Drug InteractionsRae Yuan, Soraya Madani, Xiao-Xiong Wei, Kellie Reynolds and Shiew-Mei HuangDrug Metabolism and Disposition December 2002, 30 (12) 1311-1319; DOI: https://doi.org/10.1124/dmd.30.12.1311
Riddick, David S.
- You have accessSuppression of Cytochrome P450 2C11 by Aromatic Hydrocarbons: Mechanistic Insights from Studies of the 5′-Flanking Region of theCYP2C11 GeneAnahita Bhathena, Chunja Lee and David S. RiddickDrug Metabolism and Disposition December 2002, 30 (12) 1385-1392; DOI: https://doi.org/10.1124/dmd.30.12.1385
Riley, Robert J.
- You have accessThe Influence of Nonspecific Microsomal Binding on Apparent Intrinsic Clearance, and Its Prediction from Physicochemical PropertiesRupert P. Austin, Patrick Barton, Scott L. Cockroft, Mark C. Wenlock and Robert J. RileyDrug Metabolism and Disposition December 2002, 30 (12) 1497-1503; DOI: https://doi.org/10.1124/dmd.30.12.1497
Rios, Gladys R.
- You have accessInhibition and Active Sites of UDP-Glucuronosyltransferases 2B7 and 1A1.Gladys R. Rios and Thomas R. TephlyDrug Metabolism and Disposition December 2002, 30 (12) 1364-1367; DOI: https://doi.org/10.1124/dmd.30.12.1364
Rogiers, V.
- You have accessMajor Phase I Biotransformation Pathways of Trichostatin A in Rat Hepatocytes and in Rat and Human Liver MicrosomesG. Elaut, G. Török, M. Vinken, G. Laus, P. Papeleu, D. Tourwe and V. RogiersDrug Metabolism and Disposition December 2002, 30 (12) 1320-1328; DOI: https://doi.org/10.1124/dmd.30.12.1320
Rosenkranz, Susan L.
- You have accessModel-based Analysis of the Pharmacokinetic Interactions Between Ritonavir, Nelfinavir, and Saquinavir after Simultaneous and Staggered Oral AdministrationJian-Feng Lu, Terrence F. Blaschke, Charles Flexner, Susan L. Rosenkranz, Lewis B. Sheiner and AIDS Clinical Trials Group Protocol 378 InvestigatorsDrug Metabolism and Disposition December 2002, 30 (12) 1455-1461; DOI: https://doi.org/10.1124/dmd.30.12.1455
S
Sapidou, Elpida
- You have accessDevelopment of a Novel in Vitro Model to Predict Hepatic Clearance Using Fresh, Cryopreserved, and Sandwich-Cultured HepatocytesYau Yi Lau, Elpida Sapidou, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition December 2002, 30 (12) 1446-1454; DOI: https://doi.org/10.1124/dmd.30.12.1446
Sarkar, M. A.
- You have accessIrreversible Inhibition of CYP2D6 by (−)-Chloroephedrine, a Possible Impurity in MethamphetamineB. Rege, K. M. Carter, M. A. Sarkar, G. E. Kellogg and W. H. SoineDrug Metabolism and Disposition December 2002, 30 (12) 1337-1343; DOI: https://doi.org/10.1124/dmd.30.12.1337
Sasabe, Hiroyuki
- You have accessMechanism for the Tissue Distribution of Grepafloxacin, a Fluoroquinolone Antibiotic, in RatsTakashi Suzuki, Yukio Kato, Hiroyuki Sasabe, Minoru Itose, Gohachiro Miyamoto and Yuichi SugiyamaDrug Metabolism and Disposition December 2002, 30 (12) 1393-1399; DOI: https://doi.org/10.1124/dmd.30.12.1393
Schroeder, Patricia E.
- You have accessDihydroorotase Catalyzes the Ring Opening of the Hydrolysis Intermediates of the Cardioprotective Drug Dexrazoxane (ICRF-187)Patricia E. Schroeder, Jeffrey N. Davidson and Brian B. HasinoffDrug Metabolism and Disposition December 2002, 30 (12) 1431-1435; DOI: https://doi.org/10.1124/dmd.30.12.1431
Sharma, Rajendra
- You have accessRLIP76, a Novel Transporter Catalyzing ATP-Dependent Efflux of XenobioticsSanjay Awasthi, Rajendra Sharma, Sharad S. Singhal, Piotr Zimniak and Yogesh C. AwasthiDrug Metabolism and Disposition December 2002, 30 (12) 1300-1310; DOI: https://doi.org/10.1124/dmd.30.12.1300
Shaw, Leslie M.
- You have accessRegional Pharmacokinetics of Amifostine in Anesthetized Dogs: Role of the Liver, Gastrointestinal Tract, Lungs, and KidneysMicha Levi, James A. Knol, William D. Ensminger, Susan J. DeRemer, Chunzhi Dou, Susan M. Lunte, Heather S. Bonner, Leslie M. Shaw and David E. SmithDrug Metabolism and Disposition December 2002, 30 (12) 1425-1430; DOI: https://doi.org/10.1124/dmd.30.12.1425
Sheiner, Lewis B.
- You have accessModel-based Analysis of the Pharmacokinetic Interactions Between Ritonavir, Nelfinavir, and Saquinavir after Simultaneous and Staggered Oral AdministrationJian-Feng Lu, Terrence F. Blaschke, Charles Flexner, Susan L. Rosenkranz, Lewis B. Sheiner and AIDS Clinical Trials Group Protocol 378 InvestigatorsDrug Metabolism and Disposition December 2002, 30 (12) 1455-1461; DOI: https://doi.org/10.1124/dmd.30.12.1455
Shih, Pei-Shan
- You have accessPharmacokinetics of Midazolam and 1′-Hydroxymidazolam in Chinese with Different CYP3A5 GenotypesPei-Shan Shih and Jin-Ding HuangDrug Metabolism and Disposition December 2002, 30 (12) 1491-1496; DOI: https://doi.org/10.1124/dmd.30.12.1491
Shinohara, Yoshihiko
- You have accessKinetics of Sequential Metabolism from d-Leucine tol-Leucine via α-Ketoisocaproic Acid in RatHiroshi Hasegawa, Takehisa Matsukawa, Yoshihiko Shinohara and Takao HashimotoDrug Metabolism and Disposition December 2002, 30 (12) 1436-1440; DOI: https://doi.org/10.1124/dmd.30.12.1436
Singhal, Sharad S.
- You have accessRLIP76, a Novel Transporter Catalyzing ATP-Dependent Efflux of XenobioticsSanjay Awasthi, Rajendra Sharma, Sharad S. Singhal, Piotr Zimniak and Yogesh C. AwasthiDrug Metabolism and Disposition December 2002, 30 (12) 1300-1310; DOI: https://doi.org/10.1124/dmd.30.12.1300
Sipes, I. Glenn
- You have accessComparative Pharmacokinetic and Disposition Studies of [1-14C]1-Eicosanylcyclohexane, a Surrogate Mineral Hydrocarbon, in Female Fischer-344 and Sprague-Dawley RatsJason S. Halladay, Carl R. Mackerer, Lorraine E. Twerdok and I. Glenn SipesDrug Metabolism and Disposition December 2002, 30 (12) 1470-1477; DOI: https://doi.org/10.1124/dmd.30.12.1470
Slattery, John T.
- You have accessEffects of Ethanol Dose and Ethanol Withdrawal on Rat Liver Mitochondrial Glutathione: Implication of Potentiated Acetaminophen Toxicity in AlcoholicsPing Zhao and John T. SlatteryDrug Metabolism and Disposition December 2002, 30 (12) 1413-1417; DOI: https://doi.org/10.1124/dmd.30.12.1413
Smith, David E.
- You have accessRegional Pharmacokinetics of Amifostine in Anesthetized Dogs: Role of the Liver, Gastrointestinal Tract, Lungs, and KidneysMicha Levi, James A. Knol, William D. Ensminger, Susan J. DeRemer, Chunzhi Dou, Susan M. Lunte, Heather S. Bonner, Leslie M. Shaw and David E. SmithDrug Metabolism and Disposition December 2002, 30 (12) 1425-1430; DOI: https://doi.org/10.1124/dmd.30.12.1425
Soine, W. H.
- You have accessIrreversible Inhibition of CYP2D6 by (−)-Chloroephedrine, a Possible Impurity in MethamphetamineB. Rege, K. M. Carter, M. A. Sarkar, G. E. Kellogg and W. H. SoineDrug Metabolism and Disposition December 2002, 30 (12) 1337-1343; DOI: https://doi.org/10.1124/dmd.30.12.1337
Souid, Abdul-Kader
- You have accessKinetic Study of the Reaction of Cisplatin with ThiolsJames C. Dabrowiak, Jerry Goodisman and Abdul-Kader SouidDrug Metabolism and Disposition December 2002, 30 (12) 1378-1384; DOI: https://doi.org/10.1124/dmd.30.12.1378
Strom, Stephen C.
- You have accessRegulation of CYP2B6 and CYP3A Expression by Hydroxymethylglutaryl Coenzyme A Inhibitors in Primary Cultured Human HepatocytesThomas A. Kocarek, Michael S. Dahn, Hongbo Cai, Stephen C. Strom and Nancy A. Mercer-HainesDrug Metabolism and Disposition December 2002, 30 (12) 1400-1405; DOI: https://doi.org/10.1124/dmd.30.12.1400
Sugiyama, Yuichi
- You have accessMechanism for the Tissue Distribution of Grepafloxacin, a Fluoroquinolone Antibiotic, in RatsTakashi Suzuki, Yukio Kato, Hiroyuki Sasabe, Minoru Itose, Gohachiro Miyamoto and Yuichi SugiyamaDrug Metabolism and Disposition December 2002, 30 (12) 1393-1399; DOI: https://doi.org/10.1124/dmd.30.12.1393
Suzuki, Takashi
- You have accessMechanism for the Tissue Distribution of Grepafloxacin, a Fluoroquinolone Antibiotic, in RatsTakashi Suzuki, Yukio Kato, Hiroyuki Sasabe, Minoru Itose, Gohachiro Miyamoto and Yuichi SugiyamaDrug Metabolism and Disposition December 2002, 30 (12) 1393-1399; DOI: https://doi.org/10.1124/dmd.30.12.1393
T
Tanaka, Eriko
- You have accessCharacterization of Nicotine and CotinineN-Glucuronidations in Human Liver MicrosomesMiki Nakajima, Eriko Tanaka, Jun-Tack Kwon and Tsuyoshi YokoiDrug Metabolism and Disposition December 2002, 30 (12) 1484-1490; DOI: https://doi.org/10.1124/dmd.30.12.1484
Tephly, Thomas R.
- You have accessInhibition and Active Sites of UDP-Glucuronosyltransferases 2B7 and 1A1.Gladys R. Rios and Thomas R. TephlyDrug Metabolism and Disposition December 2002, 30 (12) 1364-1367; DOI: https://doi.org/10.1124/dmd.30.12.1364
Török, G.
- You have accessMajor Phase I Biotransformation Pathways of Trichostatin A in Rat Hepatocytes and in Rat and Human Liver MicrosomesG. Elaut, G. Török, M. Vinken, G. Laus, P. Papeleu, D. Tourwe and V. RogiersDrug Metabolism and Disposition December 2002, 30 (12) 1320-1328; DOI: https://doi.org/10.1124/dmd.30.12.1320
Tourwe, D.
- You have accessMajor Phase I Biotransformation Pathways of Trichostatin A in Rat Hepatocytes and in Rat and Human Liver MicrosomesG. Elaut, G. Török, M. Vinken, G. Laus, P. Papeleu, D. Tourwe and V. RogiersDrug Metabolism and Disposition December 2002, 30 (12) 1320-1328; DOI: https://doi.org/10.1124/dmd.30.12.1320
Tran, Thanh Huu
- You have accessMicrosomal Protein Concentration Modifies the Apparent Inhibitory Potency of CYP3A InhibitorsThanh Huu Tran, Lisa L. von Moltke, Karthik Venkatakrishnan, Brian W. Granda, Megan A. Gibbs, R. Scott Obach, Jerold S. Harmatz and David J. GreenblattDrug Metabolism and Disposition December 2002, 30 (12) 1441-1445; DOI: https://doi.org/10.1124/dmd.30.12.1441
Troke, Jeff
- You have accessApplication of Directly Coupled High Performance Liquid Chromatography-NMR-Mass Spectometry and 1H NMR Spectroscopic Studies to the Investigation of 2,3-Benzofuran Metabolism in Sprague-Dawley RatsJohn C. Connelly, Susan C. Connor, Soria Monte, Nigel J.C. Bailey, Nathan Borgeaud, Elaine Holmes, Jeff Troke, Jeremy K. Nicholson and Claire L. GavaghanDrug Metabolism and Disposition December 2002, 30 (12) 1357-1363; DOI: https://doi.org/10.1124/dmd.30.12.1357
Twerdok, Lorraine E.
- You have accessComparative Pharmacokinetic and Disposition Studies of [1-14C]1-Eicosanylcyclohexane, a Surrogate Mineral Hydrocarbon, in Female Fischer-344 and Sprague-Dawley RatsJason S. Halladay, Carl R. Mackerer, Lorraine E. Twerdok and I. Glenn SipesDrug Metabolism and Disposition December 2002, 30 (12) 1470-1477; DOI: https://doi.org/10.1124/dmd.30.12.1470
Tybring, Gunnel
- You have accessEnzyme Kinetics for the Formation of 3-Hydroxyquinine and Three New Metabolites of Quinine in Vitro; 3-Hydroxylation by CYP3A4 is Indeed the Major Metabolic PathwayRajaa A. Mirghani, Ümit Yasar, Tao Zheng, James M. Cook, Lars L. Gustafsson, Gunnel Tybring and Örjan EricssonDrug Metabolism and Disposition December 2002, 30 (12) 1368-1371; DOI: https://doi.org/10.1124/dmd.30.12.1368
U
Uckun, Fatih M.
- You have accessMetabolism of Stavudine-5′-[p-Bromophenyl Methoxyalaninyl Phosphate], Stampidine, in Mice, Dogs, and CatsChun-Lin Chen, Gengli Yu, T. K. Venkatachalam and Fatih M. UckunDrug Metabolism and Disposition December 2002, 30 (12) 1523-1531; DOI: https://doi.org/10.1124/dmd.30.12.1523
Ueda, Osamu
- You have accessDeacylation of N-Arylformamides andN-Arylacetamides by Formamidase in Rat LiverOsamu Ueda, Shigeyuki Kitamura and Shigeru OhtaDrug Metabolism and Disposition December 2002, 30 (12) 1297-1299; DOI: https://doi.org/10.1124/dmd.30.12.1297
V
Venkatachalam, T. K.
- You have accessMetabolism of Stavudine-5′-[p-Bromophenyl Methoxyalaninyl Phosphate], Stampidine, in Mice, Dogs, and CatsChun-Lin Chen, Gengli Yu, T. K. Venkatachalam and Fatih M. UckunDrug Metabolism and Disposition December 2002, 30 (12) 1523-1531; DOI: https://doi.org/10.1124/dmd.30.12.1523
Venkatakrishnan, Karthik
- You have accessMicrosomal Protein Concentration Modifies the Apparent Inhibitory Potency of CYP3A InhibitorsThanh Huu Tran, Lisa L. von Moltke, Karthik Venkatakrishnan, Brian W. Granda, Megan A. Gibbs, R. Scott Obach, Jerold S. Harmatz and David J. GreenblattDrug Metabolism and Disposition December 2002, 30 (12) 1441-1445; DOI: https://doi.org/10.1124/dmd.30.12.1441
Vinken, M.
- You have accessMajor Phase I Biotransformation Pathways of Trichostatin A in Rat Hepatocytes and in Rat and Human Liver MicrosomesG. Elaut, G. Török, M. Vinken, G. Laus, P. Papeleu, D. Tourwe and V. RogiersDrug Metabolism and Disposition December 2002, 30 (12) 1320-1328; DOI: https://doi.org/10.1124/dmd.30.12.1320
von Moltke, Lisa L.
- You have accessMicrosomal Protein Concentration Modifies the Apparent Inhibitory Potency of CYP3A InhibitorsThanh Huu Tran, Lisa L. von Moltke, Karthik Venkatakrishnan, Brian W. Granda, Megan A. Gibbs, R. Scott Obach, Jerold S. Harmatz and David J. GreenblattDrug Metabolism and Disposition December 2002, 30 (12) 1441-1445; DOI: https://doi.org/10.1124/dmd.30.12.1441
W
Wang, Jun-Sheng
- You have accessGemfibrozil Inhibits CYP2C8-Mediated Cerivastatin Metabolism in Human Liver MicrosomesJun-Sheng Wang, Mikko Neuvonen, Xia Wen, Janne T. Backman and Pertti J. NeuvonenDrug Metabolism and Disposition December 2002, 30 (12) 1352-1356; DOI: https://doi.org/10.1124/dmd.30.12.1352
Watanabe, Yuichiro
- You have accessTroglitazone Glucuronidation in Human Liver and Intestine Microsomes: High Catalytic Activity of UGT1A8 and UGT1A10Yuichiro Watanabe, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition December 2002, 30 (12) 1462-1469; DOI: https://doi.org/10.1124/dmd.30.12.1462
Wei, Xiao-Xiong
- You have accessEvaluation of Cytochrome P450 Probe Substrates Commonly Used by the Pharmaceutical Industry to Study in Vitro Drug InteractionsRae Yuan, Soraya Madani, Xiao-Xiong Wei, Kellie Reynolds and Shiew-Mei HuangDrug Metabolism and Disposition December 2002, 30 (12) 1311-1319; DOI: https://doi.org/10.1124/dmd.30.12.1311
Wen, Xia
- You have accessGemfibrozil Inhibits CYP2C8-Mediated Cerivastatin Metabolism in Human Liver MicrosomesJun-Sheng Wang, Mikko Neuvonen, Xia Wen, Janne T. Backman and Pertti J. NeuvonenDrug Metabolism and Disposition December 2002, 30 (12) 1352-1356; DOI: https://doi.org/10.1124/dmd.30.12.1352
Wenlock, Mark C.
- You have accessThe Influence of Nonspecific Microsomal Binding on Apparent Intrinsic Clearance, and Its Prediction from Physicochemical PropertiesRupert P. Austin, Patrick Barton, Scott L. Cockroft, Mark C. Wenlock and Robert J. RileyDrug Metabolism and Disposition December 2002, 30 (12) 1497-1503; DOI: https://doi.org/10.1124/dmd.30.12.1497
White, Ronald E.
- You have accessDevelopment of a Novel in Vitro Model to Predict Hepatic Clearance Using Fresh, Cryopreserved, and Sandwich-Cultured HepatocytesYau Yi Lau, Elpida Sapidou, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition December 2002, 30 (12) 1446-1454; DOI: https://doi.org/10.1124/dmd.30.12.1446
Wienkers, Larry C.
- You have accessMultiple Cytochrome P450 Enzymes Responsible for the Oxidative Metabolism of the Substituted (S)-3-Phenylpiperidine, (S,S)-3-[3-(Methylsulfonyl)phenyl]-1-propylpiperidine Hydrochloride, in Human Liver MicrosomesLarry C. Wienkers and Michael A. WynaldaDrug Metabolism and Disposition December 2002, 30 (12) 1372-1377; DOI: https://doi.org/10.1124/dmd.30.12.1372
Wynalda, Michael A.
- You have accessMultiple Cytochrome P450 Enzymes Responsible for the Oxidative Metabolism of the Substituted (S)-3-Phenylpiperidine, (S,S)-3-[3-(Methylsulfonyl)phenyl]-1-propylpiperidine Hydrochloride, in Human Liver MicrosomesLarry C. Wienkers and Michael A. WynaldaDrug Metabolism and Disposition December 2002, 30 (12) 1372-1377; DOI: https://doi.org/10.1124/dmd.30.12.1372
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Yasar, Ümit
- You have accessEnzyme Kinetics for the Formation of 3-Hydroxyquinine and Three New Metabolites of Quinine in Vitro; 3-Hydroxylation by CYP3A4 is Indeed the Major Metabolic PathwayRajaa A. Mirghani, Ümit Yasar, Tao Zheng, James M. Cook, Lars L. Gustafsson, Gunnel Tybring and Örjan EricssonDrug Metabolism and Disposition December 2002, 30 (12) 1368-1371; DOI: https://doi.org/10.1124/dmd.30.12.1368
Yokoi, Tsuyoshi
- You have accessTroglitazone Glucuronidation in Human Liver and Intestine Microsomes: High Catalytic Activity of UGT1A8 and UGT1A10Yuichiro Watanabe, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition December 2002, 30 (12) 1462-1469; DOI: https://doi.org/10.1124/dmd.30.12.1462
- You have accessCharacterization of Nicotine and CotinineN-Glucuronidations in Human Liver MicrosomesMiki Nakajima, Eriko Tanaka, Jun-Tack Kwon and Tsuyoshi YokoiDrug Metabolism and Disposition December 2002, 30 (12) 1484-1490; DOI: https://doi.org/10.1124/dmd.30.12.1484
Yu, Gengli
- You have accessMetabolism of Stavudine-5′-[p-Bromophenyl Methoxyalaninyl Phosphate], Stampidine, in Mice, Dogs, and CatsChun-Lin Chen, Gengli Yu, T. K. Venkatachalam and Fatih M. UckunDrug Metabolism and Disposition December 2002, 30 (12) 1523-1531; DOI: https://doi.org/10.1124/dmd.30.12.1523
Yuan, Rae
- You have accessEvaluation of Cytochrome P450 Probe Substrates Commonly Used by the Pharmaceutical Industry to Study in Vitro Drug InteractionsRae Yuan, Soraya Madani, Xiao-Xiong Wei, Kellie Reynolds and Shiew-Mei HuangDrug Metabolism and Disposition December 2002, 30 (12) 1311-1319; DOI: https://doi.org/10.1124/dmd.30.12.1311
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Zhang, Liming
- You have accessInvolvement of CYP3A in the Metabolism of Eplerenone in Humans and Dogs: Differential Metabolism by CYP3A4 and CYP3A5Chyung S. Cook, Loren M. Berry, David H. Kim, Earl G. Burton, Jeremy D. Hribar and Liming ZhangDrug Metabolism and Disposition December 2002, 30 (12) 1344-1351; DOI: https://doi.org/10.1124/dmd.30.12.1344
Zhao, Ping
- You have accessEffects of Ethanol Dose and Ethanol Withdrawal on Rat Liver Mitochondrial Glutathione: Implication of Potentiated Acetaminophen Toxicity in AlcoholicsPing Zhao and John T. SlatteryDrug Metabolism and Disposition December 2002, 30 (12) 1413-1417; DOI: https://doi.org/10.1124/dmd.30.12.1413
Zheng, Tao
- You have accessEnzyme Kinetics for the Formation of 3-Hydroxyquinine and Three New Metabolites of Quinine in Vitro; 3-Hydroxylation by CYP3A4 is Indeed the Major Metabolic PathwayRajaa A. Mirghani, Ümit Yasar, Tao Zheng, James M. Cook, Lars L. Gustafsson, Gunnel Tybring and Örjan EricssonDrug Metabolism and Disposition December 2002, 30 (12) 1368-1371; DOI: https://doi.org/10.1124/dmd.30.12.1368
Zimniak, Piotr
- You have accessRLIP76, a Novel Transporter Catalyzing ATP-Dependent Efflux of XenobioticsSanjay Awasthi, Rajendra Sharma, Sharad S. Singhal, Piotr Zimniak and Yogesh C. AwasthiDrug Metabolism and Disposition December 2002, 30 (12) 1300-1310; DOI: https://doi.org/10.1124/dmd.30.12.1300