Index by author
August 01, 2002; Volume 30,Issue 8
A
Augustijns, P.
- You have accessIntestinal Absorption Enhancement of the Ester Prodrug Tenofovir Disoproxil Fumarate through Modulation of the Biochemical Barrier by Defined Ester MixturesJ. van Gelder, S. Deferme, L. Naesens, E. De Clercq, G. van den Mooter, R. Kinget and P. AugustijnsDrug Metabolism and Disposition August 2002, 30 (8) 924-930; DOI: https://doi.org/10.1124/dmd.30.8.924
B
Brouwer, Kim L. R.
- You have accessRole of Constitutive Androstane Receptor in the In Vivo Induction of Mrp3 and CYP2B1/2 by PhenobarbitalHao Xiong, Kouichi Yoshinari, Kim L. R. Brouwer and Masahiko NegishiDrug Metabolism and Disposition August 2002, 30 (8) 918-923; DOI: https://doi.org/10.1124/dmd.30.8.918
C
Cantrell, Varon E.
- You have accessComparative Metabolic Capabilities of CYP3A4, CYP3A5, and CYP3A7J. Andrew Williams, Barbara J. Ring, Varon E. Cantrell, David R. Jones, James Eckstein, Kenneth Ruterbories, Mitchell A. Hamman, Stephen D. Hall and Steven A. WrightonDrug Metabolism and Disposition August 2002, 30 (8) 883-891; DOI: https://doi.org/10.1124/dmd.30.8.883
Chanas, Brian
- You have accessCytochrome P450 2E1 (CYP2E1) is Essential for Acrylonitrile Metabolism to Cyanide: Comparative Studies Using CYP2E1-Null and Wild-Type MiceHongbing Wang, Brian Chanas and Burhan I. GhanayemDrug Metabolism and Disposition August 2002, 30 (8) 911-917; DOI: https://doi.org/10.1124/dmd.30.8.911
Chiba, Masato
- You have accessPrediction of Hepatic Clearance and Availability by Cryopreserved Human Hepatocytes: An Application of Serum Incubation MethodYoshihiro Shibata, Hiroyuki Takahashi, Masato Chiba and Yasuyuki IshiiDrug Metabolism and Disposition August 2002, 30 (8) 892-896; DOI: https://doi.org/10.1124/dmd.30.8.892
Chiu, Shuet-Hing L.
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
Crewe, H. Kim
- You have accessMetabolism of Tamoxifen by Recombinant Human Cytochrome P450 Enzymes: Formation of the 4-Hydroxy, 4′-Hydroxy andN-Desmethyl Metabolites and Isomerization oftrans-4-HydroxytamoxifenH. Kim Crewe, Lisa M. Notley, Rebecca M. Wunsch, Martin S. Lennard and Elizabeth M. J. GillamDrug Metabolism and Disposition August 2002, 30 (8) 869-874; DOI: https://doi.org/10.1124/dmd.30.8.869
Curtis, Neil
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
D
Dabrowiak, James C.
- You have accessKinetic Analysis of the Reactions of 4-Hydroperoxycyclophosphamide and Acrolein With Glutathione, Mesna, and Wr-1065Kirk A. Tacka, James C. Dabrowiak, Jerry Goodisman and Abdul-Kader SouidDrug Metabolism and Disposition August 2002, 30 (8) 875-882; DOI: https://doi.org/10.1124/dmd.30.8.875
Dean, Dennis C.
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
De Clercq, E.
- You have accessIntestinal Absorption Enhancement of the Ester Prodrug Tenofovir Disoproxil Fumarate through Modulation of the Biochemical Barrier by Defined Ester MixturesJ. van Gelder, S. Deferme, L. Naesens, E. De Clercq, G. van den Mooter, R. Kinget and P. AugustijnsDrug Metabolism and Disposition August 2002, 30 (8) 924-930; DOI: https://doi.org/10.1124/dmd.30.8.924
Deferme, S.
- You have accessIntestinal Absorption Enhancement of the Ester Prodrug Tenofovir Disoproxil Fumarate through Modulation of the Biochemical Barrier by Defined Ester MixturesJ. van Gelder, S. Deferme, L. Naesens, E. De Clercq, G. van den Mooter, R. Kinget and P. AugustijnsDrug Metabolism and Disposition August 2002, 30 (8) 924-930; DOI: https://doi.org/10.1124/dmd.30.8.924
E
Eckstein, James
- You have accessComparative Metabolic Capabilities of CYP3A4, CYP3A5, and CYP3A7J. Andrew Williams, Barbara J. Ring, Varon E. Cantrell, David R. Jones, James Eckstein, Kenneth Ruterbories, Mitchell A. Hamman, Stephen D. Hall and Steven A. WrightonDrug Metabolism and Disposition August 2002, 30 (8) 883-891; DOI: https://doi.org/10.1124/dmd.30.8.883
Elipe, Maria Victoria Silva
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
Elliott, Jason
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
Evans, David C.
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
F
Friedman, Michael
- You have accessPharmacokinetic-Pharmacodynamic Analysis of the Glucose-Lowering Effect of Metformin in Diabetic Rats Reveals First-Pass Pharmacodynamic EffectDavid Stepensky, Michael Friedman, Itamar Raz and Amnon HoffmanDrug Metabolism and Disposition August 2002, 30 (8) 861-868; DOI: https://doi.org/10.1124/dmd.30.8.861
G
Gerhard, Ute
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
Ghanayem, Burhan I.
- You have accessCytochrome P450 2E1 (CYP2E1) is Essential for Acrylonitrile Metabolism to Cyanide: Comparative Studies Using CYP2E1-Null and Wild-Type MiceHongbing Wang, Brian Chanas and Burhan I. GhanayemDrug Metabolism and Disposition August 2002, 30 (8) 911-917; DOI: https://doi.org/10.1124/dmd.30.8.911
Gillam, Elizabeth M. J.
- You have accessMetabolism of Tamoxifen by Recombinant Human Cytochrome P450 Enzymes: Formation of the 4-Hydroxy, 4′-Hydroxy andN-Desmethyl Metabolites and Isomerization oftrans-4-HydroxytamoxifenH. Kim Crewe, Lisa M. Notley, Rebecca M. Wunsch, Martin S. Lennard and Elizabeth M. J. GillamDrug Metabolism and Disposition August 2002, 30 (8) 869-874; DOI: https://doi.org/10.1124/dmd.30.8.869
Goodisman, Jerry
- You have accessKinetic Analysis of the Reactions of 4-Hydroperoxycyclophosphamide and Acrolein With Glutathione, Mesna, and Wr-1065Kirk A. Tacka, James C. Dabrowiak, Jerry Goodisman and Abdul-Kader SouidDrug Metabolism and Disposition August 2002, 30 (8) 875-882; DOI: https://doi.org/10.1124/dmd.30.8.875
H
Hall, Stephen D.
- You have accessComparative Metabolic Capabilities of CYP3A4, CYP3A5, and CYP3A7J. Andrew Williams, Barbara J. Ring, Varon E. Cantrell, David R. Jones, James Eckstein, Kenneth Ruterbories, Mitchell A. Hamman, Stephen D. Hall and Steven A. WrightonDrug Metabolism and Disposition August 2002, 30 (8) 883-891; DOI: https://doi.org/10.1124/dmd.30.8.883
Hamman, Mitchell A.
- You have accessComparative Metabolic Capabilities of CYP3A4, CYP3A5, and CYP3A7J. Andrew Williams, Barbara J. Ring, Varon E. Cantrell, David R. Jones, James Eckstein, Kenneth Ruterbories, Mitchell A. Hamman, Stephen D. Hall and Steven A. WrightonDrug Metabolism and Disposition August 2002, 30 (8) 883-891; DOI: https://doi.org/10.1124/dmd.30.8.883
Hoffman, Amnon
- You have accessPharmacokinetic-Pharmacodynamic Analysis of the Glucose-Lowering Effect of Metformin in Diabetic Rats Reveals First-Pass Pharmacodynamic EffectDavid Stepensky, Michael Friedman, Itamar Raz and Amnon HoffmanDrug Metabolism and Disposition August 2002, 30 (8) 861-868; DOI: https://doi.org/10.1124/dmd.30.8.861
Honma, Wataru
- You have accessPhenol Sulfotransferase, ST1A3, as the Main Enzyme Catalyzing Sulfation of Troglitazone in Human LiverWataru Honma, Miki Shimada, Hironobu Sasano, Shogo Ozawa, Masaaki Miyata, Kiyoshi Nagata, Toshihiko Ikeda and Yasushi YamazoeDrug Metabolism and Disposition August 2002, 30 (8) 944-949; DOI: https://doi.org/10.1124/dmd.30.8.944
Hop, Cornelis E. C. A.
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
I
Ikeda, Toshihiko
- You have accessSex Difference in Inhibition of In Vitro Mexazolam Metabolism by Various 3-Hydroxy-3-Methylglutaryl-Coenzyme A Reductase Inhibitors in Rat Liver MicrosomesMichi Ishigami, Wataru Takasaki, Toshihiko Ikeda, Toru Komai, Kiyomi Ito and Yuichi SugiyamaDrug Metabolism and Disposition August 2002, 30 (8) 904-910; DOI: https://doi.org/10.1124/dmd.30.8.904
- You have accessPhenol Sulfotransferase, ST1A3, as the Main Enzyme Catalyzing Sulfation of Troglitazone in Human LiverWataru Honma, Miki Shimada, Hironobu Sasano, Shogo Ozawa, Masaaki Miyata, Kiyoshi Nagata, Toshihiko Ikeda and Yasushi YamazoeDrug Metabolism and Disposition August 2002, 30 (8) 944-949; DOI: https://doi.org/10.1124/dmd.30.8.944
Ishibashi, Fumihide
- You have accessAmino Acid Residues Affecting the Activities of Human Cytochrome P450 2C9 and 2C19Toshiro Niwa, Akira Kageyama, Kae Kishimoto, Yoshiyasu Yabusaki, Fumihide Ishibashi and Masanao KatagiriDrug Metabolism and Disposition August 2002, 30 (8) 931-936; DOI: https://doi.org/10.1124/dmd.30.8.931
Ishigami, Michi
- You have accessSex Difference in Inhibition of In Vitro Mexazolam Metabolism by Various 3-Hydroxy-3-Methylglutaryl-Coenzyme A Reductase Inhibitors in Rat Liver MicrosomesMichi Ishigami, Wataru Takasaki, Toshihiko Ikeda, Toru Komai, Kiyomi Ito and Yuichi SugiyamaDrug Metabolism and Disposition August 2002, 30 (8) 904-910; DOI: https://doi.org/10.1124/dmd.30.8.904
Ishii, Yasuyuki
- You have accessPrediction of Hepatic Clearance and Availability by Cryopreserved Human Hepatocytes: An Application of Serum Incubation MethodYoshihiro Shibata, Hiroyuki Takahashi, Masato Chiba and Yasuyuki IshiiDrug Metabolism and Disposition August 2002, 30 (8) 892-896; DOI: https://doi.org/10.1124/dmd.30.8.892
Ito, Kiyomi
- You have accessSex Difference in Inhibition of In Vitro Mexazolam Metabolism by Various 3-Hydroxy-3-Methylglutaryl-Coenzyme A Reductase Inhibitors in Rat Liver MicrosomesMichi Ishigami, Wataru Takasaki, Toshihiko Ikeda, Toru Komai, Kiyomi Ito and Yuichi SugiyamaDrug Metabolism and Disposition August 2002, 30 (8) 904-910; DOI: https://doi.org/10.1124/dmd.30.8.904
J
Jones, David R.
- You have accessComparative Metabolic Capabilities of CYP3A4, CYP3A5, and CYP3A7J. Andrew Williams, Barbara J. Ring, Varon E. Cantrell, David R. Jones, James Eckstein, Kenneth Ruterbories, Mitchell A. Hamman, Stephen D. Hall and Steven A. WrightonDrug Metabolism and Disposition August 2002, 30 (8) 883-891; DOI: https://doi.org/10.1124/dmd.30.8.883
K
Kageyama, Akira
- You have accessAmino Acid Residues Affecting the Activities of Human Cytochrome P450 2C9 and 2C19Toshiro Niwa, Akira Kageyama, Kae Kishimoto, Yoshiyasu Yabusaki, Fumihide Ishibashi and Masanao KatagiriDrug Metabolism and Disposition August 2002, 30 (8) 931-936; DOI: https://doi.org/10.1124/dmd.30.8.931
Katagiri, Masanao
- You have accessAmino Acid Residues Affecting the Activities of Human Cytochrome P450 2C9 and 2C19Toshiro Niwa, Akira Kageyama, Kae Kishimoto, Yoshiyasu Yabusaki, Fumihide Ishibashi and Masanao KatagiriDrug Metabolism and Disposition August 2002, 30 (8) 931-936; DOI: https://doi.org/10.1124/dmd.30.8.931
Keohane, Carol-Ann
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
Kinget, R.
- You have accessIntestinal Absorption Enhancement of the Ester Prodrug Tenofovir Disoproxil Fumarate through Modulation of the Biochemical Barrier by Defined Ester MixturesJ. van Gelder, S. Deferme, L. Naesens, E. De Clercq, G. van den Mooter, R. Kinget and P. AugustijnsDrug Metabolism and Disposition August 2002, 30 (8) 924-930; DOI: https://doi.org/10.1124/dmd.30.8.924
Kishimoto, Kae
- You have accessAmino Acid Residues Affecting the Activities of Human Cytochrome P450 2C9 and 2C19Toshiro Niwa, Akira Kageyama, Kae Kishimoto, Yoshiyasu Yabusaki, Fumihide Ishibashi and Masanao KatagiriDrug Metabolism and Disposition August 2002, 30 (8) 931-936; DOI: https://doi.org/10.1124/dmd.30.8.931
Komai, Toru
- You have accessSex Difference in Inhibition of In Vitro Mexazolam Metabolism by Various 3-Hydroxy-3-Methylglutaryl-Coenzyme A Reductase Inhibitors in Rat Liver MicrosomesMichi Ishigami, Wataru Takasaki, Toshihiko Ikeda, Toru Komai, Kiyomi Ito and Yuichi SugiyamaDrug Metabolism and Disposition August 2002, 30 (8) 904-910; DOI: https://doi.org/10.1124/dmd.30.8.904
Kumar, Sanjeev
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
L
Lennard, Martin S.
- You have accessMetabolism of Tamoxifen by Recombinant Human Cytochrome P450 Enzymes: Formation of the 4-Hydroxy, 4′-Hydroxy andN-Desmethyl Metabolites and Isomerization oftrans-4-HydroxytamoxifenH. Kim Crewe, Lisa M. Notley, Rebecca M. Wunsch, Martin S. Lennard and Elizabeth M. J. GillamDrug Metabolism and Disposition August 2002, 30 (8) 869-874; DOI: https://doi.org/10.1124/dmd.30.8.869
Locker, Karen
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
M
Miyata, Masaaki
- You have accessPhenol Sulfotransferase, ST1A3, as the Main Enzyme Catalyzing Sulfation of Troglitazone in Human LiverWataru Honma, Miki Shimada, Hironobu Sasano, Shogo Ozawa, Masaaki Miyata, Kiyoshi Nagata, Toshihiko Ikeda and Yasushi YamazoeDrug Metabolism and Disposition August 2002, 30 (8) 944-949; DOI: https://doi.org/10.1124/dmd.30.8.944
Morrison, Denise
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
Mortishire-Smith, Russell
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
N
Naesens, L.
- You have accessIntestinal Absorption Enhancement of the Ester Prodrug Tenofovir Disoproxil Fumarate through Modulation of the Biochemical Barrier by Defined Ester MixturesJ. van Gelder, S. Deferme, L. Naesens, E. De Clercq, G. van den Mooter, R. Kinget and P. AugustijnsDrug Metabolism and Disposition August 2002, 30 (8) 924-930; DOI: https://doi.org/10.1124/dmd.30.8.924
Nagata, Kiyoshi
- You have accessPhenol Sulfotransferase, ST1A3, as the Main Enzyme Catalyzing Sulfation of Troglitazone in Human LiverWataru Honma, Miki Shimada, Hironobu Sasano, Shogo Ozawa, Masaaki Miyata, Kiyoshi Nagata, Toshihiko Ikeda and Yasushi YamazoeDrug Metabolism and Disposition August 2002, 30 (8) 944-949; DOI: https://doi.org/10.1124/dmd.30.8.944
Negishi, Masahiko
- You have accessRole of Constitutive Androstane Receptor in the In Vivo Induction of Mrp3 and CYP2B1/2 by PhenobarbitalHao Xiong, Kouichi Yoshinari, Kim L. R. Brouwer and Masahiko NegishiDrug Metabolism and Disposition August 2002, 30 (8) 918-923; DOI: https://doi.org/10.1124/dmd.30.8.918
Niwa, Toshiro
- You have accessAmino Acid Residues Affecting the Activities of Human Cytochrome P450 2C9 and 2C19Toshiro Niwa, Akira Kageyama, Kae Kishimoto, Yoshiyasu Yabusaki, Fumihide Ishibashi and Masanao KatagiriDrug Metabolism and Disposition August 2002, 30 (8) 931-936; DOI: https://doi.org/10.1124/dmd.30.8.931
Notley, Lisa M.
- You have accessMetabolism of Tamoxifen by Recombinant Human Cytochrome P450 Enzymes: Formation of the 4-Hydroxy, 4′-Hydroxy andN-Desmethyl Metabolites and Isomerization oftrans-4-HydroxytamoxifenH. Kim Crewe, Lisa M. Notley, Rebecca M. Wunsch, Martin S. Lennard and Elizabeth M. J. GillamDrug Metabolism and Disposition August 2002, 30 (8) 869-874; DOI: https://doi.org/10.1124/dmd.30.8.869
O
Ozawa, Shogo
- You have accessPhenol Sulfotransferase, ST1A3, as the Main Enzyme Catalyzing Sulfation of Troglitazone in Human LiverWataru Honma, Miki Shimada, Hironobu Sasano, Shogo Ozawa, Masaaki Miyata, Kiyoshi Nagata, Toshihiko Ikeda and Yasushi YamazoeDrug Metabolism and Disposition August 2002, 30 (8) 944-949; DOI: https://doi.org/10.1124/dmd.30.8.944
P
Poon, Grace K.
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
R
Raab, Conrad E.
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
Raz, Itamar
- You have accessPharmacokinetic-Pharmacodynamic Analysis of the Glucose-Lowering Effect of Metformin in Diabetic Rats Reveals First-Pass Pharmacodynamic EffectDavid Stepensky, Michael Friedman, Itamar Raz and Amnon HoffmanDrug Metabolism and Disposition August 2002, 30 (8) 861-868; DOI: https://doi.org/10.1124/dmd.30.8.861
Ring, Barbara J.
- You have accessComparative Metabolic Capabilities of CYP3A4, CYP3A5, and CYP3A7J. Andrew Williams, Barbara J. Ring, Varon E. Cantrell, David R. Jones, James Eckstein, Kenneth Ruterbories, Mitchell A. Hamman, Stephen D. Hall and Steven A. WrightonDrug Metabolism and Disposition August 2002, 30 (8) 883-891; DOI: https://doi.org/10.1124/dmd.30.8.883
Ruterbories, Kenneth
- You have accessComparative Metabolic Capabilities of CYP3A4, CYP3A5, and CYP3A7J. Andrew Williams, Barbara J. Ring, Varon E. Cantrell, David R. Jones, James Eckstein, Kenneth Ruterbories, Mitchell A. Hamman, Stephen D. Hall and Steven A. WrightonDrug Metabolism and Disposition August 2002, 30 (8) 883-891; DOI: https://doi.org/10.1124/dmd.30.8.883
S
Sasano, Hironobu
- You have accessPhenol Sulfotransferase, ST1A3, as the Main Enzyme Catalyzing Sulfation of Troglitazone in Human LiverWataru Honma, Miki Shimada, Hironobu Sasano, Shogo Ozawa, Masaaki Miyata, Kiyoshi Nagata, Toshihiko Ikeda and Yasushi YamazoeDrug Metabolism and Disposition August 2002, 30 (8) 944-949; DOI: https://doi.org/10.1124/dmd.30.8.944
Shibata, Yoshihiro
- You have accessPrediction of Hepatic Clearance and Availability by Cryopreserved Human Hepatocytes: An Application of Serum Incubation MethodYoshihiro Shibata, Hiroyuki Takahashi, Masato Chiba and Yasuyuki IshiiDrug Metabolism and Disposition August 2002, 30 (8) 892-896; DOI: https://doi.org/10.1124/dmd.30.8.892
Shimada, Miki
- You have accessPhenol Sulfotransferase, ST1A3, as the Main Enzyme Catalyzing Sulfation of Troglitazone in Human LiverWataru Honma, Miki Shimada, Hironobu Sasano, Shogo Ozawa, Masaaki Miyata, Kiyoshi Nagata, Toshihiko Ikeda and Yasushi YamazoeDrug Metabolism and Disposition August 2002, 30 (8) 944-949; DOI: https://doi.org/10.1124/dmd.30.8.944
Souid, Abdul-Kader
- You have accessKinetic Analysis of the Reactions of 4-Hydroperoxycyclophosphamide and Acrolein With Glutathione, Mesna, and Wr-1065Kirk A. Tacka, James C. Dabrowiak, Jerry Goodisman and Abdul-Kader SouidDrug Metabolism and Disposition August 2002, 30 (8) 875-882; DOI: https://doi.org/10.1124/dmd.30.8.875
Stepensky, David
- You have accessPharmacokinetic-Pharmacodynamic Analysis of the Glucose-Lowering Effect of Metformin in Diabetic Rats Reveals First-Pass Pharmacodynamic EffectDavid Stepensky, Michael Friedman, Itamar Raz and Amnon HoffmanDrug Metabolism and Disposition August 2002, 30 (8) 861-868; DOI: https://doi.org/10.1124/dmd.30.8.861
Strauss, John
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
Sugiyama, Yuichi
- You have accessSex Difference in Inhibition of In Vitro Mexazolam Metabolism by Various 3-Hydroxy-3-Methylglutaryl-Coenzyme A Reductase Inhibitors in Rat Liver MicrosomesMichi Ishigami, Wataru Takasaki, Toshihiko Ikeda, Toru Komai, Kiyomi Ito and Yuichi SugiyamaDrug Metabolism and Disposition August 2002, 30 (8) 904-910; DOI: https://doi.org/10.1124/dmd.30.8.904
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Tacka, Kirk A.
- You have accessKinetic Analysis of the Reactions of 4-Hydroperoxycyclophosphamide and Acrolein With Glutathione, Mesna, and Wr-1065Kirk A. Tacka, James C. Dabrowiak, Jerry Goodisman and Abdul-Kader SouidDrug Metabolism and Disposition August 2002, 30 (8) 875-882; DOI: https://doi.org/10.1124/dmd.30.8.875
Takahashi, Hiroyuki
- You have accessPrediction of Hepatic Clearance and Availability by Cryopreserved Human Hepatocytes: An Application of Serum Incubation MethodYoshihiro Shibata, Hiroyuki Takahashi, Masato Chiba and Yasuyuki IshiiDrug Metabolism and Disposition August 2002, 30 (8) 892-896; DOI: https://doi.org/10.1124/dmd.30.8.892
Takasaki, Wataru
- You have accessSex Difference in Inhibition of In Vitro Mexazolam Metabolism by Various 3-Hydroxy-3-Methylglutaryl-Coenzyme A Reductase Inhibitors in Rat Liver MicrosomesMichi Ishigami, Wataru Takasaki, Toshihiko Ikeda, Toru Komai, Kiyomi Ito and Yuichi SugiyamaDrug Metabolism and Disposition August 2002, 30 (8) 904-910; DOI: https://doi.org/10.1124/dmd.30.8.904
Thomas, Steven
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
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Vaidyanathan, Jaya Bharathi
- You have accessGlucuronidation and Sulfation of the Tea Flavonoid (−)-Epicatechin by the Human and Rat EnzymesJaya Bharathi Vaidyanathan and Thomas WalleDrug Metabolism and Disposition August 2002, 30 (8) 897-903; DOI: https://doi.org/10.1124/dmd.30.8.897
van den Mooter, G.
- You have accessIntestinal Absorption Enhancement of the Ester Prodrug Tenofovir Disoproxil Fumarate through Modulation of the Biochemical Barrier by Defined Ester MixturesJ. van Gelder, S. Deferme, L. Naesens, E. De Clercq, G. van den Mooter, R. Kinget and P. AugustijnsDrug Metabolism and Disposition August 2002, 30 (8) 924-930; DOI: https://doi.org/10.1124/dmd.30.8.924
van Gelder, J.
- You have accessIntestinal Absorption Enhancement of the Ester Prodrug Tenofovir Disoproxil Fumarate through Modulation of the Biochemical Barrier by Defined Ester MixturesJ. van Gelder, S. Deferme, L. Naesens, E. De Clercq, G. van den Mooter, R. Kinget and P. AugustijnsDrug Metabolism and Disposition August 2002, 30 (8) 924-930; DOI: https://doi.org/10.1124/dmd.30.8.924
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Walle, Thomas
- You have accessGlucuronidation and Sulfation of the Tea Flavonoid (−)-Epicatechin by the Human and Rat EnzymesJaya Bharathi Vaidyanathan and Thomas WalleDrug Metabolism and Disposition August 2002, 30 (8) 897-903; DOI: https://doi.org/10.1124/dmd.30.8.897
Wang, Hongbing
- You have accessCytochrome P450 2E1 (CYP2E1) is Essential for Acrylonitrile Metabolism to Cyanide: Comparative Studies Using CYP2E1-Null and Wild-Type MiceHongbing Wang, Brian Chanas and Burhan I. GhanayemDrug Metabolism and Disposition August 2002, 30 (8) 911-917; DOI: https://doi.org/10.1124/dmd.30.8.911
Wang, Yanfeng
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
Watt, Alan P.
- You have accessIdentification of Metabolites of a Substance P (Neurokinin 1 Receptor) Antagonist in Rat Hepatocytes and Rat PlasmaCornelis E. C. A. Hop, Yanfeng Wang, Sanjeev Kumar, Maria Victoria Silva Elipe, Conrad E. Raab, Dennis C. Dean, Grace K. Poon, Carol-Ann Keohane, John Strauss, Shuet-Hing L. Chiu, Neil Curtis, Jason Elliott, Ute Gerhard, Karen Locker, Denise Morrison, Russell Mortishire-Smith, Steven Thomas, Alan P. Watt and David C. EvansDrug Metabolism and Disposition August 2002, 30 (8) 937-943; DOI: https://doi.org/10.1124/dmd.30.8.937
Williams, J. Andrew
- You have accessComparative Metabolic Capabilities of CYP3A4, CYP3A5, and CYP3A7J. Andrew Williams, Barbara J. Ring, Varon E. Cantrell, David R. Jones, James Eckstein, Kenneth Ruterbories, Mitchell A. Hamman, Stephen D. Hall and Steven A. WrightonDrug Metabolism and Disposition August 2002, 30 (8) 883-891; DOI: https://doi.org/10.1124/dmd.30.8.883
Wrighton, Steven A.
- You have accessComparative Metabolic Capabilities of CYP3A4, CYP3A5, and CYP3A7J. Andrew Williams, Barbara J. Ring, Varon E. Cantrell, David R. Jones, James Eckstein, Kenneth Ruterbories, Mitchell A. Hamman, Stephen D. Hall and Steven A. WrightonDrug Metabolism and Disposition August 2002, 30 (8) 883-891; DOI: https://doi.org/10.1124/dmd.30.8.883
Wunsch, Rebecca M.
- You have accessMetabolism of Tamoxifen by Recombinant Human Cytochrome P450 Enzymes: Formation of the 4-Hydroxy, 4′-Hydroxy andN-Desmethyl Metabolites and Isomerization oftrans-4-HydroxytamoxifenH. Kim Crewe, Lisa M. Notley, Rebecca M. Wunsch, Martin S. Lennard and Elizabeth M. J. GillamDrug Metabolism and Disposition August 2002, 30 (8) 869-874; DOI: https://doi.org/10.1124/dmd.30.8.869
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Xiong, Hao
- You have accessRole of Constitutive Androstane Receptor in the In Vivo Induction of Mrp3 and CYP2B1/2 by PhenobarbitalHao Xiong, Kouichi Yoshinari, Kim L. R. Brouwer and Masahiko NegishiDrug Metabolism and Disposition August 2002, 30 (8) 918-923; DOI: https://doi.org/10.1124/dmd.30.8.918
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Yabusaki, Yoshiyasu
- You have accessAmino Acid Residues Affecting the Activities of Human Cytochrome P450 2C9 and 2C19Toshiro Niwa, Akira Kageyama, Kae Kishimoto, Yoshiyasu Yabusaki, Fumihide Ishibashi and Masanao KatagiriDrug Metabolism and Disposition August 2002, 30 (8) 931-936; DOI: https://doi.org/10.1124/dmd.30.8.931
Yamazoe, Yasushi
- You have accessPhenol Sulfotransferase, ST1A3, as the Main Enzyme Catalyzing Sulfation of Troglitazone in Human LiverWataru Honma, Miki Shimada, Hironobu Sasano, Shogo Ozawa, Masaaki Miyata, Kiyoshi Nagata, Toshihiko Ikeda and Yasushi YamazoeDrug Metabolism and Disposition August 2002, 30 (8) 944-949; DOI: https://doi.org/10.1124/dmd.30.8.944
Yoshinari, Kouichi
- You have accessRole of Constitutive Androstane Receptor in the In Vivo Induction of Mrp3 and CYP2B1/2 by PhenobarbitalHao Xiong, Kouichi Yoshinari, Kim L. R. Brouwer and Masahiko NegishiDrug Metabolism and Disposition August 2002, 30 (8) 918-923; DOI: https://doi.org/10.1124/dmd.30.8.918