Index by author
September 01, 2003; Volume 31,Issue 9
B
Bajpai, Manoj
- You have accessONLY TRUNCATED, NOT COMPLETE CYTOCHROME P450 2D6 RNA TRANSCRIPT AND NO DETECTABLE ENZYME ACTIVITY ARE EXPRESSED IN HUMAN LYMPHOCYTESLisa A. McConnachie, Brian Phillips, Manoj Bajpai, Danny D. Shen and Rodney J. Y. HoDrug Metabolism and Disposition September 2003, 31 (9) 1103-1107; DOI: https://doi.org/10.1124/dmd.31.9.1103
Bedard, Leanne L.
- You have accessBIOTRANSFORMATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE (NNK) IN PERIPHERAL HUMAN LUNG MICROSOMESGraeme B. J. Smith, John R. Bend, Leanne L. Bedard, Ken R. Reid, Dimitri Petsikas and Thomas E. MasseyDrug Metabolism and Disposition September 2003, 31 (9) 1134-1141; DOI: https://doi.org/10.1124/dmd.31.9.1134
Bend, John R.
- You have accessBIOTRANSFORMATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE (NNK) IN PERIPHERAL HUMAN LUNG MICROSOMESGraeme B. J. Smith, John R. Bend, Leanne L. Bedard, Ken R. Reid, Dimitri Petsikas and Thomas E. MasseyDrug Metabolism and Disposition September 2003, 31 (9) 1134-1141; DOI: https://doi.org/10.1124/dmd.31.9.1134
Benedek, Irma H.
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Berbaum, Jennifer
- You have accessGENERATION AND VALIDATION OF RAPID COMPUTATIONAL FILTERS FOR CYP2D6 AND CYP3A4Sean Ekins, Jennifer Berbaum and Richard K. HarrisonDrug Metabolism and Disposition September 2003, 31 (9) 1077-1080; DOI: https://doi.org/10.1124/dmd.31.9.1077
Boobis, Alan R.
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Brennan, James M.
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Burchell, Brian
- You have accessCONJUGATION OF CATECHOLS BY RECOMBINANT HUMAN SULFOTRANSFERASES, UDP-GLUCURONOSYLTRANSFERASES, AND SOLUBLE CATECHOL O-METHYLTRANSFERASE: STRUCTURE-CONJUGATION RELATIONSHIPS AND PREDICTIVE MODELSJyrki Taskinen, Brian T. Ethell, Pia Pihlavisto, Alan M. Hood, Brian Burchell and Michael W. H. CoughtrieDrug Metabolism and Disposition September 2003, 31 (9) 1187-1197; DOI: https://doi.org/10.1124/dmd.31.9.1187
C
Caggana, Michele
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS OF THE HUMAN CYP2A13 GENE: EVIDENCE FOR A NULL ALLELEXiuling Zhang, Ying Chen, Yiqin Liu, Xiang Ren, Qing-Yu Zhang, Michele Caggana and Xinxin DingDrug Metabolism and Disposition September 2003, 31 (9) 1081-1085; DOI: https://doi.org/10.1124/dmd.31.9.1081
Castell, José V.
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Charman, William N.
- You have accessAPPLICATION OF COMPARTMENTAL MODELING TO AN EXAMINATION OF IN VITRO INTESTINAL PERMEABILITY DATA: ASSESSING THE IMPACT OF TISSUE UPTAKE, P-GLYCOPROTEIN, AND CYP3ABrendan M. Johnson, William N. Charman and Christopher J. H. PorterDrug Metabolism and Disposition September 2003, 31 (9) 1151-1160; DOI: https://doi.org/10.1124/dmd.31.9.1151
Chen, Ying
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS OF THE HUMAN CYP2A13 GENE: EVIDENCE FOR A NULL ALLELEXiuling Zhang, Ying Chen, Yiqin Liu, Xiang Ren, Qing-Yu Zhang, Michele Caggana and Xinxin DingDrug Metabolism and Disposition September 2003, 31 (9) 1081-1085; DOI: https://doi.org/10.1124/dmd.31.9.1081
Cherrington, N. J.
- You have accessINDUCTION OF MULTIDRUG RESISTANCE PROTEIN 3 IN RAT LIVER IS ASSOCIATED WITH ALTERED VECTORIAL EXCRETION OF ACETAMINOPHEN METABOLITESA. L. Slitt, N. J. Cherrington, J. M. Maher and C. D. KlaassenDrug Metabolism and Disposition September 2003, 31 (9) 1176-1186; DOI: https://doi.org/10.1124/dmd.31.9.1176
Clarke, Stephen E.
- You have accessMULTISITE KINETIC ANALYSIS OF INTERACTIONS BETWEEN PROTOTYPICAL CYP3A4 SUBGROUP SUBSTRATES: MIDAZOLAM, TESTOSTERONE, AND NIFEDIPINEAleksandra Galetin, Stephen E. Clarke and J. Brian HoustonDrug Metabolism and Disposition September 2003, 31 (9) 1108-1116; DOI: https://doi.org/10.1124/dmd.31.9.1108
Corcos, Laurent
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Coughtrie, Michael W. H.
- You have accessCONJUGATION OF CATECHOLS BY RECOMBINANT HUMAN SULFOTRANSFERASES, UDP-GLUCURONOSYLTRANSFERASES, AND SOLUBLE CATECHOL O-METHYLTRANSFERASE: STRUCTURE-CONJUGATION RELATIONSHIPS AND PREDICTIVE MODELSJyrki Taskinen, Brian T. Ethell, Pia Pihlavisto, Alan M. Hood, Brian Burchell and Michael W. H. CoughtrieDrug Metabolism and Disposition September 2003, 31 (9) 1187-1197; DOI: https://doi.org/10.1124/dmd.31.9.1187
Court, Michael H.
- You have accessEVALUATION OF 3′-AZIDO-3′-DEOXYTHYMIDINE, MORPHINE, AND CODEINE AS PROBE SUBSTRATES FOR UDP-GLUCURONOSYLTRANSFERASE 2B7 (UGT2B7) IN HUMAN LIVER MICROSOMES: SPECIFICITY AND INFLUENCE OF THE UGT2B7*2 POLYMORPHISMMichael H. Court, Soundarajan Krishnaswamy, Qin Hao, Su X. Duan, Christopher J. Patten, Lisa L. von Moltke and David J. GreenblattDrug Metabolism and Disposition September 2003, 31 (9) 1125-1133; DOI: https://doi.org/10.1124/dmd.31.9.1125
D
Dai, Renke
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Ding, Xinxin
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS OF THE HUMAN CYP2A13 GENE: EVIDENCE FOR A NULL ALLELEXiuling Zhang, Ying Chen, Yiqin Liu, Xiang Ren, Qing-Yu Zhang, Michele Caggana and Xinxin DingDrug Metabolism and Disposition September 2003, 31 (9) 1081-1085; DOI: https://doi.org/10.1124/dmd.31.9.1081
Duan, Su X.
- You have accessEVALUATION OF 3′-AZIDO-3′-DEOXYTHYMIDINE, MORPHINE, AND CODEINE AS PROBE SUBSTRATES FOR UDP-GLUCURONOSYLTRANSFERASE 2B7 (UGT2B7) IN HUMAN LIVER MICROSOMES: SPECIFICITY AND INFLUENCE OF THE UGT2B7*2 POLYMORPHISMMichael H. Court, Soundarajan Krishnaswamy, Qin Hao, Su X. Duan, Christopher J. Patten, Lisa L. von Moltke and David J. GreenblattDrug Metabolism and Disposition September 2003, 31 (9) 1125-1133; DOI: https://doi.org/10.1124/dmd.31.9.1125
E
Edwards, Robert J.
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Ekins, Sean
- You have accessGENERATION AND VALIDATION OF RAPID COMPUTATIONAL FILTERS FOR CYP2D6 AND CYP3A4Sean Ekins, Jennifer Berbaum and Richard K. HarrisonDrug Metabolism and Disposition September 2003, 31 (9) 1077-1080; DOI: https://doi.org/10.1124/dmd.31.9.1077
Ethell, Brian T.
- You have accessCONJUGATION OF CATECHOLS BY RECOMBINANT HUMAN SULFOTRANSFERASES, UDP-GLUCURONOSYLTRANSFERASES, AND SOLUBLE CATECHOL O-METHYLTRANSFERASE: STRUCTURE-CONJUGATION RELATIONSHIPS AND PREDICTIVE MODELSJyrki Taskinen, Brian T. Ethell, Pia Pihlavisto, Alan M. Hood, Brian Burchell and Michael W. H. CoughtrieDrug Metabolism and Disposition September 2003, 31 (9) 1187-1197; DOI: https://doi.org/10.1124/dmd.31.9.1187
F
Finel, Moshe
- You have accessGLUCURONIDATION OF ANABOLIC ANDROGENIC STEROIDS BY RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESTiia Kuuranne, Mika Kurkela, Mario Thevis, Wilhelm Schänzer, Moshe Finel and Risto KostiainenDrug Metabolism and Disposition September 2003, 31 (9) 1117-1124; DOI: https://doi.org/10.1124/dmd.31.9.1117
Fiske, William D.
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
G
Galetin, Aleksandra
- You have accessISOFORM SELECTIVITY AND KINETICS OF MORPHINE 3- AND 6-GLUCURONIDATION BY HUMAN UDP-GLUCURONOSYLTRANSFERASES: EVIDENCE FOR ATYPICAL GLUCURONIDATION KINETICS BY UGT2B7Andrew N. Stone, Peter I. Mackenzie, Aleksandra Galetin, J. Brian Houston and John O. MinersDrug Metabolism and Disposition September 2003, 31 (9) 1086-1089; DOI: https://doi.org/10.1124/dmd.31.9.1086
- You have accessMULTISITE KINETIC ANALYSIS OF INTERACTIONS BETWEEN PROTOTYPICAL CYP3A4 SUBGROUP SUBSTRATES: MIDAZOLAM, TESTOSTERONE, AND NIFEDIPINEAleksandra Galetin, Stephen E. Clarke and J. Brian HoustonDrug Metabolism and Disposition September 2003, 31 (9) 1108-1116; DOI: https://doi.org/10.1124/dmd.31.9.1108
Gan, Liang-Shang
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Gilbert, Darryl
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Gillespie, T. A.
- You have accessMETABOLISM, EXCRETION, AND PHARMACOKINETICS OF DULOXETINE IN HEALTHY HUMAN SUBJECTSR. J. Lantz, T. A. Gillespie, T. J. Rash, F. Kuo, M. Skinner, H-Y. Kuan and M. P. KnadlerDrug Metabolism and Disposition September 2003, 31 (9) 1142-1150; DOI: https://doi.org/10.1124/dmd.31.9.1142
Goldfarb, Peter S.
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Gómez-Lechón, Maria-José
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Greenblatt, David J.
- You have accessEVALUATION OF 3′-AZIDO-3′-DEOXYTHYMIDINE, MORPHINE, AND CODEINE AS PROBE SUBSTRATES FOR UDP-GLUCURONOSYLTRANSFERASE 2B7 (UGT2B7) IN HUMAN LIVER MICROSOMES: SPECIFICITY AND INFLUENCE OF THE UGT2B7*2 POLYMORPHISMMichael H. Court, Soundarajan Krishnaswamy, Qin Hao, Su X. Duan, Christopher J. Patten, Lisa L. von Moltke and David J. GreenblattDrug Metabolism and Disposition September 2003, 31 (9) 1125-1133; DOI: https://doi.org/10.1124/dmd.31.9.1125
Guillouzo, Andre
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
H
Hao, Qin
- You have accessEVALUATION OF 3′-AZIDO-3′-DEOXYTHYMIDINE, MORPHINE, AND CODEINE AS PROBE SUBSTRATES FOR UDP-GLUCURONOSYLTRANSFERASE 2B7 (UGT2B7) IN HUMAN LIVER MICROSOMES: SPECIFICITY AND INFLUENCE OF THE UGT2B7*2 POLYMORPHISMMichael H. Court, Soundarajan Krishnaswamy, Qin Hao, Su X. Duan, Christopher J. Patten, Lisa L. von Moltke and David J. GreenblattDrug Metabolism and Disposition September 2003, 31 (9) 1125-1133; DOI: https://doi.org/10.1124/dmd.31.9.1125
Harrison, Richard K.
- You have accessGENERATION AND VALIDATION OF RAPID COMPUTATIONAL FILTERS FOR CYP2D6 AND CYP3A4Sean Ekins, Jennifer Berbaum and Richard K. HarrisonDrug Metabolism and Disposition September 2003, 31 (9) 1077-1080; DOI: https://doi.org/10.1124/dmd.31.9.1077
Hidestrand, Mats
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Hines, Ronald N.
- You have accessPUBLICATION OF STAND-ALONE SINGLE NUCLEOTIDE POLYMORPHISM (SNP) DISCOVERY DATARonald N. HinesDrug Metabolism and Disposition September 2003, 31 (9) 1073; DOI: https://doi.org/10.1124/dmd.31.9.1073
Ho, Rodney J. Y.
- You have accessONLY TRUNCATED, NOT COMPLETE CYTOCHROME P450 2D6 RNA TRANSCRIPT AND NO DETECTABLE ENZYME ACTIVITY ARE EXPRESSED IN HUMAN LYMPHOCYTESLisa A. McConnachie, Brian Phillips, Manoj Bajpai, Danny D. Shen and Rodney J. Y. HoDrug Metabolism and Disposition September 2003, 31 (9) 1103-1107; DOI: https://doi.org/10.1124/dmd.31.9.1103
Hood, Alan M.
- You have accessCONJUGATION OF CATECHOLS BY RECOMBINANT HUMAN SULFOTRANSFERASES, UDP-GLUCURONOSYLTRANSFERASES, AND SOLUBLE CATECHOL O-METHYLTRANSFERASE: STRUCTURE-CONJUGATION RELATIONSHIPS AND PREDICTIVE MODELSJyrki Taskinen, Brian T. Ethell, Pia Pihlavisto, Alan M. Hood, Brian Burchell and Michael W. H. CoughtrieDrug Metabolism and Disposition September 2003, 31 (9) 1187-1197; DOI: https://doi.org/10.1124/dmd.31.9.1187
Houston, J. Brian
- You have accessISOFORM SELECTIVITY AND KINETICS OF MORPHINE 3- AND 6-GLUCURONIDATION BY HUMAN UDP-GLUCURONOSYLTRANSFERASES: EVIDENCE FOR ATYPICAL GLUCURONIDATION KINETICS BY UGT2B7Andrew N. Stone, Peter I. Mackenzie, Aleksandra Galetin, J. Brian Houston and John O. MinersDrug Metabolism and Disposition September 2003, 31 (9) 1086-1089; DOI: https://doi.org/10.1124/dmd.31.9.1086
- You have accessMULTISITE KINETIC ANALYSIS OF INTERACTIONS BETWEEN PROTOTYPICAL CYP3A4 SUBGROUP SUBSTRATES: MIDAZOLAM, TESTOSTERONE, AND NIFEDIPINEAleksandra Galetin, Stephen E. Clarke and J. Brian HoustonDrug Metabolism and Disposition September 2003, 31 (9) 1108-1116; DOI: https://doi.org/10.1124/dmd.31.9.1108
I
Ingelman-Sundberg, Magnus
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
J
Johnson, Brendan M.
- You have accessAPPLICATION OF COMPARTMENTAL MODELING TO AN EXAMINATION OF IN VITRO INTESTINAL PERMEABILITY DATA: ASSESSING THE IMPACT OF TISSUE UPTAKE, P-GLYCOPROTEIN, AND CYP3ABrendan M. Johnson, William N. Charman and Christopher J. H. PorterDrug Metabolism and Disposition September 2003, 31 (9) 1151-1160; DOI: https://doi.org/10.1124/dmd.31.9.1151
Jolley, Summer
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
K
Kim, Kyoung-Ah
- You have accessINHIBITORY EFFECT OF GLYBURIDE ON HUMAN CYTOCHROME P450 ISOFORMS IN HUMAN LIVER MICROSOMESKyoung-Ah Kim and Ji-Young ParkDrug Metabolism and Disposition September 2003, 31 (9) 1090-1092; DOI: https://doi.org/10.1124/dmd.31.9.1090
Kim, Sean
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Klaassen, C. D.
- You have accessINDUCTION OF MULTIDRUG RESISTANCE PROTEIN 3 IN RAT LIVER IS ASSOCIATED WITH ALTERED VECTORIAL EXCRETION OF ACETAMINOPHEN METABOLITESA. L. Slitt, N. J. Cherrington, J. M. Maher and C. D. KlaassenDrug Metabolism and Disposition September 2003, 31 (9) 1176-1186; DOI: https://doi.org/10.1124/dmd.31.9.1176
Knadler, M. P.
- You have accessMETABOLISM, EXCRETION, AND PHARMACOKINETICS OF DULOXETINE IN HEALTHY HUMAN SUBJECTSR. J. Lantz, T. A. Gillespie, T. J. Rash, F. Kuo, M. Skinner, H-Y. Kuan and M. P. KnadlerDrug Metabolism and Disposition September 2003, 31 (9) 1142-1150; DOI: https://doi.org/10.1124/dmd.31.9.1142
Kostiainen, Risto
- You have accessGLUCURONIDATION OF ANABOLIC ANDROGENIC STEROIDS BY RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESTiia Kuuranne, Mika Kurkela, Mario Thevis, Wilhelm Schänzer, Moshe Finel and Risto KostiainenDrug Metabolism and Disposition September 2003, 31 (9) 1117-1124; DOI: https://doi.org/10.1124/dmd.31.9.1117
Krishnaswamy, Soundarajan
- You have accessEVALUATION OF 3′-AZIDO-3′-DEOXYTHYMIDINE, MORPHINE, AND CODEINE AS PROBE SUBSTRATES FOR UDP-GLUCURONOSYLTRANSFERASE 2B7 (UGT2B7) IN HUMAN LIVER MICROSOMES: SPECIFICITY AND INFLUENCE OF THE UGT2B7*2 POLYMORPHISMMichael H. Court, Soundarajan Krishnaswamy, Qin Hao, Su X. Duan, Christopher J. Patten, Lisa L. von Moltke and David J. GreenblattDrug Metabolism and Disposition September 2003, 31 (9) 1125-1133; DOI: https://doi.org/10.1124/dmd.31.9.1125
Kuan, H-Y.
- You have accessMETABOLISM, EXCRETION, AND PHARMACOKINETICS OF DULOXETINE IN HEALTHY HUMAN SUBJECTSR. J. Lantz, T. A. Gillespie, T. J. Rash, F. Kuo, M. Skinner, H-Y. Kuan and M. P. KnadlerDrug Metabolism and Disposition September 2003, 31 (9) 1142-1150; DOI: https://doi.org/10.1124/dmd.31.9.1142
Kuo, F.
- You have accessMETABOLISM, EXCRETION, AND PHARMACOKINETICS OF DULOXETINE IN HEALTHY HUMAN SUBJECTSR. J. Lantz, T. A. Gillespie, T. J. Rash, F. Kuo, M. Skinner, H-Y. Kuan and M. P. KnadlerDrug Metabolism and Disposition September 2003, 31 (9) 1142-1150; DOI: https://doi.org/10.1124/dmd.31.9.1142
Kurkela, Mika
- You have accessGLUCURONIDATION OF ANABOLIC ANDROGENIC STEROIDS BY RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESTiia Kuuranne, Mika Kurkela, Mario Thevis, Wilhelm Schänzer, Moshe Finel and Risto KostiainenDrug Metabolism and Disposition September 2003, 31 (9) 1117-1124; DOI: https://doi.org/10.1124/dmd.31.9.1117
Kuuranne, Tiia
- You have accessGLUCURONIDATION OF ANABOLIC ANDROGENIC STEROIDS BY RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESTiia Kuuranne, Mika Kurkela, Mario Thevis, Wilhelm Schänzer, Moshe Finel and Risto KostiainenDrug Metabolism and Disposition September 2003, 31 (9) 1117-1124; DOI: https://doi.org/10.1124/dmd.31.9.1117
L
Lake, Brian G.
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Lantz, R. J.
- You have accessMETABOLISM, EXCRETION, AND PHARMACOKINETICS OF DULOXETINE IN HEALTHY HUMAN SUBJECTSR. J. Lantz, T. A. Gillespie, T. J. Rash, F. Kuo, M. Skinner, H-Y. Kuan and M. P. KnadlerDrug Metabolism and Disposition September 2003, 31 (9) 1142-1150; DOI: https://doi.org/10.1124/dmd.31.9.1142
LeCluyse, Edward
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Lee, Frank W.
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Lewis, David F.V.
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Li, Yinghe
- You have accessSUBSTRATE SPECIFICITY AND KINETIC PROPERTIES OF SEVEN HETEROLOGOUSLY EXPRESSED DOG CYTOCHROMES P450Magang Shou, Ryan Norcross, Grit Sandig, Ping Lu, Yinghe Li, Yuh Lin, Qin Mei, A. David Rodrigues and Thomas H. RushmoreDrug Metabolism and Disposition September 2003, 31 (9) 1161-1169; DOI: https://doi.org/10.1124/dmd.31.9.1161
Lin, Jianrong
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Lin, Yuh
- You have accessSUBSTRATE SPECIFICITY AND KINETIC PROPERTIES OF SEVEN HETEROLOGOUSLY EXPRESSED DOG CYTOCHROMES P450Magang Shou, Ryan Norcross, Grit Sandig, Ping Lu, Yinghe Li, Yuh Lin, Qin Mei, A. David Rodrigues and Thomas H. RushmoreDrug Metabolism and Disposition September 2003, 31 (9) 1161-1169; DOI: https://doi.org/10.1124/dmd.31.9.1161
Liu, Yiqin
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS OF THE HUMAN CYP2A13 GENE: EVIDENCE FOR A NULL ALLELEXiuling Zhang, Ying Chen, Yiqin Liu, Xiang Ren, Qing-Yu Zhang, Michele Caggana and Xinxin DingDrug Metabolism and Disposition September 2003, 31 (9) 1081-1085; DOI: https://doi.org/10.1124/dmd.31.9.1081
Lu, Ping
- You have accessSUBSTRATE SPECIFICITY AND KINETIC PROPERTIES OF SEVEN HETEROLOGOUSLY EXPRESSED DOG CYTOCHROMES P450Magang Shou, Ryan Norcross, Grit Sandig, Ping Lu, Yinghe Li, Yuh Lin, Qin Mei, A. David Rodrigues and Thomas H. RushmoreDrug Metabolism and Disposition September 2003, 31 (9) 1161-1169; DOI: https://doi.org/10.1124/dmd.31.9.1161
Luo, Gang
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
M
Mackenzie, Peter I.
- You have accessISOFORM SELECTIVITY AND KINETICS OF MORPHINE 3- AND 6-GLUCURONIDATION BY HUMAN UDP-GLUCURONOSYLTRANSFERASES: EVIDENCE FOR ATYPICAL GLUCURONIDATION KINETICS BY UGT2B7Andrew N. Stone, Peter I. Mackenzie, Aleksandra Galetin, J. Brian Houston and John O. MinersDrug Metabolism and Disposition September 2003, 31 (9) 1086-1089; DOI: https://doi.org/10.1124/dmd.31.9.1086
Maher, J. M.
- You have accessINDUCTION OF MULTIDRUG RESISTANCE PROTEIN 3 IN RAT LIVER IS ASSOCIATED WITH ALTERED VECTORIAL EXCRETION OF ACETAMINOPHEN METABOLITESA. L. Slitt, N. J. Cherrington, J. M. Maher and C. D. KlaassenDrug Metabolism and Disposition September 2003, 31 (9) 1176-1186; DOI: https://doi.org/10.1124/dmd.31.9.1176
Massey, Thomas E.
- You have accessBIOTRANSFORMATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE (NNK) IN PERIPHERAL HUMAN LUNG MICROSOMESGraeme B. J. Smith, John R. Bend, Leanne L. Bedard, Ken R. Reid, Dimitri Petsikas and Thomas E. MasseyDrug Metabolism and Disposition September 2003, 31 (9) 1134-1141; DOI: https://doi.org/10.1124/dmd.31.9.1134
McConnachie, Lisa A.
- You have accessONLY TRUNCATED, NOT COMPLETE CYTOCHROME P450 2D6 RNA TRANSCRIPT AND NO DETECTABLE ENZYME ACTIVITY ARE EXPRESSED IN HUMAN LYMPHOCYTESLisa A. McConnachie, Brian Phillips, Manoj Bajpai, Danny D. Shen and Rodney J. Y. HoDrug Metabolism and Disposition September 2003, 31 (9) 1103-1107; DOI: https://doi.org/10.1124/dmd.31.9.1103
Mei, Qin
- You have accessSUBSTRATE SPECIFICITY AND KINETIC PROPERTIES OF SEVEN HETEROLOGOUSLY EXPRESSED DOG CYTOCHROMES P450Magang Shou, Ryan Norcross, Grit Sandig, Ping Lu, Yinghe Li, Yuh Lin, Qin Mei, A. David Rodrigues and Thomas H. RushmoreDrug Metabolism and Disposition September 2003, 31 (9) 1161-1169; DOI: https://doi.org/10.1124/dmd.31.9.1161
Miners, John O.
- You have accessISOFORM SELECTIVITY AND KINETICS OF MORPHINE 3- AND 6-GLUCURONIDATION BY HUMAN UDP-GLUCURONOSYLTRANSFERASES: EVIDENCE FOR ATYPICAL GLUCURONIDATION KINETICS BY UGT2B7Andrew N. Stone, Peter I. Mackenzie, Aleksandra Galetin, J. Brian Houston and John O. MinersDrug Metabolism and Disposition September 2003, 31 (9) 1086-1089; DOI: https://doi.org/10.1124/dmd.31.9.1086
N
Norcross, Ryan
- You have accessSUBSTRATE SPECIFICITY AND KINETIC PROPERTIES OF SEVEN HETEROLOGOUSLY EXPRESSED DOG CYTOCHROMES P450Magang Shou, Ryan Norcross, Grit Sandig, Ping Lu, Yinghe Li, Yuh Lin, Qin Mei, A. David Rodrigues and Thomas H. RushmoreDrug Metabolism and Disposition September 2003, 31 (9) 1161-1169; DOI: https://doi.org/10.1124/dmd.31.9.1161
Nyman, Leena
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
P
Park, Ji-Young
- You have accessINHIBITORY EFFECT OF GLYBURIDE ON HUMAN CYTOCHROME P450 ISOFORMS IN HUMAN LIVER MICROSOMESKyoung-Ah Kim and Ji-Young ParkDrug Metabolism and Disposition September 2003, 31 (9) 1090-1092; DOI: https://doi.org/10.1124/dmd.31.9.1090
Patten, Christopher J.
- You have accessEVALUATION OF 3′-AZIDO-3′-DEOXYTHYMIDINE, MORPHINE, AND CODEINE AS PROBE SUBSTRATES FOR UDP-GLUCURONOSYLTRANSFERASE 2B7 (UGT2B7) IN HUMAN LIVER MICROSOMES: SPECIFICITY AND INFLUENCE OF THE UGT2B7*2 POLYMORPHISMMichael H. Court, Soundarajan Krishnaswamy, Qin Hao, Su X. Duan, Christopher J. Patten, Lisa L. von Moltke and David J. GreenblattDrug Metabolism and Disposition September 2003, 31 (9) 1125-1133; DOI: https://doi.org/10.1124/dmd.31.9.1125
Pelkonen, Olavi
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Periandythevar, Parameswaran
- You have accessSPURIOUS OBSERVATION OF SPLENIC CYP2B1 EXPRESSIONMeena R. Sharma, Parameswaran Periandythevar and Bernard H. ShapiroDrug Metabolism and Disposition September 2003, 31 (9) 1074-1076; DOI: https://doi.org/10.1124/dmd.31.9.1074
Petsikas, Dimitri
- You have accessBIOTRANSFORMATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE (NNK) IN PERIPHERAL HUMAN LUNG MICROSOMESGraeme B. J. Smith, John R. Bend, Leanne L. Bedard, Ken R. Reid, Dimitri Petsikas and Thomas E. MasseyDrug Metabolism and Disposition September 2003, 31 (9) 1134-1141; DOI: https://doi.org/10.1124/dmd.31.9.1134
Phillips, Brian
- You have accessONLY TRUNCATED, NOT COMPLETE CYTOCHROME P450 2D6 RNA TRANSCRIPT AND NO DETECTABLE ENZYME ACTIVITY ARE EXPRESSED IN HUMAN LYMPHOCYTESLisa A. McConnachie, Brian Phillips, Manoj Bajpai, Danny D. Shen and Rodney J. Y. HoDrug Metabolism and Disposition September 2003, 31 (9) 1103-1107; DOI: https://doi.org/10.1124/dmd.31.9.1103
Pihlavisto, Pia
- You have accessCONJUGATION OF CATECHOLS BY RECOMBINANT HUMAN SULFOTRANSFERASES, UDP-GLUCURONOSYLTRANSFERASES, AND SOLUBLE CATECHOL O-METHYLTRANSFERASE: STRUCTURE-CONJUGATION RELATIONSHIPS AND PREDICTIVE MODELSJyrki Taskinen, Brian T. Ethell, Pia Pihlavisto, Alan M. Hood, Brian Burchell and Michael W. H. CoughtrieDrug Metabolism and Disposition September 2003, 31 (9) 1187-1197; DOI: https://doi.org/10.1124/dmd.31.9.1187
Porter, Christopher J. H.
- You have accessAPPLICATION OF COMPARTMENTAL MODELING TO AN EXAMINATION OF IN VITRO INTESTINAL PERMEABILITY DATA: ASSESSING THE IMPACT OF TISSUE UPTAKE, P-GLYCOPROTEIN, AND CYP3ABrendan M. Johnson, William N. Charman and Christopher J. H. PorterDrug Metabolism and Disposition September 2003, 31 (9) 1151-1160; DOI: https://doi.org/10.1124/dmd.31.9.1151
Price, Roger J.
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
R
Rash, T. J.
- You have accessMETABOLISM, EXCRETION, AND PHARMACOKINETICS OF DULOXETINE IN HEALTHY HUMAN SUBJECTSR. J. Lantz, T. A. Gillespie, T. J. Rash, F. Kuo, M. Skinner, H-Y. Kuan and M. P. KnadlerDrug Metabolism and Disposition September 2003, 31 (9) 1142-1150; DOI: https://doi.org/10.1124/dmd.31.9.1142
Reid, Ken R.
- You have accessBIOTRANSFORMATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE (NNK) IN PERIPHERAL HUMAN LUNG MICROSOMESGraeme B. J. Smith, John R. Bend, Leanne L. Bedard, Ken R. Reid, Dimitri Petsikas and Thomas E. MasseyDrug Metabolism and Disposition September 2003, 31 (9) 1134-1141; DOI: https://doi.org/10.1124/dmd.31.9.1134
Ren, Xiang
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS OF THE HUMAN CYP2A13 GENE: EVIDENCE FOR A NULL ALLELEXiuling Zhang, Ying Chen, Yiqin Liu, Xiang Ren, Qing-Yu Zhang, Michele Caggana and Xinxin DingDrug Metabolism and Disposition September 2003, 31 (9) 1081-1085; DOI: https://doi.org/10.1124/dmd.31.9.1081
Renwick, Anthony B.
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Rodrigues, A. David
- You have accessSUBSTRATE SPECIFICITY AND KINETIC PROPERTIES OF SEVEN HETEROLOGOUSLY EXPRESSED DOG CYTOCHROMES P450Magang Shou, Ryan Norcross, Grit Sandig, Ping Lu, Yinghe Li, Yuh Lin, Qin Mei, A. David Rodrigues and Thomas H. RushmoreDrug Metabolism and Disposition September 2003, 31 (9) 1161-1169; DOI: https://doi.org/10.1124/dmd.31.9.1161
Rushmore, Thomas H.
- You have accessSUBSTRATE SPECIFICITY AND KINETIC PROPERTIES OF SEVEN HETEROLOGOUSLY EXPRESSED DOG CYTOCHROMES P450Magang Shou, Ryan Norcross, Grit Sandig, Ping Lu, Yinghe Li, Yuh Lin, Qin Mei, A. David Rodrigues and Thomas H. RushmoreDrug Metabolism and Disposition September 2003, 31 (9) 1161-1169; DOI: https://doi.org/10.1124/dmd.31.9.1161
S
Salonen, Jarmo S.
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Sandig, Grit
- You have accessSUBSTRATE SPECIFICITY AND KINETIC PROPERTIES OF SEVEN HETEROLOGOUSLY EXPRESSED DOG CYTOCHROMES P450Magang Shou, Ryan Norcross, Grit Sandig, Ping Lu, Yinghe Li, Yuh Lin, Qin Mei, A. David Rodrigues and Thomas H. RushmoreDrug Metabolism and Disposition September 2003, 31 (9) 1161-1169; DOI: https://doi.org/10.1124/dmd.31.9.1161
Schänzer, Wilhelm
- You have accessGLUCURONIDATION OF ANABOLIC ANDROGENIC STEROIDS BY RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESTiia Kuuranne, Mika Kurkela, Mario Thevis, Wilhelm Schänzer, Moshe Finel and Risto KostiainenDrug Metabolism and Disposition September 2003, 31 (9) 1117-1124; DOI: https://doi.org/10.1124/dmd.31.9.1117
Shapiro, Bernard H.
- You have accessSPURIOUS OBSERVATION OF SPLENIC CYP2B1 EXPRESSIONMeena R. Sharma, Parameswaran Periandythevar and Bernard H. ShapiroDrug Metabolism and Disposition September 2003, 31 (9) 1074-1076; DOI: https://doi.org/10.1124/dmd.31.9.1074
Sharma, Meena R.
- You have accessSPURIOUS OBSERVATION OF SPLENIC CYP2B1 EXPRESSIONMeena R. Sharma, Parameswaran Periandythevar and Bernard H. ShapiroDrug Metabolism and Disposition September 2003, 31 (9) 1074-1076; DOI: https://doi.org/10.1124/dmd.31.9.1074
Shen, Danny D.
- You have accessONLY TRUNCATED, NOT COMPLETE CYTOCHROME P450 2D6 RNA TRANSCRIPT AND NO DETECTABLE ENZYME ACTIVITY ARE EXPRESSED IN HUMAN LYMPHOCYTESLisa A. McConnachie, Brian Phillips, Manoj Bajpai, Danny D. Shen and Rodney J. Y. HoDrug Metabolism and Disposition September 2003, 31 (9) 1103-1107; DOI: https://doi.org/10.1124/dmd.31.9.1103
Shou, Magang
- You have accessSUBSTRATE SPECIFICITY AND KINETIC PROPERTIES OF SEVEN HETEROLOGOUSLY EXPRESSED DOG CYTOCHROMES P450Magang Shou, Ryan Norcross, Grit Sandig, Ping Lu, Yinghe Li, Yuh Lin, Qin Mei, A. David Rodrigues and Thomas H. RushmoreDrug Metabolism and Disposition September 2003, 31 (9) 1161-1169; DOI: https://doi.org/10.1124/dmd.31.9.1161
Sinz, Michael
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Skinner, M.
- You have accessMETABOLISM, EXCRETION, AND PHARMACOKINETICS OF DULOXETINE IN HEALTHY HUMAN SUBJECTSR. J. Lantz, T. A. Gillespie, T. J. Rash, F. Kuo, M. Skinner, H-Y. Kuan and M. P. KnadlerDrug Metabolism and Disposition September 2003, 31 (9) 1142-1150; DOI: https://doi.org/10.1124/dmd.31.9.1142
Slitt, A. L.
- You have accessINDUCTION OF MULTIDRUG RESISTANCE PROTEIN 3 IN RAT LIVER IS ASSOCIATED WITH ALTERED VECTORIAL EXCRETION OF ACETAMINOPHEN METABOLITESA. L. Slitt, N. J. Cherrington, J. M. Maher and C. D. KlaassenDrug Metabolism and Disposition September 2003, 31 (9) 1176-1186; DOI: https://doi.org/10.1124/dmd.31.9.1176
Smith, Graeme B. J.
- You have accessBIOTRANSFORMATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE (NNK) IN PERIPHERAL HUMAN LUNG MICROSOMESGraeme B. J. Smith, John R. Bend, Leanne L. Bedard, Ken R. Reid, Dimitri Petsikas and Thomas E. MasseyDrug Metabolism and Disposition September 2003, 31 (9) 1134-1141; DOI: https://doi.org/10.1124/dmd.31.9.1134
Solon, Eric
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Stone, Andrew N.
- You have accessISOFORM SELECTIVITY AND KINETICS OF MORPHINE 3- AND 6-GLUCURONIDATION BY HUMAN UDP-GLUCURONOSYLTRANSFERASES: EVIDENCE FOR ATYPICAL GLUCURONIDATION KINETICS BY UGT2B7Andrew N. Stone, Peter I. Mackenzie, Aleksandra Galetin, J. Brian Houston and John O. MinersDrug Metabolism and Disposition September 2003, 31 (9) 1086-1089; DOI: https://doi.org/10.1124/dmd.31.9.1086
T
Taavitsainen, Päivi
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
Taskinen, Jyrki
- You have accessCONJUGATION OF CATECHOLS BY RECOMBINANT HUMAN SULFOTRANSFERASES, UDP-GLUCURONOSYLTRANSFERASES, AND SOLUBLE CATECHOL O-METHYLTRANSFERASE: STRUCTURE-CONJUGATION RELATIONSHIPS AND PREDICTIVE MODELSJyrki Taskinen, Brian T. Ethell, Pia Pihlavisto, Alan M. Hood, Brian Burchell and Michael W. H. CoughtrieDrug Metabolism and Disposition September 2003, 31 (9) 1187-1197; DOI: https://doi.org/10.1124/dmd.31.9.1187
Thevis, Mario
- You have accessGLUCURONIDATION OF ANABOLIC ANDROGENIC STEROIDS BY RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESTiia Kuuranne, Mika Kurkela, Mario Thevis, Wilhelm Schänzer, Moshe Finel and Risto KostiainenDrug Metabolism and Disposition September 2003, 31 (9) 1117-1124; DOI: https://doi.org/10.1124/dmd.31.9.1117
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von Moltke, Lisa L.
- You have accessEVALUATION OF 3′-AZIDO-3′-DEOXYTHYMIDINE, MORPHINE, AND CODEINE AS PROBE SUBSTRATES FOR UDP-GLUCURONOSYLTRANSFERASE 2B7 (UGT2B7) IN HUMAN LIVER MICROSOMES: SPECIFICITY AND INFLUENCE OF THE UGT2B7*2 POLYMORPHISMMichael H. Court, Soundarajan Krishnaswamy, Qin Hao, Su X. Duan, Christopher J. Patten, Lisa L. von Moltke and David J. GreenblattDrug Metabolism and Disposition September 2003, 31 (9) 1125-1133; DOI: https://doi.org/10.1124/dmd.31.9.1125
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Wang, Lifei
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
Watts, Patricia
- You have accessCOMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMSJarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen and Olavi PelkonenDrug Metabolism and Disposition September 2003, 31 (9) 1093-1102; DOI: https://doi.org/10.1124/dmd.31.9.1093
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Yang, Tian J.
- You have accessCONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN l-VALINAMIDE DERIVATIVEGang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee and Liang-Shang GanDrug Metabolism and Disposition September 2003, 31 (9) 1170-1175; DOI: https://doi.org/10.1124/dmd.31.9.1170
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Zhang, Qing-Yu
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS OF THE HUMAN CYP2A13 GENE: EVIDENCE FOR A NULL ALLELEXiuling Zhang, Ying Chen, Yiqin Liu, Xiang Ren, Qing-Yu Zhang, Michele Caggana and Xinxin DingDrug Metabolism and Disposition September 2003, 31 (9) 1081-1085; DOI: https://doi.org/10.1124/dmd.31.9.1081
Zhang, Xiuling
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS OF THE HUMAN CYP2A13 GENE: EVIDENCE FOR A NULL ALLELEXiuling Zhang, Ying Chen, Yiqin Liu, Xiang Ren, Qing-Yu Zhang, Michele Caggana and Xinxin DingDrug Metabolism and Disposition September 2003, 31 (9) 1081-1085; DOI: https://doi.org/10.1124/dmd.31.9.1081