Index by author
October 01, 2004; Volume 32,Issue 10
A
Aboagye, E. O.
- You have accessPLASMA PHARMACOKINETICS AND METABOLISM OF THE HISTONE DEACETYLASE INHIBITOR TRICHOSTATIN A AFTER INTRAPERITONEAL ADMINISTRATION TO MICEL. Sanderson, G. W. Taylor, E. O. Aboagye, J. P. Alao, J. R. Latigo, R. C. Coombes and D. M. VigushinDrug Metabolism and Disposition October 2004, 32 (10) 1132-1138; DOI: https://doi.org/10.1124/dmd.104.000638
Alao, J. P.
- You have accessPLASMA PHARMACOKINETICS AND METABOLISM OF THE HISTONE DEACETYLASE INHIBITOR TRICHOSTATIN A AFTER INTRAPERITONEAL ADMINISTRATION TO MICEL. Sanderson, G. W. Taylor, E. O. Aboagye, J. P. Alao, J. R. Latigo, R. C. Coombes and D. M. VigushinDrug Metabolism and Disposition October 2004, 32 (10) 1132-1138; DOI: https://doi.org/10.1124/dmd.104.000638
Allen, Kyle
- You have accessDIFFERENCES IN THE INHIBITION OF CYTOCHROMES P450 3A4 AND 3A5 BY METABOLITE-INHIBITOR COMPLEX-FORMING DRUGSDonavon J. McConn, Yvonne S. Lin, Kyle Allen, Kent L. Kunze and Kenneth E. ThummelDrug Metabolism and Disposition October 2004, 32 (10) 1083-1091; DOI: https://doi.org/10.1124/dmd.32.10.1083
Allen, Kyle E.
- You have accessROLE OF ITRACONAZOLE METABOLITES IN CYP3A4 INHIBITIONNina Isoherranen, Kent L. Kunze, Kyle E. Allen, Wendel L. Nelson and Kenneth E. ThummelDrug Metabolism and Disposition October 2004, 32 (10) 1121-1131; DOI: https://doi.org/10.1124/dmd.104.000315
B
Balakin, Konstantin V.
- You have accessQUANTITATIVE STRUCTURE-METABOLISM RELATIONSHIP MODELING OF METABOLIC N-DEALKYLATION REACTION RATESKonstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1111-1120; DOI: https://doi.org/10.1124/dmd.104.000364
- You have accessKOHONEN MAPS FOR PREDICTION OF BINDING TO HUMAN CYTOCHROME P450 3A4Konstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey V. Skorenko, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1183-1189; DOI: https://doi.org/10.1124/dmd.104.000356
Balani, Suresh K.
- You have accessEFFECTIVE DOSING REGIMEN OF 1-AMINOBENZOTRIAZOLE FOR INHIBITION OF ANTIPYRINE CLEARANCE IN GUINEA PIGS AND MICE USING SERIAL SAMPLINGSuresh K. Balani, Ping Li, Joanne Nguyen, Kym Cardoza, Hang Zeng, Dun-Xue Mu, Jing-Tao Wu, Liang-Shang Gan and Frank W. LeeDrug Metabolism and Disposition October 2004, 32 (10) 1092-1095; DOI: https://doi.org/10.1124/dmd.104.000349
Biba, Mirlinda
- You have accessSPECIES DIFFERENTIAL STEREOSELECTIVE OXIDATION OF A METHYLSULFIDE METABOLITE OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DUAL AGONISTBindhu V. Karanam, Christopher J. Welch, Vijay G. Reddy, Jennifer Chilenski, Mirlinda Biba and Stella VincentDrug Metabolism and Disposition October 2004, 32 (10) 1061-1068; DOI: https://doi.org/10.1124/dmd.104.000224
Blumberg, Bruce
- You have accessTOCOTRIENOLS ACTIVATE THE STEROID AND XENOBIOTIC RECEPTOR, SXR, AND SELECTIVELY REGULATE EXPRESSION OF ITS TARGET GENESChangcheng Zhou, Michelle M. Tabb, Asal Sadatrafiei, Felix Grün and Bruce BlumbergDrug Metabolism and Disposition October 2004, 32 (10) 1075-1082; DOI: https://doi.org/10.1124/dmd.104.000299
Bugrim, Andrey
- You have accessQUANTITATIVE STRUCTURE-METABOLISM RELATIONSHIP MODELING OF METABOLIC N-DEALKYLATION REACTION RATESKonstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1111-1120; DOI: https://doi.org/10.1124/dmd.104.000364
- You have accessKOHONEN MAPS FOR PREDICTION OF BINDING TO HUMAN CYTOCHROME P450 3A4Konstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey V. Skorenko, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1183-1189; DOI: https://doi.org/10.1124/dmd.104.000356
C
Cardoza, Kym
- You have accessEFFECTIVE DOSING REGIMEN OF 1-AMINOBENZOTRIAZOLE FOR INHIBITION OF ANTIPYRINE CLEARANCE IN GUINEA PIGS AND MICE USING SERIAL SAMPLINGSuresh K. Balani, Ping Li, Joanne Nguyen, Kym Cardoza, Hang Zeng, Dun-Xue Mu, Jing-Tao Wu, Liang-Shang Gan and Frank W. LeeDrug Metabolism and Disposition October 2004, 32 (10) 1092-1095; DOI: https://doi.org/10.1124/dmd.104.000349
Chiba, Kan
- You have accessIDENTIFICATION OF DI-(2-ETHYLHEXYL) PHTHALATE-INDUCED CARBOXYLESTERASE 1 IN C57BL/6 MOUSE LIVER MICROSOMES: PURIFICATION, CDNA CLONING, AND BACULOVIRUS-MEDIATED EXPRESSIONTomomi Furihata, Masakiyo Hosokawa, Nao Koyano, Takahiro Nakamura, Tetsuo Satoh and Kan ChibaDrug Metabolism and Disposition October 2004, 32 (10) 1170-1177; DOI: https://doi.org/10.1124/dmd.104.000620
Chilenski, Jennifer
- You have accessSPECIES DIFFERENTIAL STEREOSELECTIVE OXIDATION OF A METHYLSULFIDE METABOLITE OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DUAL AGONISTBindhu V. Karanam, Christopher J. Welch, Vijay G. Reddy, Jennifer Chilenski, Mirlinda Biba and Stella VincentDrug Metabolism and Disposition October 2004, 32 (10) 1061-1068; DOI: https://doi.org/10.1124/dmd.104.000224
Coombes, R. C.
- You have accessPLASMA PHARMACOKINETICS AND METABOLISM OF THE HISTONE DEACETYLASE INHIBITOR TRICHOSTATIN A AFTER INTRAPERITONEAL ADMINISTRATION TO MICEL. Sanderson, G. W. Taylor, E. O. Aboagye, J. P. Alao, J. R. Latigo, R. C. Coombes and D. M. VigushinDrug Metabolism and Disposition October 2004, 32 (10) 1132-1138; DOI: https://doi.org/10.1124/dmd.104.000638
Creighton, Mellissa
- You have accessIDENTIFICATION AND METABOLISM OF A NOVEL DIHYDROHYDROXY-S-GLUTATHIONYL CONJUGATE OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST, MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], IN RATSVijay Bhasker G. Reddy, George A. Doss, Mellissa Creighton, Christopher J. Kochansky, Stella H. Vincent, Ronald B. Franklin and Bindhu V. KaranamDrug Metabolism and Disposition October 2004, 32 (10) 1154-1161; DOI: https://doi.org/10.1124/dmd.104.000240
Criss, Anne B.
- You have accessTWO MAJOR GRAPEFRUIT JUICE COMPONENTS DIFFER IN INTESTINAL CYP3A4 INHIBITION KINETIC AND BINDING PROPERTIESMary F. Paine, Anne B. Criss and Paul B. WatkinsDrug Metabolism and Disposition October 2004, 32 (10) 1146-1153; DOI: https://doi.org/10.1124/dmd.104.000547
D
Doss, George A.
- You have accessIDENTIFICATION AND METABOLISM OF A NOVEL DIHYDROHYDROXY-S-GLUTATHIONYL CONJUGATE OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST, MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], IN RATSVijay Bhasker G. Reddy, George A. Doss, Mellissa Creighton, Christopher J. Kochansky, Stella H. Vincent, Ronald B. Franklin and Bindhu V. KaranamDrug Metabolism and Disposition October 2004, 32 (10) 1154-1161; DOI: https://doi.org/10.1124/dmd.104.000240
E
Ekins, Sean
- You have accessQUANTITATIVE STRUCTURE-METABOLISM RELATIONSHIP MODELING OF METABOLIC N-DEALKYLATION REACTION RATESKonstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1111-1120; DOI: https://doi.org/10.1124/dmd.104.000364
- You have accessKOHONEN MAPS FOR PREDICTION OF BINDING TO HUMAN CYTOCHROME P450 3A4Konstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey V. Skorenko, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1183-1189; DOI: https://doi.org/10.1124/dmd.104.000356
Endo, Yoshio
- You have accessA CRUCIAL ROLE OF URIDINE/CYTIDINE KINASE 2 IN ANTITUMOR ACTIVITY OF 3′-ETHYNYL NUCLEOSIDESDaigo Murata, Yoshio Endo, Tohru Obata, Kazuki Sakamoto, Yasuhiro Syouji, Masakazu Kadohira, Akira Matsuda and Takuma SasakiDrug Metabolism and Disposition October 2004, 32 (10) 1178-1182; DOI: https://doi.org/10.1124/dmd.104.000737
Endou, Hitoshi
- You have accessCHARACTERIZATION OF THE RENAL TUBULAR TRANSPORT OF ZONAMPANEL, A NOVEL α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID RECEPTOR ANTAGONIST, BY HUMAN ORGANIC ANION TRANSPORTERSTadashi Hashimoto, Shinichi Narikawa, Xiu-Lin Huang, Tsuyoshi Minematsu, Takashi Usui, Hidetaka Kamimura and Hitoshi EndouDrug Metabolism and Disposition October 2004, 32 (10) 1096-1102; DOI: https://doi.org/10.1124/dmd.32.10.1096
F
Falany, Charles N.
- You have accessTRICLOSAN AS A SUBSTRATE AND INHIBITOR OF 3′-PHOSPHOADENOSINE 5′-PHOSPHOSULFATE-SULFOTRANSFERASE AND UDP-GLUCURONOSYL TRANSFERASE IN HUMAN LIVER FRACTIONSLi-Quan Wang, Charles N. Falany and Margaret O. JamesDrug Metabolism and Disposition October 2004, 32 (10) 1162-1169; DOI: https://doi.org/10.1124/dmd.104.000273
Franklin, Ronald B.
- You have accessIDENTIFICATION AND METABOLISM OF A NOVEL DIHYDROHYDROXY-S-GLUTATHIONYL CONJUGATE OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST, MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], IN RATSVijay Bhasker G. Reddy, George A. Doss, Mellissa Creighton, Christopher J. Kochansky, Stella H. Vincent, Ronald B. Franklin and Bindhu V. KaranamDrug Metabolism and Disposition October 2004, 32 (10) 1154-1161; DOI: https://doi.org/10.1124/dmd.104.000240
Fukunaga, Naoko
- You have accessCONSTRUCTION OF EXPRESSION SYSTEM FOR HUMAN α1-ACID GLYCOPROTEIN IN PICHIA PASTORIS AND EVALUATION OF ITS DRUG-BINDING PROPERTIESKoji Nishi, Naoko Fukunaga and Masaki OtagiriDrug Metabolism and Disposition October 2004, 32 (10) 1069-1074; DOI: https://doi.org/10.1124/dmd.104.000513
Furihata, Tomomi
- You have accessIDENTIFICATION OF DI-(2-ETHYLHEXYL) PHTHALATE-INDUCED CARBOXYLESTERASE 1 IN C57BL/6 MOUSE LIVER MICROSOMES: PURIFICATION, CDNA CLONING, AND BACULOVIRUS-MEDIATED EXPRESSIONTomomi Furihata, Masakiyo Hosokawa, Nao Koyano, Takahiro Nakamura, Tetsuo Satoh and Kan ChibaDrug Metabolism and Disposition October 2004, 32 (10) 1170-1177; DOI: https://doi.org/10.1124/dmd.104.000620
G
Gan, Liang-Shang
- You have accessEFFECTIVE DOSING REGIMEN OF 1-AMINOBENZOTRIAZOLE FOR INHIBITION OF ANTIPYRINE CLEARANCE IN GUINEA PIGS AND MICE USING SERIAL SAMPLINGSuresh K. Balani, Ping Li, Joanne Nguyen, Kym Cardoza, Hang Zeng, Dun-Xue Mu, Jing-Tao Wu, Liang-Shang Gan and Frank W. LeeDrug Metabolism and Disposition October 2004, 32 (10) 1092-1095; DOI: https://doi.org/10.1124/dmd.104.000349
Gerk, Phillip M.
- You have accessESTRADIOL 3-GLUCURONIDE IS TRANSPORTED BY THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN 2 BUT DOES NOT ACTIVATE THE ALLOSTERIC SITE BOUND BY ESTRADIOL 17-GLUCURONIDEPhillip M. Gerk, Wei Li and Mary VoreDrug Metabolism and Disposition October 2004, 32 (10) 1139-1145; DOI: https://doi.org/10.1124/dmd.104.000372
Grün, Felix
- You have accessTOCOTRIENOLS ACTIVATE THE STEROID AND XENOBIOTIC RECEPTOR, SXR, AND SELECTIVELY REGULATE EXPRESSION OF ITS TARGET GENESChangcheng Zhou, Michelle M. Tabb, Asal Sadatrafiei, Felix Grün and Bruce BlumbergDrug Metabolism and Disposition October 2004, 32 (10) 1075-1082; DOI: https://doi.org/10.1124/dmd.104.000299
H
Hashimoto, Tadashi
- You have accessCHARACTERIZATION OF THE RENAL TUBULAR TRANSPORT OF ZONAMPANEL, A NOVEL α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID RECEPTOR ANTAGONIST, BY HUMAN ORGANIC ANION TRANSPORTERSTadashi Hashimoto, Shinichi Narikawa, Xiu-Lin Huang, Tsuyoshi Minematsu, Takashi Usui, Hidetaka Kamimura and Hitoshi EndouDrug Metabolism and Disposition October 2004, 32 (10) 1096-1102; DOI: https://doi.org/10.1124/dmd.32.10.1096
Hosokawa, Masakiyo
- You have accessIDENTIFICATION OF DI-(2-ETHYLHEXYL) PHTHALATE-INDUCED CARBOXYLESTERASE 1 IN C57BL/6 MOUSE LIVER MICROSOMES: PURIFICATION, CDNA CLONING, AND BACULOVIRUS-MEDIATED EXPRESSIONTomomi Furihata, Masakiyo Hosokawa, Nao Koyano, Takahiro Nakamura, Tetsuo Satoh and Kan ChibaDrug Metabolism and Disposition October 2004, 32 (10) 1170-1177; DOI: https://doi.org/10.1124/dmd.104.000620
Huang, Xiu-Lin
- You have accessCHARACTERIZATION OF THE RENAL TUBULAR TRANSPORT OF ZONAMPANEL, A NOVEL α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID RECEPTOR ANTAGONIST, BY HUMAN ORGANIC ANION TRANSPORTERSTadashi Hashimoto, Shinichi Narikawa, Xiu-Lin Huang, Tsuyoshi Minematsu, Takashi Usui, Hidetaka Kamimura and Hitoshi EndouDrug Metabolism and Disposition October 2004, 32 (10) 1096-1102; DOI: https://doi.org/10.1124/dmd.32.10.1096
I
Ishii, Yuji
- You have accessSIMULTANEOUS EXPRESSION OF GUINEA PIG UDP-GLUCURONOSYLTRANSFERASE 2B21 (UGT2B21) AND 2B22 IN COS-7 CELLS ENHANCES UGT2B21-CATALYZED CHLORAMPHENICOL GLUCURONIDATIONYuji Ishii, Aya Miyoshi, Daisuke Maji, Hideyuki Yamada and Kazuta OguriDrug Metabolism and Disposition October 2004, 32 (10) 1057-1060; DOI: https://doi.org/10.1124/dmd.32.10.1057
Isoherranen, Nina
- You have accessROLE OF ITRACONAZOLE METABOLITES IN CYP3A4 INHIBITIONNina Isoherranen, Kent L. Kunze, Kyle E. Allen, Wendel L. Nelson and Kenneth E. ThummelDrug Metabolism and Disposition October 2004, 32 (10) 1121-1131; DOI: https://doi.org/10.1124/dmd.104.000315
Ivanenkov, Yan A.
- You have accessQUANTITATIVE STRUCTURE-METABOLISM RELATIONSHIP MODELING OF METABOLIC N-DEALKYLATION REACTION RATESKonstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1111-1120; DOI: https://doi.org/10.1124/dmd.104.000364
- You have accessKOHONEN MAPS FOR PREDICTION OF BINDING TO HUMAN CYTOCHROME P450 3A4Konstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey V. Skorenko, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1183-1189; DOI: https://doi.org/10.1124/dmd.104.000356
Ivashchenko, Andrey A.
- You have accessQUANTITATIVE STRUCTURE-METABOLISM RELATIONSHIP MODELING OF METABOLIC N-DEALKYLATION REACTION RATESKonstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1111-1120; DOI: https://doi.org/10.1124/dmd.104.000364
- You have accessKOHONEN MAPS FOR PREDICTION OF BINDING TO HUMAN CYTOCHROME P450 3A4Konstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey V. Skorenko, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1183-1189; DOI: https://doi.org/10.1124/dmd.104.000356
J
James, Margaret O.
- You have accessTRICLOSAN AS A SUBSTRATE AND INHIBITOR OF 3′-PHOSPHOADENOSINE 5′-PHOSPHOSULFATE-SULFOTRANSFERASE AND UDP-GLUCURONOSYL TRANSFERASE IN HUMAN LIVER FRACTIONSLi-Quan Wang, Charles N. Falany and Margaret O. JamesDrug Metabolism and Disposition October 2004, 32 (10) 1162-1169; DOI: https://doi.org/10.1124/dmd.104.000273
K
Kadohira, Masakazu
- You have accessA CRUCIAL ROLE OF URIDINE/CYTIDINE KINASE 2 IN ANTITUMOR ACTIVITY OF 3′-ETHYNYL NUCLEOSIDESDaigo Murata, Yoshio Endo, Tohru Obata, Kazuki Sakamoto, Yasuhiro Syouji, Masakazu Kadohira, Akira Matsuda and Takuma SasakiDrug Metabolism and Disposition October 2004, 32 (10) 1178-1182; DOI: https://doi.org/10.1124/dmd.104.000737
Kamimura, Hidetaka
- You have accessCHARACTERIZATION OF THE RENAL TUBULAR TRANSPORT OF ZONAMPANEL, A NOVEL α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID RECEPTOR ANTAGONIST, BY HUMAN ORGANIC ANION TRANSPORTERSTadashi Hashimoto, Shinichi Narikawa, Xiu-Lin Huang, Tsuyoshi Minematsu, Takashi Usui, Hidetaka Kamimura and Hitoshi EndouDrug Metabolism and Disposition October 2004, 32 (10) 1096-1102; DOI: https://doi.org/10.1124/dmd.32.10.1096
Karanam, Bindhu V.
- You have accessSPECIES DIFFERENTIAL STEREOSELECTIVE OXIDATION OF A METHYLSULFIDE METABOLITE OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DUAL AGONISTBindhu V. Karanam, Christopher J. Welch, Vijay G. Reddy, Jennifer Chilenski, Mirlinda Biba and Stella VincentDrug Metabolism and Disposition October 2004, 32 (10) 1061-1068; DOI: https://doi.org/10.1124/dmd.104.000224
- You have accessIDENTIFICATION AND METABOLISM OF A NOVEL DIHYDROHYDROXY-S-GLUTATHIONYL CONJUGATE OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST, MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], IN RATSVijay Bhasker G. Reddy, George A. Doss, Mellissa Creighton, Christopher J. Kochansky, Stella H. Vincent, Ronald B. Franklin and Bindhu V. KaranamDrug Metabolism and Disposition October 2004, 32 (10) 1154-1161; DOI: https://doi.org/10.1124/dmd.104.000240
Katoh, Miki
- You have accessIDENTIFICATION OF THE CYTOSOLIC CARBOXYLESTERASE CATALYZING THE 5′-DEOXY-5-FLUOROCYTIDINE FORMATION FROM CAPECITABINE IN HUMAN LIVERToshiki Tabata, Miki Katoh, Shogo Tokudome, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition October 2004, 32 (10) 1103-1110; DOI: https://doi.org/10.1124/dmd.104.000554
Kochansky, Christopher J.
- You have accessIDENTIFICATION AND METABOLISM OF A NOVEL DIHYDROHYDROXY-S-GLUTATHIONYL CONJUGATE OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST, MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], IN RATSVijay Bhasker G. Reddy, George A. Doss, Mellissa Creighton, Christopher J. Kochansky, Stella H. Vincent, Ronald B. Franklin and Bindhu V. KaranamDrug Metabolism and Disposition October 2004, 32 (10) 1154-1161; DOI: https://doi.org/10.1124/dmd.104.000240
Korolev, Dmitry
- You have accessQUANTITATIVE STRUCTURE-METABOLISM RELATIONSHIP MODELING OF METABOLIC N-DEALKYLATION REACTION RATESKonstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1111-1120; DOI: https://doi.org/10.1124/dmd.104.000364
- You have accessKOHONEN MAPS FOR PREDICTION OF BINDING TO HUMAN CYTOCHROME P450 3A4Konstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey V. Skorenko, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1183-1189; DOI: https://doi.org/10.1124/dmd.104.000356
Koyano, Nao
- You have accessIDENTIFICATION OF DI-(2-ETHYLHEXYL) PHTHALATE-INDUCED CARBOXYLESTERASE 1 IN C57BL/6 MOUSE LIVER MICROSOMES: PURIFICATION, CDNA CLONING, AND BACULOVIRUS-MEDIATED EXPRESSIONTomomi Furihata, Masakiyo Hosokawa, Nao Koyano, Takahiro Nakamura, Tetsuo Satoh and Kan ChibaDrug Metabolism and Disposition October 2004, 32 (10) 1170-1177; DOI: https://doi.org/10.1124/dmd.104.000620
Kunze, Kent L.
- You have accessDIFFERENCES IN THE INHIBITION OF CYTOCHROMES P450 3A4 AND 3A5 BY METABOLITE-INHIBITOR COMPLEX-FORMING DRUGSDonavon J. McConn, Yvonne S. Lin, Kyle Allen, Kent L. Kunze and Kenneth E. ThummelDrug Metabolism and Disposition October 2004, 32 (10) 1083-1091; DOI: https://doi.org/10.1124/dmd.32.10.1083
- You have accessROLE OF ITRACONAZOLE METABOLITES IN CYP3A4 INHIBITIONNina Isoherranen, Kent L. Kunze, Kyle E. Allen, Wendel L. Nelson and Kenneth E. ThummelDrug Metabolism and Disposition October 2004, 32 (10) 1121-1131; DOI: https://doi.org/10.1124/dmd.104.000315
L
Latigo, J. R.
- You have accessPLASMA PHARMACOKINETICS AND METABOLISM OF THE HISTONE DEACETYLASE INHIBITOR TRICHOSTATIN A AFTER INTRAPERITONEAL ADMINISTRATION TO MICEL. Sanderson, G. W. Taylor, E. O. Aboagye, J. P. Alao, J. R. Latigo, R. C. Coombes and D. M. VigushinDrug Metabolism and Disposition October 2004, 32 (10) 1132-1138; DOI: https://doi.org/10.1124/dmd.104.000638
Lee, Frank W.
- You have accessEFFECTIVE DOSING REGIMEN OF 1-AMINOBENZOTRIAZOLE FOR INHIBITION OF ANTIPYRINE CLEARANCE IN GUINEA PIGS AND MICE USING SERIAL SAMPLINGSuresh K. Balani, Ping Li, Joanne Nguyen, Kym Cardoza, Hang Zeng, Dun-Xue Mu, Jing-Tao Wu, Liang-Shang Gan and Frank W. LeeDrug Metabolism and Disposition October 2004, 32 (10) 1092-1095; DOI: https://doi.org/10.1124/dmd.104.000349
Li, Ping
- You have accessEFFECTIVE DOSING REGIMEN OF 1-AMINOBENZOTRIAZOLE FOR INHIBITION OF ANTIPYRINE CLEARANCE IN GUINEA PIGS AND MICE USING SERIAL SAMPLINGSuresh K. Balani, Ping Li, Joanne Nguyen, Kym Cardoza, Hang Zeng, Dun-Xue Mu, Jing-Tao Wu, Liang-Shang Gan and Frank W. LeeDrug Metabolism and Disposition October 2004, 32 (10) 1092-1095; DOI: https://doi.org/10.1124/dmd.104.000349
Li, Wei
- You have accessESTRADIOL 3-GLUCURONIDE IS TRANSPORTED BY THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN 2 BUT DOES NOT ACTIVATE THE ALLOSTERIC SITE BOUND BY ESTRADIOL 17-GLUCURONIDEPhillip M. Gerk, Wei Li and Mary VoreDrug Metabolism and Disposition October 2004, 32 (10) 1139-1145; DOI: https://doi.org/10.1124/dmd.104.000372
Lin, Yvonne S.
- You have accessDIFFERENCES IN THE INHIBITION OF CYTOCHROMES P450 3A4 AND 3A5 BY METABOLITE-INHIBITOR COMPLEX-FORMING DRUGSDonavon J. McConn, Yvonne S. Lin, Kyle Allen, Kent L. Kunze and Kenneth E. ThummelDrug Metabolism and Disposition October 2004, 32 (10) 1083-1091; DOI: https://doi.org/10.1124/dmd.32.10.1083
M
Maji, Daisuke
- You have accessSIMULTANEOUS EXPRESSION OF GUINEA PIG UDP-GLUCURONOSYLTRANSFERASE 2B21 (UGT2B21) AND 2B22 IN COS-7 CELLS ENHANCES UGT2B21-CATALYZED CHLORAMPHENICOL GLUCURONIDATIONYuji Ishii, Aya Miyoshi, Daisuke Maji, Hideyuki Yamada and Kazuta OguriDrug Metabolism and Disposition October 2004, 32 (10) 1057-1060; DOI: https://doi.org/10.1124/dmd.32.10.1057
Matsuda, Akira
- You have accessA CRUCIAL ROLE OF URIDINE/CYTIDINE KINASE 2 IN ANTITUMOR ACTIVITY OF 3′-ETHYNYL NUCLEOSIDESDaigo Murata, Yoshio Endo, Tohru Obata, Kazuki Sakamoto, Yasuhiro Syouji, Masakazu Kadohira, Akira Matsuda and Takuma SasakiDrug Metabolism and Disposition October 2004, 32 (10) 1178-1182; DOI: https://doi.org/10.1124/dmd.104.000737
McConn, Donavon J.
- You have accessDIFFERENCES IN THE INHIBITION OF CYTOCHROMES P450 3A4 AND 3A5 BY METABOLITE-INHIBITOR COMPLEX-FORMING DRUGSDonavon J. McConn, Yvonne S. Lin, Kyle Allen, Kent L. Kunze and Kenneth E. ThummelDrug Metabolism and Disposition October 2004, 32 (10) 1083-1091; DOI: https://doi.org/10.1124/dmd.32.10.1083
Minematsu, Tsuyoshi
- You have accessCHARACTERIZATION OF THE RENAL TUBULAR TRANSPORT OF ZONAMPANEL, A NOVEL α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID RECEPTOR ANTAGONIST, BY HUMAN ORGANIC ANION TRANSPORTERSTadashi Hashimoto, Shinichi Narikawa, Xiu-Lin Huang, Tsuyoshi Minematsu, Takashi Usui, Hidetaka Kamimura and Hitoshi EndouDrug Metabolism and Disposition October 2004, 32 (10) 1096-1102; DOI: https://doi.org/10.1124/dmd.32.10.1096
Miyoshi, Aya
- You have accessSIMULTANEOUS EXPRESSION OF GUINEA PIG UDP-GLUCURONOSYLTRANSFERASE 2B21 (UGT2B21) AND 2B22 IN COS-7 CELLS ENHANCES UGT2B21-CATALYZED CHLORAMPHENICOL GLUCURONIDATIONYuji Ishii, Aya Miyoshi, Daisuke Maji, Hideyuki Yamada and Kazuta OguriDrug Metabolism and Disposition October 2004, 32 (10) 1057-1060; DOI: https://doi.org/10.1124/dmd.32.10.1057
Mu, Dun-Xue
- You have accessEFFECTIVE DOSING REGIMEN OF 1-AMINOBENZOTRIAZOLE FOR INHIBITION OF ANTIPYRINE CLEARANCE IN GUINEA PIGS AND MICE USING SERIAL SAMPLINGSuresh K. Balani, Ping Li, Joanne Nguyen, Kym Cardoza, Hang Zeng, Dun-Xue Mu, Jing-Tao Wu, Liang-Shang Gan and Frank W. LeeDrug Metabolism and Disposition October 2004, 32 (10) 1092-1095; DOI: https://doi.org/10.1124/dmd.104.000349
Murata, Daigo
- You have accessA CRUCIAL ROLE OF URIDINE/CYTIDINE KINASE 2 IN ANTITUMOR ACTIVITY OF 3′-ETHYNYL NUCLEOSIDESDaigo Murata, Yoshio Endo, Tohru Obata, Kazuki Sakamoto, Yasuhiro Syouji, Masakazu Kadohira, Akira Matsuda and Takuma SasakiDrug Metabolism and Disposition October 2004, 32 (10) 1178-1182; DOI: https://doi.org/10.1124/dmd.104.000737
N
Nakajima, Miki
- You have accessIDENTIFICATION OF THE CYTOSOLIC CARBOXYLESTERASE CATALYZING THE 5′-DEOXY-5-FLUOROCYTIDINE FORMATION FROM CAPECITABINE IN HUMAN LIVERToshiki Tabata, Miki Katoh, Shogo Tokudome, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition October 2004, 32 (10) 1103-1110; DOI: https://doi.org/10.1124/dmd.104.000554
Nakamura, Takahiro
- You have accessIDENTIFICATION OF DI-(2-ETHYLHEXYL) PHTHALATE-INDUCED CARBOXYLESTERASE 1 IN C57BL/6 MOUSE LIVER MICROSOMES: PURIFICATION, CDNA CLONING, AND BACULOVIRUS-MEDIATED EXPRESSIONTomomi Furihata, Masakiyo Hosokawa, Nao Koyano, Takahiro Nakamura, Tetsuo Satoh and Kan ChibaDrug Metabolism and Disposition October 2004, 32 (10) 1170-1177; DOI: https://doi.org/10.1124/dmd.104.000620
Narikawa, Shinichi
- You have accessCHARACTERIZATION OF THE RENAL TUBULAR TRANSPORT OF ZONAMPANEL, A NOVEL α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID RECEPTOR ANTAGONIST, BY HUMAN ORGANIC ANION TRANSPORTERSTadashi Hashimoto, Shinichi Narikawa, Xiu-Lin Huang, Tsuyoshi Minematsu, Takashi Usui, Hidetaka Kamimura and Hitoshi EndouDrug Metabolism and Disposition October 2004, 32 (10) 1096-1102; DOI: https://doi.org/10.1124/dmd.32.10.1096
Nelson, Wendel L.
- You have accessROLE OF ITRACONAZOLE METABOLITES IN CYP3A4 INHIBITIONNina Isoherranen, Kent L. Kunze, Kyle E. Allen, Wendel L. Nelson and Kenneth E. ThummelDrug Metabolism and Disposition October 2004, 32 (10) 1121-1131; DOI: https://doi.org/10.1124/dmd.104.000315
Nguyen, Joanne
- You have accessEFFECTIVE DOSING REGIMEN OF 1-AMINOBENZOTRIAZOLE FOR INHIBITION OF ANTIPYRINE CLEARANCE IN GUINEA PIGS AND MICE USING SERIAL SAMPLINGSuresh K. Balani, Ping Li, Joanne Nguyen, Kym Cardoza, Hang Zeng, Dun-Xue Mu, Jing-Tao Wu, Liang-Shang Gan and Frank W. LeeDrug Metabolism and Disposition October 2004, 32 (10) 1092-1095; DOI: https://doi.org/10.1124/dmd.104.000349
Nikolskaya, Tatiana
- You have accessQUANTITATIVE STRUCTURE-METABOLISM RELATIONSHIP MODELING OF METABOLIC N-DEALKYLATION REACTION RATESKonstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1111-1120; DOI: https://doi.org/10.1124/dmd.104.000364
- You have accessKOHONEN MAPS FOR PREDICTION OF BINDING TO HUMAN CYTOCHROME P450 3A4Konstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey V. Skorenko, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1183-1189; DOI: https://doi.org/10.1124/dmd.104.000356
Nikolsky, Yuri V.
- You have accessQUANTITATIVE STRUCTURE-METABOLISM RELATIONSHIP MODELING OF METABOLIC N-DEALKYLATION REACTION RATESKonstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1111-1120; DOI: https://doi.org/10.1124/dmd.104.000364
- You have accessKOHONEN MAPS FOR PREDICTION OF BINDING TO HUMAN CYTOCHROME P450 3A4Konstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey V. Skorenko, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1183-1189; DOI: https://doi.org/10.1124/dmd.104.000356
Nishi, Koji
- You have accessCONSTRUCTION OF EXPRESSION SYSTEM FOR HUMAN α1-ACID GLYCOPROTEIN IN PICHIA PASTORIS AND EVALUATION OF ITS DRUG-BINDING PROPERTIESKoji Nishi, Naoko Fukunaga and Masaki OtagiriDrug Metabolism and Disposition October 2004, 32 (10) 1069-1074; DOI: https://doi.org/10.1124/dmd.104.000513
Nocerini, Mark R.
- You have accessUTILITY OF WHOLE-BODY AUTORADIOLUMINOGRAPHY IN DRUG DISCOVERY FOR THE QUANTIFICATION OF TRITIUM-LABELED DRUG CANDIDATESMichael J. Potchoiba and Mark R. NoceriniDrug Metabolism and Disposition October 2004, 32 (10) 1190-1198; DOI: https://doi.org/10.1124/dmd.32.10.1190
O
Obata, Tohru
- You have accessA CRUCIAL ROLE OF URIDINE/CYTIDINE KINASE 2 IN ANTITUMOR ACTIVITY OF 3′-ETHYNYL NUCLEOSIDESDaigo Murata, Yoshio Endo, Tohru Obata, Kazuki Sakamoto, Yasuhiro Syouji, Masakazu Kadohira, Akira Matsuda and Takuma SasakiDrug Metabolism and Disposition October 2004, 32 (10) 1178-1182; DOI: https://doi.org/10.1124/dmd.104.000737
Oguri, Kazuta
- You have accessSIMULTANEOUS EXPRESSION OF GUINEA PIG UDP-GLUCURONOSYLTRANSFERASE 2B21 (UGT2B21) AND 2B22 IN COS-7 CELLS ENHANCES UGT2B21-CATALYZED CHLORAMPHENICOL GLUCURONIDATIONYuji Ishii, Aya Miyoshi, Daisuke Maji, Hideyuki Yamada and Kazuta OguriDrug Metabolism and Disposition October 2004, 32 (10) 1057-1060; DOI: https://doi.org/10.1124/dmd.32.10.1057
Otagiri, Masaki
- You have accessCONSTRUCTION OF EXPRESSION SYSTEM FOR HUMAN α1-ACID GLYCOPROTEIN IN PICHIA PASTORIS AND EVALUATION OF ITS DRUG-BINDING PROPERTIESKoji Nishi, Naoko Fukunaga and Masaki OtagiriDrug Metabolism and Disposition October 2004, 32 (10) 1069-1074; DOI: https://doi.org/10.1124/dmd.104.000513
P
Paine, Mary F.
- You have accessTWO MAJOR GRAPEFRUIT JUICE COMPONENTS DIFFER IN INTESTINAL CYP3A4 INHIBITION KINETIC AND BINDING PROPERTIESMary F. Paine, Anne B. Criss and Paul B. WatkinsDrug Metabolism and Disposition October 2004, 32 (10) 1146-1153; DOI: https://doi.org/10.1124/dmd.104.000547
Potchoiba, Michael J.
- You have accessUTILITY OF WHOLE-BODY AUTORADIOLUMINOGRAPHY IN DRUG DISCOVERY FOR THE QUANTIFICATION OF TRITIUM-LABELED DRUG CANDIDATESMichael J. Potchoiba and Mark R. NoceriniDrug Metabolism and Disposition October 2004, 32 (10) 1190-1198; DOI: https://doi.org/10.1124/dmd.32.10.1190
R
Reddy, Vijay Bhasker G.
- You have accessIDENTIFICATION AND METABOLISM OF A NOVEL DIHYDROHYDROXY-S-GLUTATHIONYL CONJUGATE OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST, MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], IN RATSVijay Bhasker G. Reddy, George A. Doss, Mellissa Creighton, Christopher J. Kochansky, Stella H. Vincent, Ronald B. Franklin and Bindhu V. KaranamDrug Metabolism and Disposition October 2004, 32 (10) 1154-1161; DOI: https://doi.org/10.1124/dmd.104.000240
Reddy, Vijay G.
- You have accessSPECIES DIFFERENTIAL STEREOSELECTIVE OXIDATION OF A METHYLSULFIDE METABOLITE OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DUAL AGONISTBindhu V. Karanam, Christopher J. Welch, Vijay G. Reddy, Jennifer Chilenski, Mirlinda Biba and Stella VincentDrug Metabolism and Disposition October 2004, 32 (10) 1061-1068; DOI: https://doi.org/10.1124/dmd.104.000224
S
Sadatrafiei, Asal
- You have accessTOCOTRIENOLS ACTIVATE THE STEROID AND XENOBIOTIC RECEPTOR, SXR, AND SELECTIVELY REGULATE EXPRESSION OF ITS TARGET GENESChangcheng Zhou, Michelle M. Tabb, Asal Sadatrafiei, Felix Grün and Bruce BlumbergDrug Metabolism and Disposition October 2004, 32 (10) 1075-1082; DOI: https://doi.org/10.1124/dmd.104.000299
Sakamoto, Kazuki
- You have accessA CRUCIAL ROLE OF URIDINE/CYTIDINE KINASE 2 IN ANTITUMOR ACTIVITY OF 3′-ETHYNYL NUCLEOSIDESDaigo Murata, Yoshio Endo, Tohru Obata, Kazuki Sakamoto, Yasuhiro Syouji, Masakazu Kadohira, Akira Matsuda and Takuma SasakiDrug Metabolism and Disposition October 2004, 32 (10) 1178-1182; DOI: https://doi.org/10.1124/dmd.104.000737
Sanderson, L.
- You have accessPLASMA PHARMACOKINETICS AND METABOLISM OF THE HISTONE DEACETYLASE INHIBITOR TRICHOSTATIN A AFTER INTRAPERITONEAL ADMINISTRATION TO MICEL. Sanderson, G. W. Taylor, E. O. Aboagye, J. P. Alao, J. R. Latigo, R. C. Coombes and D. M. VigushinDrug Metabolism and Disposition October 2004, 32 (10) 1132-1138; DOI: https://doi.org/10.1124/dmd.104.000638
Sasaki, Takuma
- You have accessA CRUCIAL ROLE OF URIDINE/CYTIDINE KINASE 2 IN ANTITUMOR ACTIVITY OF 3′-ETHYNYL NUCLEOSIDESDaigo Murata, Yoshio Endo, Tohru Obata, Kazuki Sakamoto, Yasuhiro Syouji, Masakazu Kadohira, Akira Matsuda and Takuma SasakiDrug Metabolism and Disposition October 2004, 32 (10) 1178-1182; DOI: https://doi.org/10.1124/dmd.104.000737
Satoh, Tetsuo
- You have accessIDENTIFICATION OF DI-(2-ETHYLHEXYL) PHTHALATE-INDUCED CARBOXYLESTERASE 1 IN C57BL/6 MOUSE LIVER MICROSOMES: PURIFICATION, CDNA CLONING, AND BACULOVIRUS-MEDIATED EXPRESSIONTomomi Furihata, Masakiyo Hosokawa, Nao Koyano, Takahiro Nakamura, Tetsuo Satoh and Kan ChibaDrug Metabolism and Disposition October 2004, 32 (10) 1170-1177; DOI: https://doi.org/10.1124/dmd.104.000620
Savchuk, Nikolay P.
- You have accessQUANTITATIVE STRUCTURE-METABOLISM RELATIONSHIP MODELING OF METABOLIC N-DEALKYLATION REACTION RATESKonstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1111-1120; DOI: https://doi.org/10.1124/dmd.104.000364
- You have accessKOHONEN MAPS FOR PREDICTION OF BINDING TO HUMAN CYTOCHROME P450 3A4Konstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey V. Skorenko, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1183-1189; DOI: https://doi.org/10.1124/dmd.104.000356
Skorenko, Andrey V.
- You have accessKOHONEN MAPS FOR PREDICTION OF BINDING TO HUMAN CYTOCHROME P450 3A4Konstantin V. Balakin, Sean Ekins, Andrey Bugrim, Yan A. Ivanenkov, Dmitry Korolev, Yuri V. Nikolsky, Andrey V. Skorenko, Andrey A. Ivashchenko, Nikolay P. Savchuk and Tatiana NikolskayaDrug Metabolism and Disposition October 2004, 32 (10) 1183-1189; DOI: https://doi.org/10.1124/dmd.104.000356
Syouji, Yasuhiro
- You have accessA CRUCIAL ROLE OF URIDINE/CYTIDINE KINASE 2 IN ANTITUMOR ACTIVITY OF 3′-ETHYNYL NUCLEOSIDESDaigo Murata, Yoshio Endo, Tohru Obata, Kazuki Sakamoto, Yasuhiro Syouji, Masakazu Kadohira, Akira Matsuda and Takuma SasakiDrug Metabolism and Disposition October 2004, 32 (10) 1178-1182; DOI: https://doi.org/10.1124/dmd.104.000737
T
Tabata, Toshiki
- You have accessIDENTIFICATION OF THE CYTOSOLIC CARBOXYLESTERASE CATALYZING THE 5′-DEOXY-5-FLUOROCYTIDINE FORMATION FROM CAPECITABINE IN HUMAN LIVERToshiki Tabata, Miki Katoh, Shogo Tokudome, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition October 2004, 32 (10) 1103-1110; DOI: https://doi.org/10.1124/dmd.104.000554
Tabb, Michelle M.
- You have accessTOCOTRIENOLS ACTIVATE THE STEROID AND XENOBIOTIC RECEPTOR, SXR, AND SELECTIVELY REGULATE EXPRESSION OF ITS TARGET GENESChangcheng Zhou, Michelle M. Tabb, Asal Sadatrafiei, Felix Grün and Bruce BlumbergDrug Metabolism and Disposition October 2004, 32 (10) 1075-1082; DOI: https://doi.org/10.1124/dmd.104.000299
Taylor, G. W.
- You have accessPLASMA PHARMACOKINETICS AND METABOLISM OF THE HISTONE DEACETYLASE INHIBITOR TRICHOSTATIN A AFTER INTRAPERITONEAL ADMINISTRATION TO MICEL. Sanderson, G. W. Taylor, E. O. Aboagye, J. P. Alao, J. R. Latigo, R. C. Coombes and D. M. VigushinDrug Metabolism and Disposition October 2004, 32 (10) 1132-1138; DOI: https://doi.org/10.1124/dmd.104.000638
Thummel, Kenneth E.
- You have accessDIFFERENCES IN THE INHIBITION OF CYTOCHROMES P450 3A4 AND 3A5 BY METABOLITE-INHIBITOR COMPLEX-FORMING DRUGSDonavon J. McConn, Yvonne S. Lin, Kyle Allen, Kent L. Kunze and Kenneth E. ThummelDrug Metabolism and Disposition October 2004, 32 (10) 1083-1091; DOI: https://doi.org/10.1124/dmd.32.10.1083
- You have accessROLE OF ITRACONAZOLE METABOLITES IN CYP3A4 INHIBITIONNina Isoherranen, Kent L. Kunze, Kyle E. Allen, Wendel L. Nelson and Kenneth E. ThummelDrug Metabolism and Disposition October 2004, 32 (10) 1121-1131; DOI: https://doi.org/10.1124/dmd.104.000315
Tokudome, Shogo
- You have accessIDENTIFICATION OF THE CYTOSOLIC CARBOXYLESTERASE CATALYZING THE 5′-DEOXY-5-FLUOROCYTIDINE FORMATION FROM CAPECITABINE IN HUMAN LIVERToshiki Tabata, Miki Katoh, Shogo Tokudome, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition October 2004, 32 (10) 1103-1110; DOI: https://doi.org/10.1124/dmd.104.000554
U
Usui, Takashi
- You have accessCHARACTERIZATION OF THE RENAL TUBULAR TRANSPORT OF ZONAMPANEL, A NOVEL α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID RECEPTOR ANTAGONIST, BY HUMAN ORGANIC ANION TRANSPORTERSTadashi Hashimoto, Shinichi Narikawa, Xiu-Lin Huang, Tsuyoshi Minematsu, Takashi Usui, Hidetaka Kamimura and Hitoshi EndouDrug Metabolism and Disposition October 2004, 32 (10) 1096-1102; DOI: https://doi.org/10.1124/dmd.32.10.1096
V
Vigushin, D. M.
- You have accessPLASMA PHARMACOKINETICS AND METABOLISM OF THE HISTONE DEACETYLASE INHIBITOR TRICHOSTATIN A AFTER INTRAPERITONEAL ADMINISTRATION TO MICEL. Sanderson, G. W. Taylor, E. O. Aboagye, J. P. Alao, J. R. Latigo, R. C. Coombes and D. M. VigushinDrug Metabolism and Disposition October 2004, 32 (10) 1132-1138; DOI: https://doi.org/10.1124/dmd.104.000638
Vincent, Stella
- You have accessSPECIES DIFFERENTIAL STEREOSELECTIVE OXIDATION OF A METHYLSULFIDE METABOLITE OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DUAL AGONISTBindhu V. Karanam, Christopher J. Welch, Vijay G. Reddy, Jennifer Chilenski, Mirlinda Biba and Stella VincentDrug Metabolism and Disposition October 2004, 32 (10) 1061-1068; DOI: https://doi.org/10.1124/dmd.104.000224
Vincent, Stella H.
- You have accessIDENTIFICATION AND METABOLISM OF A NOVEL DIHYDROHYDROXY-S-GLUTATHIONYL CONJUGATE OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST, MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], IN RATSVijay Bhasker G. Reddy, George A. Doss, Mellissa Creighton, Christopher J. Kochansky, Stella H. Vincent, Ronald B. Franklin and Bindhu V. KaranamDrug Metabolism and Disposition October 2004, 32 (10) 1154-1161; DOI: https://doi.org/10.1124/dmd.104.000240
Vore, Mary
- You have accessESTRADIOL 3-GLUCURONIDE IS TRANSPORTED BY THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN 2 BUT DOES NOT ACTIVATE THE ALLOSTERIC SITE BOUND BY ESTRADIOL 17-GLUCURONIDEPhillip M. Gerk, Wei Li and Mary VoreDrug Metabolism and Disposition October 2004, 32 (10) 1139-1145; DOI: https://doi.org/10.1124/dmd.104.000372
W
Wang, Li-Quan
- You have accessTRICLOSAN AS A SUBSTRATE AND INHIBITOR OF 3′-PHOSPHOADENOSINE 5′-PHOSPHOSULFATE-SULFOTRANSFERASE AND UDP-GLUCURONOSYL TRANSFERASE IN HUMAN LIVER FRACTIONSLi-Quan Wang, Charles N. Falany and Margaret O. JamesDrug Metabolism and Disposition October 2004, 32 (10) 1162-1169; DOI: https://doi.org/10.1124/dmd.104.000273
Watkins, Paul B.
- You have accessTWO MAJOR GRAPEFRUIT JUICE COMPONENTS DIFFER IN INTESTINAL CYP3A4 INHIBITION KINETIC AND BINDING PROPERTIESMary F. Paine, Anne B. Criss and Paul B. WatkinsDrug Metabolism and Disposition October 2004, 32 (10) 1146-1153; DOI: https://doi.org/10.1124/dmd.104.000547
Welch, Christopher J.
- You have accessSPECIES DIFFERENTIAL STEREOSELECTIVE OXIDATION OF A METHYLSULFIDE METABOLITE OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DUAL AGONISTBindhu V. Karanam, Christopher J. Welch, Vijay G. Reddy, Jennifer Chilenski, Mirlinda Biba and Stella VincentDrug Metabolism and Disposition October 2004, 32 (10) 1061-1068; DOI: https://doi.org/10.1124/dmd.104.000224
Wu, Jing-Tao
- You have accessEFFECTIVE DOSING REGIMEN OF 1-AMINOBENZOTRIAZOLE FOR INHIBITION OF ANTIPYRINE CLEARANCE IN GUINEA PIGS AND MICE USING SERIAL SAMPLINGSuresh K. Balani, Ping Li, Joanne Nguyen, Kym Cardoza, Hang Zeng, Dun-Xue Mu, Jing-Tao Wu, Liang-Shang Gan and Frank W. LeeDrug Metabolism and Disposition October 2004, 32 (10) 1092-1095; DOI: https://doi.org/10.1124/dmd.104.000349
Y
Yamada, Hideyuki
- You have accessSIMULTANEOUS EXPRESSION OF GUINEA PIG UDP-GLUCURONOSYLTRANSFERASE 2B21 (UGT2B21) AND 2B22 IN COS-7 CELLS ENHANCES UGT2B21-CATALYZED CHLORAMPHENICOL GLUCURONIDATIONYuji Ishii, Aya Miyoshi, Daisuke Maji, Hideyuki Yamada and Kazuta OguriDrug Metabolism and Disposition October 2004, 32 (10) 1057-1060; DOI: https://doi.org/10.1124/dmd.32.10.1057
Yokoi, Tsuyoshi
- You have accessIDENTIFICATION OF THE CYTOSOLIC CARBOXYLESTERASE CATALYZING THE 5′-DEOXY-5-FLUOROCYTIDINE FORMATION FROM CAPECITABINE IN HUMAN LIVERToshiki Tabata, Miki Katoh, Shogo Tokudome, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition October 2004, 32 (10) 1103-1110; DOI: https://doi.org/10.1124/dmd.104.000554
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Zeng, Hang
- You have accessEFFECTIVE DOSING REGIMEN OF 1-AMINOBENZOTRIAZOLE FOR INHIBITION OF ANTIPYRINE CLEARANCE IN GUINEA PIGS AND MICE USING SERIAL SAMPLINGSuresh K. Balani, Ping Li, Joanne Nguyen, Kym Cardoza, Hang Zeng, Dun-Xue Mu, Jing-Tao Wu, Liang-Shang Gan and Frank W. LeeDrug Metabolism and Disposition October 2004, 32 (10) 1092-1095; DOI: https://doi.org/10.1124/dmd.104.000349
Zhou, Changcheng
- You have accessTOCOTRIENOLS ACTIVATE THE STEROID AND XENOBIOTIC RECEPTOR, SXR, AND SELECTIVELY REGULATE EXPRESSION OF ITS TARGET GENESChangcheng Zhou, Michelle M. Tabb, Asal Sadatrafiei, Felix Grün and Bruce BlumbergDrug Metabolism and Disposition October 2004, 32 (10) 1075-1082; DOI: https://doi.org/10.1124/dmd.104.000299