Index by author
December 01, 2004; Volume 32,Issue 12
A
Adachi, Yasuhisa
- You have accessIN VITRO AND IN VIVO CORRELATION OF THE INHIBITORY EFFECT OF CYCLOSPORIN A ON THE TRANSPORTER-MEDIATED HEPATIC UPTAKE OF CERIVASTATIN IN RATSYoshihisa Shitara, Masaru Hirano, Yasuhisa Adachi, Tomoo Itoh, Hitoshi Sato and Yuichi SugiyamaDrug Metabolism and Disposition December 2004, 32 (12) 1468-1475; DOI: https://doi.org/10.1124/dmd.32.12.1468
Alley, Michael C.
- You have accessFLUORINATED 2-(4-AMINO-3-METHYLPHENYL)BENZOTHIAZOLES INDUCE CYP1A1 EXPRESSION, BECOME METABOLIZED, AND BIND TO MACROMOLECULES IN SENSITIVE HUMAN CANCER CELLSEileen Brantley, Valentina Trapani, Michael C. Alley, Curtis D. Hose, Tracey D. Bradshaw, Malcolm F. G. Stevens, Edward A. Sausville and Sherman F. StinsonDrug Metabolism and Disposition December 2004, 32 (12) 1392-1401; DOI: https://doi.org/10.1124/dmd.104.001057
Alvarez-Diez, Teresa M.
- You have accessDETECTION OF GLUTATHIONE CONJUGATES DERIVED FROM 4-IPOMEANOL METABOLISM IN BILE OF RATS BY LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYTeresa M. Alvarez-Diez and Jiang ZhengDrug Metabolism and Disposition December 2004, 32 (12) 1345-1350; DOI: https://doi.org/10.1124/dmd.104.000406
Andersson, Tommy B.
- You have accessRESPONSE: PREDICTING THE CLEARANCE OF CYP2C9 SUBSTRATESTommy B. Andersson, Eva Bredberg, Hans Ericsson and Helena SjÖbergDrug Metabolism and Disposition December 2004, 32 (12) 1523; DOI: https://doi.org/10.1124/dmd.104.002329
Antonio, Laurence
- You have accessASSESSMENT OF CATECHOL INDUCTION AND GLUCURONIDATION IN RAT LIVER MICROSOMESEivor Elovaara, Jouni Mikkola, Leena Luukkanen, Laurence Antonio, Sylvie Fournel-Gigleux, Brian Burchell, Jacques Magdalou and Jyrki TaskinenDrug Metabolism and Disposition December 2004, 32 (12) 1426-1433; DOI: https://doi.org/10.1124/dmd.104.000992
Apak, T. Idil
- You have accessINTERACTIONS OF THE STEREOISOMERS OF α-HYDROXYTAMOXIFEN WITH HUMAN HYDROXYSTEROID SULFOTRANSFERASE SULT2A1 AND RAT HYDROXYSTEROID SULFOTRANSFERASE STAT. Idil Apak and Michael W. DuffelDrug Metabolism and Disposition December 2004, 32 (12) 1501-1508; DOI: https://doi.org/10.1124/dmd.104.000919
Ardlie, Kristin G.
- You have accessDIFFERENCES IN FMO2*1 ALLELIC FREQUENCY BETWEEN HISPANICS OF PUERTO RICAN AND MEXICAN DESCENTSharon K. Krueger, Lisbeth K. Siddens, Sarah R. Martin, Zhen Yu, Clifford B. Pereira, Erwin T. Cabacungan, Ronald N. Hines, Kristin G. Ardlie, Judy L. Raucy and David E. WilliamsDrug Metabolism and Disposition December 2004, 32 (12) 1337-1340; DOI: https://doi.org/10.1124/dmd.104.001099
B
Bai, Stephen A.
- You have accessTHE CHIMPANZEE (PAN TROGLODYTES) AS A PHARMACOKINETIC MODEL FOR SELECTION OF DRUG CANDIDATES: MODEL CHARACTERIZATION AND APPLICATIONHarvey Wong, Scott J. Grossman, Stephen A. Bai, Sharon Diamond, Matthew R. Wright, James E. Grace, Mingxin Qian, Kan He, Krishnaswamy Yeleswaram and David D. ChristDrug Metabolism and Disposition December 2004, 32 (12) 1359-1369; DOI: https://doi.org/10.1124/dmd.104.000943
Basu, N. K.
- You have accessRESPONSE TO THE LETTER TO THE EDITOR BY DRS. N. PICARD AND P. MARQUET REGARDING A PUBLICATION: BASU ET AL., DRUG METABOLISM AND DISPOSITION (32:768–773, (2004)N. K. Basu, L. Kole, S. Kubota and I. S. OwensDrug Metabolism and Disposition December 2004, 32 (12) 1525; DOI: https://doi.org/10.1124/dmd.104.002345
Berry, Pamela W.
- You have accessIDENTIFICATION OF GLUTATHIONE-DERIVED METABOLITES FROM AN IP RECEPTOR ANTAGONISTWilliam L. Fitch, Pamela W. Berry, Yaping Tu, Ali Tabatabaei, Lee Lowrie, Francisco Lopez-Tapia, Yanzhou Liu, Dov Nitzan, Mohammad R. Masjedizadeh and Aravamuthan VaradarajanDrug Metabolism and Disposition December 2004, 32 (12) 1482-1490; DOI: https://doi.org/10.1124/dmd.104.000471
Bradshaw, Tracey D.
- You have accessFLUORINATED 2-(4-AMINO-3-METHYLPHENYL)BENZOTHIAZOLES INDUCE CYP1A1 EXPRESSION, BECOME METABOLIZED, AND BIND TO MACROMOLECULES IN SENSITIVE HUMAN CANCER CELLSEileen Brantley, Valentina Trapani, Michael C. Alley, Curtis D. Hose, Tracey D. Bradshaw, Malcolm F. G. Stevens, Edward A. Sausville and Sherman F. StinsonDrug Metabolism and Disposition December 2004, 32 (12) 1392-1401; DOI: https://doi.org/10.1124/dmd.104.001057
Brantley, Eileen
- You have accessFLUORINATED 2-(4-AMINO-3-METHYLPHENYL)BENZOTHIAZOLES INDUCE CYP1A1 EXPRESSION, BECOME METABOLIZED, AND BIND TO MACROMOLECULES IN SENSITIVE HUMAN CANCER CELLSEileen Brantley, Valentina Trapani, Michael C. Alley, Curtis D. Hose, Tracey D. Bradshaw, Malcolm F. G. Stevens, Edward A. Sausville and Sherman F. StinsonDrug Metabolism and Disposition December 2004, 32 (12) 1392-1401; DOI: https://doi.org/10.1124/dmd.104.001057
Bredberg, Eva
- You have accessRESPONSE: PREDICTING THE CLEARANCE OF CYP2C9 SUBSTRATESTommy B. Andersson, Eva Bredberg, Hans Ericsson and Helena SjÖbergDrug Metabolism and Disposition December 2004, 32 (12) 1523; DOI: https://doi.org/10.1124/dmd.104.002329
Brown, Caroline
- You have accessUTILITY OF RECOMBINANT ENZYME KINETICS IN PREDICTION OF HUMAN CLEARANCE: IMPACT OF VARIABILITY, CYP3A5, AND CYP2C19 ON CYP3A4 PROBE SUBSTRATESAleksandra Galetin, Caroline Brown, David Hallifax, Kiyomi Ito and J. Brian HoustonDrug Metabolism and Disposition December 2004, 32 (12) 1411-1420; DOI: https://doi.org/10.1124/dmd.104.000844
Burchell, Brian
- You have accessASSESSMENT OF CATECHOL INDUCTION AND GLUCURONIDATION IN RAT LIVER MICROSOMESEivor Elovaara, Jouni Mikkola, Leena Luukkanen, Laurence Antonio, Sylvie Fournel-Gigleux, Brian Burchell, Jacques Magdalou and Jyrki TaskinenDrug Metabolism and Disposition December 2004, 32 (12) 1426-1433; DOI: https://doi.org/10.1124/dmd.104.000992
- You have accessIDENTIFICATION OF THE RABBIT LIVER UDP-GLUCURONOSYLTRANSFERASE CATALYZING THE GLUCURONIDATION OF 4-ETHOXYPHENYLUREA (DULCIN)Yoshihiro Uesawa, Adam G. Staines, Audrey O'Sullivan, Kiminori Mohri and Brian BurchellDrug Metabolism and Disposition December 2004, 32 (12) 1476-1481; DOI: https://doi.org/10.1124/dmd.104.001206
C
Cabacungan, Erwin T.
- You have accessDIFFERENCES IN FMO2*1 ALLELIC FREQUENCY BETWEEN HISPANICS OF PUERTO RICAN AND MEXICAN DESCENTSharon K. Krueger, Lisbeth K. Siddens, Sarah R. Martin, Zhen Yu, Clifford B. Pereira, Erwin T. Cabacungan, Ronald N. Hines, Kristin G. Ardlie, Judy L. Raucy and David E. WilliamsDrug Metabolism and Disposition December 2004, 32 (12) 1337-1340; DOI: https://doi.org/10.1124/dmd.104.001099
Calamia, Justina C.
- You have accessEVIDENCE OF SIGNIFICANT CONTRIBUTION FROM CYP3A5 TO HEPATIC DRUG METABOLISMWeili Huang, Yvonne S. Lin, Donavon J. McConn, Justina C. Calamia, Rheem A. Totah, Nina Isoherranen, Mary Glodowski and Kenneth E. ThummelDrug Metabolism and Disposition December 2004, 32 (12) 1434-1445; DOI: https://doi.org/10.1124/dmd.104.001313
Chauret, Nathalie
- You have accessUSE OF A BENZYLOXY-SUBSTITUTED LACTONE CYCLOOXYGENASE-2 INHIBITOR AS A SELECTIVE FLUORESCENT PROBE FOR CYP3A ACTIVITY IN PRIMARY CULTURED RAT AND HUMAN HEPATOCYTESDeborah A. Nicoll-Griffith, Nathalie Chauret, Robert Houle, Stephen H. Day, Michelle D'Antoni and José M. SilvaDrug Metabolism and Disposition December 2004, 32 (12) 1509-1515; DOI: https://doi.org/10.1124/dmd.32.12.1509
Chavin, Kenneth D.
- You have accessMULTIPLE NIGHT-TIME DOSES OF VALERIAN (Valeriana officinalis) HAD MINIMAL EFFECTS ON CYP3A4 ACTIVITY AND NO EFFECT ON CYP2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, C. Lindsay DeVane, Kenneth D. Chavin, Jun-Sheng Wang, Bryan B. Gibson, Holly A. Gefroh and John S. MarkowitzDrug Metabolism and Disposition December 2004, 32 (12) 1333-1336; DOI: https://doi.org/10.1124/dmd.104.001164
Chen, Chuan
- You have accessTISSUE DISTRIBUTION OF CONCENTRATIVE AND EQUILIBRATIVE NUCLEOSIDE TRANSPORTERS IN MALE AND FEMALE RATS AND MICEHong Lu, Chuan Chen and Curtis KlaassenDrug Metabolism and Disposition December 2004, 32 (12) 1455-1461; DOI: https://doi.org/10.1124/dmd.104.001123
Cho, Joo-Youn
- You have accessHAPLOTYPE STRUCTURE AND ALLELE FREQUENCIES OF CYP2B6 IN A KOREAN POPULATIONJoo-Youn Cho, Hyeong-Seok Lim, Jae-Yong Chung, Kyung-Sang Yu, Jung-Ryul Kim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition December 2004, 32 (12) 1341-1344; DOI: https://doi.org/10.1124/dmd.104.001107
Christ, David D.
- You have accessTHE CHIMPANZEE (PAN TROGLODYTES) AS A PHARMACOKINETIC MODEL FOR SELECTION OF DRUG CANDIDATES: MODEL CHARACTERIZATION AND APPLICATIONHarvey Wong, Scott J. Grossman, Stephen A. Bai, Sharon Diamond, Matthew R. Wright, James E. Grace, Mingxin Qian, Kan He, Krishnaswamy Yeleswaram and David D. ChristDrug Metabolism and Disposition December 2004, 32 (12) 1359-1369; DOI: https://doi.org/10.1124/dmd.104.000943
Chung, Jae-Yong
- You have accessHAPLOTYPE STRUCTURE AND ALLELE FREQUENCIES OF CYP2B6 IN A KOREAN POPULATIONJoo-Youn Cho, Hyeong-Seok Lim, Jae-Yong Chung, Kyung-Sang Yu, Jung-Ryul Kim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition December 2004, 32 (12) 1341-1344; DOI: https://doi.org/10.1124/dmd.104.001107
Claes, Kathleen
- You have accessTHE RATE OF GASTRIC EMPTYING DETERMINES THE TIMING BUT NOT THE EXTENT OF ORAL TACROLIMUS ABSORPTION: SIMULTANEOUS MEASUREMENT OF DRUG EXPOSURE AND GASTRIC EMPTYING BY CARBON-14-OCTANOIC ACID BREATH TEST IN STABLE RENAL ALLOGRAFT RECIPIENTSDirk R. J. Kuypers, Kathleen Claes, P. Evenepoel, B. Maes and Yves VanrenterghemDrug Metabolism and Disposition December 2004, 32 (12) 1421-1425; DOI: https://doi.org/10.1124/dmd.104.001503
D
D'Antoni, Michelle
- You have accessUSE OF A BENZYLOXY-SUBSTITUTED LACTONE CYCLOOXYGENASE-2 INHIBITOR AS A SELECTIVE FLUORESCENT PROBE FOR CYP3A ACTIVITY IN PRIMARY CULTURED RAT AND HUMAN HEPATOCYTESDeborah A. Nicoll-Griffith, Nathalie Chauret, Robert Houle, Stephen H. Day, Michelle D'Antoni and José M. SilvaDrug Metabolism and Disposition December 2004, 32 (12) 1509-1515; DOI: https://doi.org/10.1124/dmd.32.12.1509
Day, Stephen H.
- You have accessUSE OF A BENZYLOXY-SUBSTITUTED LACTONE CYCLOOXYGENASE-2 INHIBITOR AS A SELECTIVE FLUORESCENT PROBE FOR CYP3A ACTIVITY IN PRIMARY CULTURED RAT AND HUMAN HEPATOCYTESDeborah A. Nicoll-Griffith, Nathalie Chauret, Robert Houle, Stephen H. Day, Michelle D'Antoni and José M. SilvaDrug Metabolism and Disposition December 2004, 32 (12) 1509-1515; DOI: https://doi.org/10.1124/dmd.32.12.1509
DeLegge, Mark H.
- You have accessHIGH ABSORPTION BUT VERY LOW BIOAVAILABILITY OF ORAL RESVERATROL IN HUMANSThomas Walle, Faye Hsieh, Mark H. DeLegge, John E. Oatis and U. Kristina WalleDrug Metabolism and Disposition December 2004, 32 (12) 1377-1382; DOI: https://doi.org/10.1124/dmd.104.000885
DeVane, C. Lindsay
- You have accessMULTIPLE NIGHT-TIME DOSES OF VALERIAN (Valeriana officinalis) HAD MINIMAL EFFECTS ON CYP3A4 ACTIVITY AND NO EFFECT ON CYP2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, C. Lindsay DeVane, Kenneth D. Chavin, Jun-Sheng Wang, Bryan B. Gibson, Holly A. Gefroh and John S. MarkowitzDrug Metabolism and Disposition December 2004, 32 (12) 1333-1336; DOI: https://doi.org/10.1124/dmd.104.001164
Diamond, Sharon
- You have accessTHE CHIMPANZEE (PAN TROGLODYTES) AS A PHARMACOKINETIC MODEL FOR SELECTION OF DRUG CANDIDATES: MODEL CHARACTERIZATION AND APPLICATIONHarvey Wong, Scott J. Grossman, Stephen A. Bai, Sharon Diamond, Matthew R. Wright, James E. Grace, Mingxin Qian, Kan He, Krishnaswamy Yeleswaram and David D. ChristDrug Metabolism and Disposition December 2004, 32 (12) 1359-1369; DOI: https://doi.org/10.1124/dmd.104.000943
Ding, Xinxin
- You have accessIDENTIFICATION OF CRITICAL AMINO ACID RESIDUES OF HUMAN CYP2A13 FOR THE METABOLIC ACTIVATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE, A TOBACCO-SPECIFIC CARCINOGENXiao-Yang He, Jian Shen, Xinxin Ding, Anthony Y. H. Lu and Jun-Yan HongDrug Metabolism and Disposition December 2004, 32 (12) 1516-1521; DOI: https://doi.org/10.1124/dmd.104.001370
Donovan, Jennifer L.
- You have accessMULTIPLE NIGHT-TIME DOSES OF VALERIAN (Valeriana officinalis) HAD MINIMAL EFFECTS ON CYP3A4 ACTIVITY AND NO EFFECT ON CYP2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, C. Lindsay DeVane, Kenneth D. Chavin, Jun-Sheng Wang, Bryan B. Gibson, Holly A. Gefroh and John S. MarkowitzDrug Metabolism and Disposition December 2004, 32 (12) 1333-1336; DOI: https://doi.org/10.1124/dmd.104.001164
Duffel, Michael W.
- You have accessINTERACTIONS OF THE STEREOISOMERS OF α-HYDROXYTAMOXIFEN WITH HUMAN HYDROXYSTEROID SULFOTRANSFERASE SULT2A1 AND RAT HYDROXYSTEROID SULFOTRANSFERASE STAT. Idil Apak and Michael W. DuffelDrug Metabolism and Disposition December 2004, 32 (12) 1501-1508; DOI: https://doi.org/10.1124/dmd.104.000919
E
Elovaara, Eivor
- You have accessASSESSMENT OF CATECHOL INDUCTION AND GLUCURONIDATION IN RAT LIVER MICROSOMESEivor Elovaara, Jouni Mikkola, Leena Luukkanen, Laurence Antonio, Sylvie Fournel-Gigleux, Brian Burchell, Jacques Magdalou and Jyrki TaskinenDrug Metabolism and Disposition December 2004, 32 (12) 1426-1433; DOI: https://doi.org/10.1124/dmd.104.000992
Ericsson, Hans
- You have accessRESPONSE: PREDICTING THE CLEARANCE OF CYP2C9 SUBSTRATESTommy B. Andersson, Eva Bredberg, Hans Ericsson and Helena SjÖbergDrug Metabolism and Disposition December 2004, 32 (12) 1523; DOI: https://doi.org/10.1124/dmd.104.002329
Evenepoel, P.
- You have accessTHE RATE OF GASTRIC EMPTYING DETERMINES THE TIMING BUT NOT THE EXTENT OF ORAL TACROLIMUS ABSORPTION: SIMULTANEOUS MEASUREMENT OF DRUG EXPOSURE AND GASTRIC EMPTYING BY CARBON-14-OCTANOIC ACID BREATH TEST IN STABLE RENAL ALLOGRAFT RECIPIENTSDirk R. J. Kuypers, Kathleen Claes, P. Evenepoel, B. Maes and Yves VanrenterghemDrug Metabolism and Disposition December 2004, 32 (12) 1421-1425; DOI: https://doi.org/10.1124/dmd.104.001503
F
Fitch, William L.
- You have accessIDENTIFICATION OF GLUTATHIONE-DERIVED METABOLITES FROM AN IP RECEPTOR ANTAGONISTWilliam L. Fitch, Pamela W. Berry, Yaping Tu, Ali Tabatabaei, Lee Lowrie, Francisco Lopez-Tapia, Yanzhou Liu, Dov Nitzan, Mohammad R. Masjedizadeh and Aravamuthan VaradarajanDrug Metabolism and Disposition December 2004, 32 (12) 1482-1490; DOI: https://doi.org/10.1124/dmd.104.000471
Fournel-Gigleux, Sylvie
- You have accessASSESSMENT OF CATECHOL INDUCTION AND GLUCURONIDATION IN RAT LIVER MICROSOMESEivor Elovaara, Jouni Mikkola, Leena Luukkanen, Laurence Antonio, Sylvie Fournel-Gigleux, Brian Burchell, Jacques Magdalou and Jyrki TaskinenDrug Metabolism and Disposition December 2004, 32 (12) 1426-1433; DOI: https://doi.org/10.1124/dmd.104.000992
G
Galetin, Aleksandra
- You have accessUTILITY OF RECOMBINANT ENZYME KINETICS IN PREDICTION OF HUMAN CLEARANCE: IMPACT OF VARIABILITY, CYP3A5, AND CYP2C19 ON CYP3A4 PROBE SUBSTRATESAleksandra Galetin, Caroline Brown, David Hallifax, Kiyomi Ito and J. Brian HoustonDrug Metabolism and Disposition December 2004, 32 (12) 1411-1420; DOI: https://doi.org/10.1124/dmd.104.000844
Gefroh, Holly A.
- You have accessMULTIPLE NIGHT-TIME DOSES OF VALERIAN (Valeriana officinalis) HAD MINIMAL EFFECTS ON CYP3A4 ACTIVITY AND NO EFFECT ON CYP2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, C. Lindsay DeVane, Kenneth D. Chavin, Jun-Sheng Wang, Bryan B. Gibson, Holly A. Gefroh and John S. MarkowitzDrug Metabolism and Disposition December 2004, 32 (12) 1333-1336; DOI: https://doi.org/10.1124/dmd.104.001164
Ghoborah, Hesham
- You have accessMETABOLISM AND DISPOSITION OF CALCIMIMETIC AGENT CINACALCET HCL IN HUMANS AND ANIMAL MODELSGondi N. Kumar, Christopher Sproul, Leszek Poppe, Sharon Turner, Mark Gohdes, Hesham Ghoborah, Desmond Padhi and Lorin RoskosDrug Metabolism and Disposition December 2004, 32 (12) 1491-1500; DOI: https://doi.org/10.1124/dmd.104.000604
Gibson, Bryan B.
- You have accessMULTIPLE NIGHT-TIME DOSES OF VALERIAN (Valeriana officinalis) HAD MINIMAL EFFECTS ON CYP3A4 ACTIVITY AND NO EFFECT ON CYP2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, C. Lindsay DeVane, Kenneth D. Chavin, Jun-Sheng Wang, Bryan B. Gibson, Holly A. Gefroh and John S. MarkowitzDrug Metabolism and Disposition December 2004, 32 (12) 1333-1336; DOI: https://doi.org/10.1124/dmd.104.001164
Gibson, Gordon
- You have accessEFFECTS OF AVASIMIBE ON CYTOCHROME P450 2C9 EXPRESSION IN VITRO AND IN VIVOJasminder Sahi, Ralph H. Stern, Mark A. Milad, Kelly A. Rose, Gordon Gibson, Xianxian Zheng, Linda Stilgenbauer, Nalini Sadagopan, Summer Jolley, Darryl Gilbert and Edward L. LeCluyseDrug Metabolism and Disposition December 2004, 32 (12) 1370-1376; DOI: https://doi.org/10.1124/dmd.104.000208
Gilbert, Darryl
- You have accessEFFECTS OF AVASIMIBE ON CYTOCHROME P450 2C9 EXPRESSION IN VITRO AND IN VIVOJasminder Sahi, Ralph H. Stern, Mark A. Milad, Kelly A. Rose, Gordon Gibson, Xianxian Zheng, Linda Stilgenbauer, Nalini Sadagopan, Summer Jolley, Darryl Gilbert and Edward L. LeCluyseDrug Metabolism and Disposition December 2004, 32 (12) 1370-1376; DOI: https://doi.org/10.1124/dmd.104.000208
Glodowski, Mary
- You have accessEVIDENCE OF SIGNIFICANT CONTRIBUTION FROM CYP3A5 TO HEPATIC DRUG METABOLISMWeili Huang, Yvonne S. Lin, Donavon J. McConn, Justina C. Calamia, Rheem A. Totah, Nina Isoherranen, Mary Glodowski and Kenneth E. ThummelDrug Metabolism and Disposition December 2004, 32 (12) 1434-1445; DOI: https://doi.org/10.1124/dmd.104.001313
Gohdes, Mark
- You have accessMETABOLISM AND DISPOSITION OF CALCIMIMETIC AGENT CINACALCET HCL IN HUMANS AND ANIMAL MODELSGondi N. Kumar, Christopher Sproul, Leszek Poppe, Sharon Turner, Mark Gohdes, Hesham Ghoborah, Desmond Padhi and Lorin RoskosDrug Metabolism and Disposition December 2004, 32 (12) 1491-1500; DOI: https://doi.org/10.1124/dmd.104.000604
Grace, James E.
- You have accessTHE CHIMPANZEE (PAN TROGLODYTES) AS A PHARMACOKINETIC MODEL FOR SELECTION OF DRUG CANDIDATES: MODEL CHARACTERIZATION AND APPLICATIONHarvey Wong, Scott J. Grossman, Stephen A. Bai, Sharon Diamond, Matthew R. Wright, James E. Grace, Mingxin Qian, Kan He, Krishnaswamy Yeleswaram and David D. ChristDrug Metabolism and Disposition December 2004, 32 (12) 1359-1369; DOI: https://doi.org/10.1124/dmd.104.000943
Grossman, Scott J.
- You have accessTHE CHIMPANZEE (PAN TROGLODYTES) AS A PHARMACOKINETIC MODEL FOR SELECTION OF DRUG CANDIDATES: MODEL CHARACTERIZATION AND APPLICATIONHarvey Wong, Scott J. Grossman, Stephen A. Bai, Sharon Diamond, Matthew R. Wright, James E. Grace, Mingxin Qian, Kan He, Krishnaswamy Yeleswaram and David D. ChristDrug Metabolism and Disposition December 2004, 32 (12) 1359-1369; DOI: https://doi.org/10.1124/dmd.104.000943
H
Hallifax, David
- You have accessUTILITY OF RECOMBINANT ENZYME KINETICS IN PREDICTION OF HUMAN CLEARANCE: IMPACT OF VARIABILITY, CYP3A5, AND CYP2C19 ON CYP3A4 PROBE SUBSTRATESAleksandra Galetin, Caroline Brown, David Hallifax, Kiyomi Ito and J. Brian HoustonDrug Metabolism and Disposition December 2004, 32 (12) 1411-1420; DOI: https://doi.org/10.1124/dmd.104.000844
He, Kan
- You have accessTHE CHIMPANZEE (PAN TROGLODYTES) AS A PHARMACOKINETIC MODEL FOR SELECTION OF DRUG CANDIDATES: MODEL CHARACTERIZATION AND APPLICATIONHarvey Wong, Scott J. Grossman, Stephen A. Bai, Sharon Diamond, Matthew R. Wright, James E. Grace, Mingxin Qian, Kan He, Krishnaswamy Yeleswaram and David D. ChristDrug Metabolism and Disposition December 2004, 32 (12) 1359-1369; DOI: https://doi.org/10.1124/dmd.104.000943
He, Xiao-Yang
- You have accessIDENTIFICATION OF CRITICAL AMINO ACID RESIDUES OF HUMAN CYP2A13 FOR THE METABOLIC ACTIVATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE, A TOBACCO-SPECIFIC CARCINOGENXiao-Yang He, Jian Shen, Xinxin Ding, Anthony Y. H. Lu and Jun-Yan HongDrug Metabolism and Disposition December 2004, 32 (12) 1516-1521; DOI: https://doi.org/10.1124/dmd.104.001370
Hines, Ronald N.
- You have accessDIFFERENCES IN FMO2*1 ALLELIC FREQUENCY BETWEEN HISPANICS OF PUERTO RICAN AND MEXICAN DESCENTSharon K. Krueger, Lisbeth K. Siddens, Sarah R. Martin, Zhen Yu, Clifford B. Pereira, Erwin T. Cabacungan, Ronald N. Hines, Kristin G. Ardlie, Judy L. Raucy and David E. WilliamsDrug Metabolism and Disposition December 2004, 32 (12) 1337-1340; DOI: https://doi.org/10.1124/dmd.104.001099
Hirani, Vandana N.
- You have accessCONVERSION OF THE HIV PROTEASE INHIBITOR NELFINAVIR TO A BIOACTIVE METABOLITE BY HUMAN LIVER CYP2C19Vandana N. Hirani, Judy L. Raucy and Jerome M. LaskerDrug Metabolism and Disposition December 2004, 32 (12) 1462-1467; DOI: https://doi.org/10.1124/dmd.104.001743
Hirano, Masaru
- You have accessIN VITRO AND IN VIVO CORRELATION OF THE INHIBITORY EFFECT OF CYCLOSPORIN A ON THE TRANSPORTER-MEDIATED HEPATIC UPTAKE OF CERIVASTATIN IN RATSYoshihisa Shitara, Masaru Hirano, Yasuhisa Adachi, Tomoo Itoh, Hitoshi Sato and Yuichi SugiyamaDrug Metabolism and Disposition December 2004, 32 (12) 1468-1475; DOI: https://doi.org/10.1124/dmd.32.12.1468
Hiratsuka, Akira
- You have accessIDENTIFICATION AND CHARACTERIZATION OF POTENT CYP3A4 INHIBITORS IN SCHISANDRA FRUIT EXTRACTHiroshi Iwata, Yasuhiro Tezuka, Shigetoshi Kadota, Akira Hiratsuka and Tadashi WatabeDrug Metabolism and Disposition December 2004, 32 (12) 1351-1358; DOI: https://doi.org/10.1124/dmd.104.000646
Hong, Jun-Yan
- You have accessIDENTIFICATION OF CRITICAL AMINO ACID RESIDUES OF HUMAN CYP2A13 FOR THE METABOLIC ACTIVATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE, A TOBACCO-SPECIFIC CARCINOGENXiao-Yang He, Jian Shen, Xinxin Ding, Anthony Y. H. Lu and Jun-Yan HongDrug Metabolism and Disposition December 2004, 32 (12) 1516-1521; DOI: https://doi.org/10.1124/dmd.104.001370
Horie, Toru
- You have accessEXPRESSION OF HUMAN CYTOCHROMES P450 IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Miki Nakajima, Chise Tateno, Miho Kataoka, Yoshinori Soeno, Toru Horie, Kazuhide Iwasaki, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition December 2004, 32 (12) 1402-1410; DOI: https://doi.org/10.1124/dmd.104.001347
Hose, Curtis D.
- You have accessFLUORINATED 2-(4-AMINO-3-METHYLPHENYL)BENZOTHIAZOLES INDUCE CYP1A1 EXPRESSION, BECOME METABOLIZED, AND BIND TO MACROMOLECULES IN SENSITIVE HUMAN CANCER CELLSEileen Brantley, Valentina Trapani, Michael C. Alley, Curtis D. Hose, Tracey D. Bradshaw, Malcolm F. G. Stevens, Edward A. Sausville and Sherman F. StinsonDrug Metabolism and Disposition December 2004, 32 (12) 1392-1401; DOI: https://doi.org/10.1124/dmd.104.001057
Houle, Robert
- You have accessUSE OF A BENZYLOXY-SUBSTITUTED LACTONE CYCLOOXYGENASE-2 INHIBITOR AS A SELECTIVE FLUORESCENT PROBE FOR CYP3A ACTIVITY IN PRIMARY CULTURED RAT AND HUMAN HEPATOCYTESDeborah A. Nicoll-Griffith, Nathalie Chauret, Robert Houle, Stephen H. Day, Michelle D'Antoni and José M. SilvaDrug Metabolism and Disposition December 2004, 32 (12) 1509-1515; DOI: https://doi.org/10.1124/dmd.32.12.1509
Houston, J. Brian
- You have accessUTILITY OF RECOMBINANT ENZYME KINETICS IN PREDICTION OF HUMAN CLEARANCE: IMPACT OF VARIABILITY, CYP3A5, AND CYP2C19 ON CYP3A4 PROBE SUBSTRATESAleksandra Galetin, Caroline Brown, David Hallifax, Kiyomi Ito and J. Brian HoustonDrug Metabolism and Disposition December 2004, 32 (12) 1411-1420; DOI: https://doi.org/10.1124/dmd.104.000844
Howgate, Eleanor M.
- You have accessPREDICTING THE CLEARANCE OF CYP2C9 SUBSTRATESKaren Rowland Yeo, Eleanor M. Howgate, Geoffrey T. Tucker and Amin Rostami-HodjeganDrug Metabolism and Disposition December 2004, 32 (12) 1522; DOI: https://doi.org/10.1124/dmd.104.001792
Hsieh, Faye
- You have accessHIGH ABSORPTION BUT VERY LOW BIOAVAILABILITY OF ORAL RESVERATROL IN HUMANSThomas Walle, Faye Hsieh, Mark H. DeLegge, John E. Oatis and U. Kristina WalleDrug Metabolism and Disposition December 2004, 32 (12) 1377-1382; DOI: https://doi.org/10.1124/dmd.104.000885
Huang, Weili
- You have accessEVIDENCE OF SIGNIFICANT CONTRIBUTION FROM CYP3A5 TO HEPATIC DRUG METABOLISMWeili Huang, Yvonne S. Lin, Donavon J. McConn, Justina C. Calamia, Rheem A. Totah, Nina Isoherranen, Mary Glodowski and Kenneth E. ThummelDrug Metabolism and Disposition December 2004, 32 (12) 1434-1445; DOI: https://doi.org/10.1124/dmd.104.001313
I
Inagaki, Haruhisa
- You have accessMECHANISM OF THE DRUG INTERACTION BETWEEN VALPROIC ACID AND CARBAPENEM ANTIBIOTICS IN MONKEYS AND RATSYoshitsugu Nakajima, Minoru Mizobuchi, Masahiro Nakamura, Hidetoshi Takagi, Haruhisa Inagaki, Goro Kominami, Masahiro Koike and Toshiro YamaguchiDrug Metabolism and Disposition December 2004, 32 (12) 1383-1391; DOI: https://doi.org/10.1124/dmd.104.000661
Isoherranen, Nina
- You have accessEVIDENCE OF SIGNIFICANT CONTRIBUTION FROM CYP3A5 TO HEPATIC DRUG METABOLISMWeili Huang, Yvonne S. Lin, Donavon J. McConn, Justina C. Calamia, Rheem A. Totah, Nina Isoherranen, Mary Glodowski and Kenneth E. ThummelDrug Metabolism and Disposition December 2004, 32 (12) 1434-1445; DOI: https://doi.org/10.1124/dmd.104.001313
Ito, Kiyomi
- You have accessUTILITY OF RECOMBINANT ENZYME KINETICS IN PREDICTION OF HUMAN CLEARANCE: IMPACT OF VARIABILITY, CYP3A5, AND CYP2C19 ON CYP3A4 PROBE SUBSTRATESAleksandra Galetin, Caroline Brown, David Hallifax, Kiyomi Ito and J. Brian HoustonDrug Metabolism and Disposition December 2004, 32 (12) 1411-1420; DOI: https://doi.org/10.1124/dmd.104.000844
Itoh, Tomoo
- You have accessIN VITRO AND IN VIVO CORRELATION OF THE INHIBITORY EFFECT OF CYCLOSPORIN A ON THE TRANSPORTER-MEDIATED HEPATIC UPTAKE OF CERIVASTATIN IN RATSYoshihisa Shitara, Masaru Hirano, Yasuhisa Adachi, Tomoo Itoh, Hitoshi Sato and Yuichi SugiyamaDrug Metabolism and Disposition December 2004, 32 (12) 1468-1475; DOI: https://doi.org/10.1124/dmd.32.12.1468
Iwasaki, Kazuhide
- You have accessEXPRESSION OF HUMAN CYTOCHROMES P450 IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Miki Nakajima, Chise Tateno, Miho Kataoka, Yoshinori Soeno, Toru Horie, Kazuhide Iwasaki, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition December 2004, 32 (12) 1402-1410; DOI: https://doi.org/10.1124/dmd.104.001347
Iwata, Hiroshi
- You have accessIDENTIFICATION AND CHARACTERIZATION OF POTENT CYP3A4 INHIBITORS IN SCHISANDRA FRUIT EXTRACTHiroshi Iwata, Yasuhiro Tezuka, Shigetoshi Kadota, Akira Hiratsuka and Tadashi WatabeDrug Metabolism and Disposition December 2004, 32 (12) 1351-1358; DOI: https://doi.org/10.1124/dmd.104.000646
J
Jang, In-Jin
- You have accessHAPLOTYPE STRUCTURE AND ALLELE FREQUENCIES OF CYP2B6 IN A KOREAN POPULATIONJoo-Youn Cho, Hyeong-Seok Lim, Jae-Yong Chung, Kyung-Sang Yu, Jung-Ryul Kim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition December 2004, 32 (12) 1341-1344; DOI: https://doi.org/10.1124/dmd.104.001107
Jolley, Summer
- You have accessEFFECTS OF AVASIMIBE ON CYTOCHROME P450 2C9 EXPRESSION IN VITRO AND IN VIVOJasminder Sahi, Ralph H. Stern, Mark A. Milad, Kelly A. Rose, Gordon Gibson, Xianxian Zheng, Linda Stilgenbauer, Nalini Sadagopan, Summer Jolley, Darryl Gilbert and Edward L. LeCluyseDrug Metabolism and Disposition December 2004, 32 (12) 1370-1376; DOI: https://doi.org/10.1124/dmd.104.000208
K
Kadota, Shigetoshi
- You have accessIDENTIFICATION AND CHARACTERIZATION OF POTENT CYP3A4 INHIBITORS IN SCHISANDRA FRUIT EXTRACTHiroshi Iwata, Yasuhiro Tezuka, Shigetoshi Kadota, Akira Hiratsuka and Tadashi WatabeDrug Metabolism and Disposition December 2004, 32 (12) 1351-1358; DOI: https://doi.org/10.1124/dmd.104.000646
Kataoka, Miho
- You have accessEXPRESSION OF HUMAN CYTOCHROMES P450 IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Miki Nakajima, Chise Tateno, Miho Kataoka, Yoshinori Soeno, Toru Horie, Kazuhide Iwasaki, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition December 2004, 32 (12) 1402-1410; DOI: https://doi.org/10.1124/dmd.104.001347
Katoh, Miki
- You have accessEXPRESSION OF HUMAN CYTOCHROMES P450 IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Miki Nakajima, Chise Tateno, Miho Kataoka, Yoshinori Soeno, Toru Horie, Kazuhide Iwasaki, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition December 2004, 32 (12) 1402-1410; DOI: https://doi.org/10.1124/dmd.104.001347
Kim, Jung-Ryul
- You have accessHAPLOTYPE STRUCTURE AND ALLELE FREQUENCIES OF CYP2B6 IN A KOREAN POPULATIONJoo-Youn Cho, Hyeong-Seok Lim, Jae-Yong Chung, Kyung-Sang Yu, Jung-Ryul Kim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition December 2004, 32 (12) 1341-1344; DOI: https://doi.org/10.1124/dmd.104.001107
Klaassen, Curtis
- You have accessTISSUE DISTRIBUTION OF CONCENTRATIVE AND EQUILIBRATIVE NUCLEOSIDE TRANSPORTERS IN MALE AND FEMALE RATS AND MICEHong Lu, Chuan Chen and Curtis KlaassenDrug Metabolism and Disposition December 2004, 32 (12) 1455-1461; DOI: https://doi.org/10.1124/dmd.104.001123
Koike, Masahiro
- You have accessMECHANISM OF THE DRUG INTERACTION BETWEEN VALPROIC ACID AND CARBAPENEM ANTIBIOTICS IN MONKEYS AND RATSYoshitsugu Nakajima, Minoru Mizobuchi, Masahiro Nakamura, Hidetoshi Takagi, Haruhisa Inagaki, Goro Kominami, Masahiro Koike and Toshiro YamaguchiDrug Metabolism and Disposition December 2004, 32 (12) 1383-1391; DOI: https://doi.org/10.1124/dmd.104.000661
Kole, L.
- You have accessRESPONSE TO THE LETTER TO THE EDITOR BY DRS. N. PICARD AND P. MARQUET REGARDING A PUBLICATION: BASU ET AL., DRUG METABOLISM AND DISPOSITION (32:768–773, (2004)N. K. Basu, L. Kole, S. Kubota and I. S. OwensDrug Metabolism and Disposition December 2004, 32 (12) 1525; DOI: https://doi.org/10.1124/dmd.104.002345
Kominami, Goro
- You have accessMECHANISM OF THE DRUG INTERACTION BETWEEN VALPROIC ACID AND CARBAPENEM ANTIBIOTICS IN MONKEYS AND RATSYoshitsugu Nakajima, Minoru Mizobuchi, Masahiro Nakamura, Hidetoshi Takagi, Haruhisa Inagaki, Goro Kominami, Masahiro Koike and Toshiro YamaguchiDrug Metabolism and Disposition December 2004, 32 (12) 1383-1391; DOI: https://doi.org/10.1124/dmd.104.000661
Krueger, Sharon K.
- You have accessDIFFERENCES IN FMO2*1 ALLELIC FREQUENCY BETWEEN HISPANICS OF PUERTO RICAN AND MEXICAN DESCENTSharon K. Krueger, Lisbeth K. Siddens, Sarah R. Martin, Zhen Yu, Clifford B. Pereira, Erwin T. Cabacungan, Ronald N. Hines, Kristin G. Ardlie, Judy L. Raucy and David E. WilliamsDrug Metabolism and Disposition December 2004, 32 (12) 1337-1340; DOI: https://doi.org/10.1124/dmd.104.001099
Kubota, S.
- You have accessRESPONSE TO THE LETTER TO THE EDITOR BY DRS. N. PICARD AND P. MARQUET REGARDING A PUBLICATION: BASU ET AL., DRUG METABOLISM AND DISPOSITION (32:768–773, (2004)N. K. Basu, L. Kole, S. Kubota and I. S. OwensDrug Metabolism and Disposition December 2004, 32 (12) 1525; DOI: https://doi.org/10.1124/dmd.104.002345
Kumar, Gondi N.
- You have accessMETABOLISM AND DISPOSITION OF CALCIMIMETIC AGENT CINACALCET HCL IN HUMANS AND ANIMAL MODELSGondi N. Kumar, Christopher Sproul, Leszek Poppe, Sharon Turner, Mark Gohdes, Hesham Ghoborah, Desmond Padhi and Lorin RoskosDrug Metabolism and Disposition December 2004, 32 (12) 1491-1500; DOI: https://doi.org/10.1124/dmd.104.000604
Kuypers, Dirk R. J.
- You have accessTHE RATE OF GASTRIC EMPTYING DETERMINES THE TIMING BUT NOT THE EXTENT OF ORAL TACROLIMUS ABSORPTION: SIMULTANEOUS MEASUREMENT OF DRUG EXPOSURE AND GASTRIC EMPTYING BY CARBON-14-OCTANOIC ACID BREATH TEST IN STABLE RENAL ALLOGRAFT RECIPIENTSDirk R. J. Kuypers, Kathleen Claes, P. Evenepoel, B. Maes and Yves VanrenterghemDrug Metabolism and Disposition December 2004, 32 (12) 1421-1425; DOI: https://doi.org/10.1124/dmd.104.001503
L
Lasker, Jerome M.
- You have accessCONVERSION OF THE HIV PROTEASE INHIBITOR NELFINAVIR TO A BIOACTIVE METABOLITE BY HUMAN LIVER CYP2C19Vandana N. Hirani, Judy L. Raucy and Jerome M. LaskerDrug Metabolism and Disposition December 2004, 32 (12) 1462-1467; DOI: https://doi.org/10.1124/dmd.104.001743
LeCluyse, Edward L.
- You have accessEFFECTS OF AVASIMIBE ON CYTOCHROME P450 2C9 EXPRESSION IN VITRO AND IN VIVOJasminder Sahi, Ralph H. Stern, Mark A. Milad, Kelly A. Rose, Gordon Gibson, Xianxian Zheng, Linda Stilgenbauer, Nalini Sadagopan, Summer Jolley, Darryl Gilbert and Edward L. LeCluyseDrug Metabolism and Disposition December 2004, 32 (12) 1370-1376; DOI: https://doi.org/10.1124/dmd.104.000208
Lim, Hyeong-Seok
- You have accessHAPLOTYPE STRUCTURE AND ALLELE FREQUENCIES OF CYP2B6 IN A KOREAN POPULATIONJoo-Youn Cho, Hyeong-Seok Lim, Jae-Yong Chung, Kyung-Sang Yu, Jung-Ryul Kim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition December 2004, 32 (12) 1341-1344; DOI: https://doi.org/10.1124/dmd.104.001107
Lin, Yvonne S.
- You have accessEVIDENCE OF SIGNIFICANT CONTRIBUTION FROM CYP3A5 TO HEPATIC DRUG METABOLISMWeili Huang, Yvonne S. Lin, Donavon J. McConn, Justina C. Calamia, Rheem A. Totah, Nina Isoherranen, Mary Glodowski and Kenneth E. ThummelDrug Metabolism and Disposition December 2004, 32 (12) 1434-1445; DOI: https://doi.org/10.1124/dmd.104.001313
Liu, Yanzhou
- You have accessIDENTIFICATION OF GLUTATHIONE-DERIVED METABOLITES FROM AN IP RECEPTOR ANTAGONISTWilliam L. Fitch, Pamela W. Berry, Yaping Tu, Ali Tabatabaei, Lee Lowrie, Francisco Lopez-Tapia, Yanzhou Liu, Dov Nitzan, Mohammad R. Masjedizadeh and Aravamuthan VaradarajanDrug Metabolism and Disposition December 2004, 32 (12) 1482-1490; DOI: https://doi.org/10.1124/dmd.104.000471
Lopez-Tapia, Francisco
- You have accessIDENTIFICATION OF GLUTATHIONE-DERIVED METABOLITES FROM AN IP RECEPTOR ANTAGONISTWilliam L. Fitch, Pamela W. Berry, Yaping Tu, Ali Tabatabaei, Lee Lowrie, Francisco Lopez-Tapia, Yanzhou Liu, Dov Nitzan, Mohammad R. Masjedizadeh and Aravamuthan VaradarajanDrug Metabolism and Disposition December 2004, 32 (12) 1482-1490; DOI: https://doi.org/10.1124/dmd.104.000471
Lowrie, Lee
- You have accessIDENTIFICATION OF GLUTATHIONE-DERIVED METABOLITES FROM AN IP RECEPTOR ANTAGONISTWilliam L. Fitch, Pamela W. Berry, Yaping Tu, Ali Tabatabaei, Lee Lowrie, Francisco Lopez-Tapia, Yanzhou Liu, Dov Nitzan, Mohammad R. Masjedizadeh and Aravamuthan VaradarajanDrug Metabolism and Disposition December 2004, 32 (12) 1482-1490; DOI: https://doi.org/10.1124/dmd.104.000471
Lu, Anthony Y. H.
- You have accessIDENTIFICATION OF CRITICAL AMINO ACID RESIDUES OF HUMAN CYP2A13 FOR THE METABOLIC ACTIVATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE, A TOBACCO-SPECIFIC CARCINOGENXiao-Yang He, Jian Shen, Xinxin Ding, Anthony Y. H. Lu and Jun-Yan HongDrug Metabolism and Disposition December 2004, 32 (12) 1516-1521; DOI: https://doi.org/10.1124/dmd.104.001370
Lu, Hong
- You have accessTISSUE DISTRIBUTION OF CONCENTRATIVE AND EQUILIBRATIVE NUCLEOSIDE TRANSPORTERS IN MALE AND FEMALE RATS AND MICEHong Lu, Chuan Chen and Curtis KlaassenDrug Metabolism and Disposition December 2004, 32 (12) 1455-1461; DOI: https://doi.org/10.1124/dmd.104.001123
Luukkanen, Leena
- You have accessASSESSMENT OF CATECHOL INDUCTION AND GLUCURONIDATION IN RAT LIVER MICROSOMESEivor Elovaara, Jouni Mikkola, Leena Luukkanen, Laurence Antonio, Sylvie Fournel-Gigleux, Brian Burchell, Jacques Magdalou and Jyrki TaskinenDrug Metabolism and Disposition December 2004, 32 (12) 1426-1433; DOI: https://doi.org/10.1124/dmd.104.000992
M
Maes, B.
- You have accessTHE RATE OF GASTRIC EMPTYING DETERMINES THE TIMING BUT NOT THE EXTENT OF ORAL TACROLIMUS ABSORPTION: SIMULTANEOUS MEASUREMENT OF DRUG EXPOSURE AND GASTRIC EMPTYING BY CARBON-14-OCTANOIC ACID BREATH TEST IN STABLE RENAL ALLOGRAFT RECIPIENTSDirk R. J. Kuypers, Kathleen Claes, P. Evenepoel, B. Maes and Yves VanrenterghemDrug Metabolism and Disposition December 2004, 32 (12) 1421-1425; DOI: https://doi.org/10.1124/dmd.104.001503
Magdalou, Jacques
- You have accessASSESSMENT OF CATECHOL INDUCTION AND GLUCURONIDATION IN RAT LIVER MICROSOMESEivor Elovaara, Jouni Mikkola, Leena Luukkanen, Laurence Antonio, Sylvie Fournel-Gigleux, Brian Burchell, Jacques Magdalou and Jyrki TaskinenDrug Metabolism and Disposition December 2004, 32 (12) 1426-1433; DOI: https://doi.org/10.1124/dmd.104.000992
Markowitz, John S.
- You have accessMULTIPLE NIGHT-TIME DOSES OF VALERIAN (Valeriana officinalis) HAD MINIMAL EFFECTS ON CYP3A4 ACTIVITY AND NO EFFECT ON CYP2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, C. Lindsay DeVane, Kenneth D. Chavin, Jun-Sheng Wang, Bryan B. Gibson, Holly A. Gefroh and John S. MarkowitzDrug Metabolism and Disposition December 2004, 32 (12) 1333-1336; DOI: https://doi.org/10.1124/dmd.104.001164
Marquet, Pierre
- You have accessIN VITRO STUDY OF MYCOPHENOLIC ACID GLUCURONIDATIONNicolas Picard and Pierre MarquetDrug Metabolism and Disposition December 2004, 32 (12) 1524; DOI: https://doi.org/10.1124/dmd.104.001982
Martin, Sarah R.
- You have accessDIFFERENCES IN FMO2*1 ALLELIC FREQUENCY BETWEEN HISPANICS OF PUERTO RICAN AND MEXICAN DESCENTSharon K. Krueger, Lisbeth K. Siddens, Sarah R. Martin, Zhen Yu, Clifford B. Pereira, Erwin T. Cabacungan, Ronald N. Hines, Kristin G. Ardlie, Judy L. Raucy and David E. WilliamsDrug Metabolism and Disposition December 2004, 32 (12) 1337-1340; DOI: https://doi.org/10.1124/dmd.104.001099
Masjedizadeh, Mohammad R.
- You have accessIDENTIFICATION OF GLUTATHIONE-DERIVED METABOLITES FROM AN IP RECEPTOR ANTAGONISTWilliam L. Fitch, Pamela W. Berry, Yaping Tu, Ali Tabatabaei, Lee Lowrie, Francisco Lopez-Tapia, Yanzhou Liu, Dov Nitzan, Mohammad R. Masjedizadeh and Aravamuthan VaradarajanDrug Metabolism and Disposition December 2004, 32 (12) 1482-1490; DOI: https://doi.org/10.1124/dmd.104.000471
Matsui, Tomohito
- You have accessEXPRESSION OF HUMAN CYTOCHROMES P450 IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Miki Nakajima, Chise Tateno, Miho Kataoka, Yoshinori Soeno, Toru Horie, Kazuhide Iwasaki, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition December 2004, 32 (12) 1402-1410; DOI: https://doi.org/10.1124/dmd.104.001347
McConn, Donavon J.
- You have accessEVIDENCE OF SIGNIFICANT CONTRIBUTION FROM CYP3A5 TO HEPATIC DRUG METABOLISMWeili Huang, Yvonne S. Lin, Donavon J. McConn, Justina C. Calamia, Rheem A. Totah, Nina Isoherranen, Mary Glodowski and Kenneth E. ThummelDrug Metabolism and Disposition December 2004, 32 (12) 1434-1445; DOI: https://doi.org/10.1124/dmd.104.001313
Mehvar, Reza
- You have accessSHORT-TERM INHIBITORY EFFECTS OF NITRIC OXIDE ON CYTOCHROME P450-MEDIATED DRUG METABOLISM: TIME DEPENDENCY AND REVERSIBILITY PROFILES IN ISOLATED PERFUSED RAT LIVERSRagini Vuppugalla and Reza MehvarDrug Metabolism and Disposition December 2004, 32 (12) 1446-1454; DOI: https://doi.org/10.1124/dmd.104.001487
Mikkola, Jouni
- You have accessASSESSMENT OF CATECHOL INDUCTION AND GLUCURONIDATION IN RAT LIVER MICROSOMESEivor Elovaara, Jouni Mikkola, Leena Luukkanen, Laurence Antonio, Sylvie Fournel-Gigleux, Brian Burchell, Jacques Magdalou and Jyrki TaskinenDrug Metabolism and Disposition December 2004, 32 (12) 1426-1433; DOI: https://doi.org/10.1124/dmd.104.000992
Milad, Mark A.
- You have accessEFFECTS OF AVASIMIBE ON CYTOCHROME P450 2C9 EXPRESSION IN VITRO AND IN VIVOJasminder Sahi, Ralph H. Stern, Mark A. Milad, Kelly A. Rose, Gordon Gibson, Xianxian Zheng, Linda Stilgenbauer, Nalini Sadagopan, Summer Jolley, Darryl Gilbert and Edward L. LeCluyseDrug Metabolism and Disposition December 2004, 32 (12) 1370-1376; DOI: https://doi.org/10.1124/dmd.104.000208
Mizobuchi, Minoru
- You have accessMECHANISM OF THE DRUG INTERACTION BETWEEN VALPROIC ACID AND CARBAPENEM ANTIBIOTICS IN MONKEYS AND RATSYoshitsugu Nakajima, Minoru Mizobuchi, Masahiro Nakamura, Hidetoshi Takagi, Haruhisa Inagaki, Goro Kominami, Masahiro Koike and Toshiro YamaguchiDrug Metabolism and Disposition December 2004, 32 (12) 1383-1391; DOI: https://doi.org/10.1124/dmd.104.000661
Mohri, Kiminori
- You have accessIDENTIFICATION OF THE RABBIT LIVER UDP-GLUCURONOSYLTRANSFERASE CATALYZING THE GLUCURONIDATION OF 4-ETHOXYPHENYLUREA (DULCIN)Yoshihiro Uesawa, Adam G. Staines, Audrey O'Sullivan, Kiminori Mohri and Brian BurchellDrug Metabolism and Disposition December 2004, 32 (12) 1476-1481; DOI: https://doi.org/10.1124/dmd.104.001206
N
Nakajima, Miki
- You have accessEXPRESSION OF HUMAN CYTOCHROMES P450 IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Miki Nakajima, Chise Tateno, Miho Kataoka, Yoshinori Soeno, Toru Horie, Kazuhide Iwasaki, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition December 2004, 32 (12) 1402-1410; DOI: https://doi.org/10.1124/dmd.104.001347
Nakajima, Yoshitsugu
- You have accessMECHANISM OF THE DRUG INTERACTION BETWEEN VALPROIC ACID AND CARBAPENEM ANTIBIOTICS IN MONKEYS AND RATSYoshitsugu Nakajima, Minoru Mizobuchi, Masahiro Nakamura, Hidetoshi Takagi, Haruhisa Inagaki, Goro Kominami, Masahiro Koike and Toshiro YamaguchiDrug Metabolism and Disposition December 2004, 32 (12) 1383-1391; DOI: https://doi.org/10.1124/dmd.104.000661
Nakamura, Masahiro
- You have accessMECHANISM OF THE DRUG INTERACTION BETWEEN VALPROIC ACID AND CARBAPENEM ANTIBIOTICS IN MONKEYS AND RATSYoshitsugu Nakajima, Minoru Mizobuchi, Masahiro Nakamura, Hidetoshi Takagi, Haruhisa Inagaki, Goro Kominami, Masahiro Koike and Toshiro YamaguchiDrug Metabolism and Disposition December 2004, 32 (12) 1383-1391; DOI: https://doi.org/10.1124/dmd.104.000661
Nicoll-Griffith, Deborah A.
- You have accessUSE OF A BENZYLOXY-SUBSTITUTED LACTONE CYCLOOXYGENASE-2 INHIBITOR AS A SELECTIVE FLUORESCENT PROBE FOR CYP3A ACTIVITY IN PRIMARY CULTURED RAT AND HUMAN HEPATOCYTESDeborah A. Nicoll-Griffith, Nathalie Chauret, Robert Houle, Stephen H. Day, Michelle D'Antoni and José M. SilvaDrug Metabolism and Disposition December 2004, 32 (12) 1509-1515; DOI: https://doi.org/10.1124/dmd.32.12.1509
Nitzan, Dov
- You have accessIDENTIFICATION OF GLUTATHIONE-DERIVED METABOLITES FROM AN IP RECEPTOR ANTAGONISTWilliam L. Fitch, Pamela W. Berry, Yaping Tu, Ali Tabatabaei, Lee Lowrie, Francisco Lopez-Tapia, Yanzhou Liu, Dov Nitzan, Mohammad R. Masjedizadeh and Aravamuthan VaradarajanDrug Metabolism and Disposition December 2004, 32 (12) 1482-1490; DOI: https://doi.org/10.1124/dmd.104.000471
O
O'Sullivan, Audrey
- You have accessIDENTIFICATION OF THE RABBIT LIVER UDP-GLUCURONOSYLTRANSFERASE CATALYZING THE GLUCURONIDATION OF 4-ETHOXYPHENYLUREA (DULCIN)Yoshihiro Uesawa, Adam G. Staines, Audrey O'Sullivan, Kiminori Mohri and Brian BurchellDrug Metabolism and Disposition December 2004, 32 (12) 1476-1481; DOI: https://doi.org/10.1124/dmd.104.001206
Oatis, John E.
- You have accessHIGH ABSORPTION BUT VERY LOW BIOAVAILABILITY OF ORAL RESVERATROL IN HUMANSThomas Walle, Faye Hsieh, Mark H. DeLegge, John E. Oatis and U. Kristina WalleDrug Metabolism and Disposition December 2004, 32 (12) 1377-1382; DOI: https://doi.org/10.1124/dmd.104.000885
Owens, I. S.
- You have accessRESPONSE TO THE LETTER TO THE EDITOR BY DRS. N. PICARD AND P. MARQUET REGARDING A PUBLICATION: BASU ET AL., DRUG METABOLISM AND DISPOSITION (32:768–773, (2004)N. K. Basu, L. Kole, S. Kubota and I. S. OwensDrug Metabolism and Disposition December 2004, 32 (12) 1525; DOI: https://doi.org/10.1124/dmd.104.002345
P
Padhi, Desmond
- You have accessMETABOLISM AND DISPOSITION OF CALCIMIMETIC AGENT CINACALCET HCL IN HUMANS AND ANIMAL MODELSGondi N. Kumar, Christopher Sproul, Leszek Poppe, Sharon Turner, Mark Gohdes, Hesham Ghoborah, Desmond Padhi and Lorin RoskosDrug Metabolism and Disposition December 2004, 32 (12) 1491-1500; DOI: https://doi.org/10.1124/dmd.104.000604
Pereira, Clifford B.
- You have accessDIFFERENCES IN FMO2*1 ALLELIC FREQUENCY BETWEEN HISPANICS OF PUERTO RICAN AND MEXICAN DESCENTSharon K. Krueger, Lisbeth K. Siddens, Sarah R. Martin, Zhen Yu, Clifford B. Pereira, Erwin T. Cabacungan, Ronald N. Hines, Kristin G. Ardlie, Judy L. Raucy and David E. WilliamsDrug Metabolism and Disposition December 2004, 32 (12) 1337-1340; DOI: https://doi.org/10.1124/dmd.104.001099
Picard, Nicolas
- You have accessIN VITRO STUDY OF MYCOPHENOLIC ACID GLUCURONIDATIONNicolas Picard and Pierre MarquetDrug Metabolism and Disposition December 2004, 32 (12) 1524; DOI: https://doi.org/10.1124/dmd.104.001982
Poppe, Leszek
- You have accessMETABOLISM AND DISPOSITION OF CALCIMIMETIC AGENT CINACALCET HCL IN HUMANS AND ANIMAL MODELSGondi N. Kumar, Christopher Sproul, Leszek Poppe, Sharon Turner, Mark Gohdes, Hesham Ghoborah, Desmond Padhi and Lorin RoskosDrug Metabolism and Disposition December 2004, 32 (12) 1491-1500; DOI: https://doi.org/10.1124/dmd.104.000604
Q
Qian, Mingxin
- You have accessTHE CHIMPANZEE (PAN TROGLODYTES) AS A PHARMACOKINETIC MODEL FOR SELECTION OF DRUG CANDIDATES: MODEL CHARACTERIZATION AND APPLICATIONHarvey Wong, Scott J. Grossman, Stephen A. Bai, Sharon Diamond, Matthew R. Wright, James E. Grace, Mingxin Qian, Kan He, Krishnaswamy Yeleswaram and David D. ChristDrug Metabolism and Disposition December 2004, 32 (12) 1359-1369; DOI: https://doi.org/10.1124/dmd.104.000943
R
Raucy, Judy L.
- You have accessDIFFERENCES IN FMO2*1 ALLELIC FREQUENCY BETWEEN HISPANICS OF PUERTO RICAN AND MEXICAN DESCENTSharon K. Krueger, Lisbeth K. Siddens, Sarah R. Martin, Zhen Yu, Clifford B. Pereira, Erwin T. Cabacungan, Ronald N. Hines, Kristin G. Ardlie, Judy L. Raucy and David E. WilliamsDrug Metabolism and Disposition December 2004, 32 (12) 1337-1340; DOI: https://doi.org/10.1124/dmd.104.001099
- You have accessCONVERSION OF THE HIV PROTEASE INHIBITOR NELFINAVIR TO A BIOACTIVE METABOLITE BY HUMAN LIVER CYP2C19Vandana N. Hirani, Judy L. Raucy and Jerome M. LaskerDrug Metabolism and Disposition December 2004, 32 (12) 1462-1467; DOI: https://doi.org/10.1124/dmd.104.001743
Rose, Kelly A.
- You have accessEFFECTS OF AVASIMIBE ON CYTOCHROME P450 2C9 EXPRESSION IN VITRO AND IN VIVOJasminder Sahi, Ralph H. Stern, Mark A. Milad, Kelly A. Rose, Gordon Gibson, Xianxian Zheng, Linda Stilgenbauer, Nalini Sadagopan, Summer Jolley, Darryl Gilbert and Edward L. LeCluyseDrug Metabolism and Disposition December 2004, 32 (12) 1370-1376; DOI: https://doi.org/10.1124/dmd.104.000208
Roskos, Lorin
- You have accessMETABOLISM AND DISPOSITION OF CALCIMIMETIC AGENT CINACALCET HCL IN HUMANS AND ANIMAL MODELSGondi N. Kumar, Christopher Sproul, Leszek Poppe, Sharon Turner, Mark Gohdes, Hesham Ghoborah, Desmond Padhi and Lorin RoskosDrug Metabolism and Disposition December 2004, 32 (12) 1491-1500; DOI: https://doi.org/10.1124/dmd.104.000604
Rostami-Hodjegan, Amin
- You have accessPREDICTING THE CLEARANCE OF CYP2C9 SUBSTRATESKaren Rowland Yeo, Eleanor M. Howgate, Geoffrey T. Tucker and Amin Rostami-HodjeganDrug Metabolism and Disposition December 2004, 32 (12) 1522; DOI: https://doi.org/10.1124/dmd.104.001792
S
Sadagopan, Nalini
- You have accessEFFECTS OF AVASIMIBE ON CYTOCHROME P450 2C9 EXPRESSION IN VITRO AND IN VIVOJasminder Sahi, Ralph H. Stern, Mark A. Milad, Kelly A. Rose, Gordon Gibson, Xianxian Zheng, Linda Stilgenbauer, Nalini Sadagopan, Summer Jolley, Darryl Gilbert and Edward L. LeCluyseDrug Metabolism and Disposition December 2004, 32 (12) 1370-1376; DOI: https://doi.org/10.1124/dmd.104.000208
Sahi, Jasminder
- You have accessEFFECTS OF AVASIMIBE ON CYTOCHROME P450 2C9 EXPRESSION IN VITRO AND IN VIVOJasminder Sahi, Ralph H. Stern, Mark A. Milad, Kelly A. Rose, Gordon Gibson, Xianxian Zheng, Linda Stilgenbauer, Nalini Sadagopan, Summer Jolley, Darryl Gilbert and Edward L. LeCluyseDrug Metabolism and Disposition December 2004, 32 (12) 1370-1376; DOI: https://doi.org/10.1124/dmd.104.000208
Sato, Hitoshi
- You have accessIN VITRO AND IN VIVO CORRELATION OF THE INHIBITORY EFFECT OF CYCLOSPORIN A ON THE TRANSPORTER-MEDIATED HEPATIC UPTAKE OF CERIVASTATIN IN RATSYoshihisa Shitara, Masaru Hirano, Yasuhisa Adachi, Tomoo Itoh, Hitoshi Sato and Yuichi SugiyamaDrug Metabolism and Disposition December 2004, 32 (12) 1468-1475; DOI: https://doi.org/10.1124/dmd.32.12.1468
Sausville, Edward A.
- You have accessFLUORINATED 2-(4-AMINO-3-METHYLPHENYL)BENZOTHIAZOLES INDUCE CYP1A1 EXPRESSION, BECOME METABOLIZED, AND BIND TO MACROMOLECULES IN SENSITIVE HUMAN CANCER CELLSEileen Brantley, Valentina Trapani, Michael C. Alley, Curtis D. Hose, Tracey D. Bradshaw, Malcolm F. G. Stevens, Edward A. Sausville and Sherman F. StinsonDrug Metabolism and Disposition December 2004, 32 (12) 1392-1401; DOI: https://doi.org/10.1124/dmd.104.001057
Shen, Jian
- You have accessIDENTIFICATION OF CRITICAL AMINO ACID RESIDUES OF HUMAN CYP2A13 FOR THE METABOLIC ACTIVATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE, A TOBACCO-SPECIFIC CARCINOGENXiao-Yang He, Jian Shen, Xinxin Ding, Anthony Y. H. Lu and Jun-Yan HongDrug Metabolism and Disposition December 2004, 32 (12) 1516-1521; DOI: https://doi.org/10.1124/dmd.104.001370
Shin, Sang-Goo
- You have accessHAPLOTYPE STRUCTURE AND ALLELE FREQUENCIES OF CYP2B6 IN A KOREAN POPULATIONJoo-Youn Cho, Hyeong-Seok Lim, Jae-Yong Chung, Kyung-Sang Yu, Jung-Ryul Kim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition December 2004, 32 (12) 1341-1344; DOI: https://doi.org/10.1124/dmd.104.001107
Shitara, Yoshihisa
- You have accessIN VITRO AND IN VIVO CORRELATION OF THE INHIBITORY EFFECT OF CYCLOSPORIN A ON THE TRANSPORTER-MEDIATED HEPATIC UPTAKE OF CERIVASTATIN IN RATSYoshihisa Shitara, Masaru Hirano, Yasuhisa Adachi, Tomoo Itoh, Hitoshi Sato and Yuichi SugiyamaDrug Metabolism and Disposition December 2004, 32 (12) 1468-1475; DOI: https://doi.org/10.1124/dmd.32.12.1468
Siddens, Lisbeth K.
- You have accessDIFFERENCES IN FMO2*1 ALLELIC FREQUENCY BETWEEN HISPANICS OF PUERTO RICAN AND MEXICAN DESCENTSharon K. Krueger, Lisbeth K. Siddens, Sarah R. Martin, Zhen Yu, Clifford B. Pereira, Erwin T. Cabacungan, Ronald N. Hines, Kristin G. Ardlie, Judy L. Raucy and David E. WilliamsDrug Metabolism and Disposition December 2004, 32 (12) 1337-1340; DOI: https://doi.org/10.1124/dmd.104.001099
Silva, José M.
- You have accessUSE OF A BENZYLOXY-SUBSTITUTED LACTONE CYCLOOXYGENASE-2 INHIBITOR AS A SELECTIVE FLUORESCENT PROBE FOR CYP3A ACTIVITY IN PRIMARY CULTURED RAT AND HUMAN HEPATOCYTESDeborah A. Nicoll-Griffith, Nathalie Chauret, Robert Houle, Stephen H. Day, Michelle D'Antoni and José M. SilvaDrug Metabolism and Disposition December 2004, 32 (12) 1509-1515; DOI: https://doi.org/10.1124/dmd.32.12.1509
SjÖberg, Helena
- You have accessRESPONSE: PREDICTING THE CLEARANCE OF CYP2C9 SUBSTRATESTommy B. Andersson, Eva Bredberg, Hans Ericsson and Helena SjÖbergDrug Metabolism and Disposition December 2004, 32 (12) 1523; DOI: https://doi.org/10.1124/dmd.104.002329
Soeno, Yoshinori
- You have accessEXPRESSION OF HUMAN CYTOCHROMES P450 IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Miki Nakajima, Chise Tateno, Miho Kataoka, Yoshinori Soeno, Toru Horie, Kazuhide Iwasaki, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition December 2004, 32 (12) 1402-1410; DOI: https://doi.org/10.1124/dmd.104.001347
Sproul, Christopher
- You have accessMETABOLISM AND DISPOSITION OF CALCIMIMETIC AGENT CINACALCET HCL IN HUMANS AND ANIMAL MODELSGondi N. Kumar, Christopher Sproul, Leszek Poppe, Sharon Turner, Mark Gohdes, Hesham Ghoborah, Desmond Padhi and Lorin RoskosDrug Metabolism and Disposition December 2004, 32 (12) 1491-1500; DOI: https://doi.org/10.1124/dmd.104.000604
Staines, Adam G.
- You have accessIDENTIFICATION OF THE RABBIT LIVER UDP-GLUCURONOSYLTRANSFERASE CATALYZING THE GLUCURONIDATION OF 4-ETHOXYPHENYLUREA (DULCIN)Yoshihiro Uesawa, Adam G. Staines, Audrey O'Sullivan, Kiminori Mohri and Brian BurchellDrug Metabolism and Disposition December 2004, 32 (12) 1476-1481; DOI: https://doi.org/10.1124/dmd.104.001206
Stern, Ralph H.
- You have accessEFFECTS OF AVASIMIBE ON CYTOCHROME P450 2C9 EXPRESSION IN VITRO AND IN VIVOJasminder Sahi, Ralph H. Stern, Mark A. Milad, Kelly A. Rose, Gordon Gibson, Xianxian Zheng, Linda Stilgenbauer, Nalini Sadagopan, Summer Jolley, Darryl Gilbert and Edward L. LeCluyseDrug Metabolism and Disposition December 2004, 32 (12) 1370-1376; DOI: https://doi.org/10.1124/dmd.104.000208
Stevens, Malcolm F. G.
- You have accessFLUORINATED 2-(4-AMINO-3-METHYLPHENYL)BENZOTHIAZOLES INDUCE CYP1A1 EXPRESSION, BECOME METABOLIZED, AND BIND TO MACROMOLECULES IN SENSITIVE HUMAN CANCER CELLSEileen Brantley, Valentina Trapani, Michael C. Alley, Curtis D. Hose, Tracey D. Bradshaw, Malcolm F. G. Stevens, Edward A. Sausville and Sherman F. StinsonDrug Metabolism and Disposition December 2004, 32 (12) 1392-1401; DOI: https://doi.org/10.1124/dmd.104.001057
Stilgenbauer, Linda
- You have accessEFFECTS OF AVASIMIBE ON CYTOCHROME P450 2C9 EXPRESSION IN VITRO AND IN VIVOJasminder Sahi, Ralph H. Stern, Mark A. Milad, Kelly A. Rose, Gordon Gibson, Xianxian Zheng, Linda Stilgenbauer, Nalini Sadagopan, Summer Jolley, Darryl Gilbert and Edward L. LeCluyseDrug Metabolism and Disposition December 2004, 32 (12) 1370-1376; DOI: https://doi.org/10.1124/dmd.104.000208
Stinson, Sherman F.
- You have accessFLUORINATED 2-(4-AMINO-3-METHYLPHENYL)BENZOTHIAZOLES INDUCE CYP1A1 EXPRESSION, BECOME METABOLIZED, AND BIND TO MACROMOLECULES IN SENSITIVE HUMAN CANCER CELLSEileen Brantley, Valentina Trapani, Michael C. Alley, Curtis D. Hose, Tracey D. Bradshaw, Malcolm F. G. Stevens, Edward A. Sausville and Sherman F. StinsonDrug Metabolism and Disposition December 2004, 32 (12) 1392-1401; DOI: https://doi.org/10.1124/dmd.104.001057
Sugiyama, Yuichi
- You have accessIN VITRO AND IN VIVO CORRELATION OF THE INHIBITORY EFFECT OF CYCLOSPORIN A ON THE TRANSPORTER-MEDIATED HEPATIC UPTAKE OF CERIVASTATIN IN RATSYoshihisa Shitara, Masaru Hirano, Yasuhisa Adachi, Tomoo Itoh, Hitoshi Sato and Yuichi SugiyamaDrug Metabolism and Disposition December 2004, 32 (12) 1468-1475; DOI: https://doi.org/10.1124/dmd.32.12.1468
T
Tabatabaei, Ali
- You have accessIDENTIFICATION OF GLUTATHIONE-DERIVED METABOLITES FROM AN IP RECEPTOR ANTAGONISTWilliam L. Fitch, Pamela W. Berry, Yaping Tu, Ali Tabatabaei, Lee Lowrie, Francisco Lopez-Tapia, Yanzhou Liu, Dov Nitzan, Mohammad R. Masjedizadeh and Aravamuthan VaradarajanDrug Metabolism and Disposition December 2004, 32 (12) 1482-1490; DOI: https://doi.org/10.1124/dmd.104.000471
Takagi, Hidetoshi
- You have accessMECHANISM OF THE DRUG INTERACTION BETWEEN VALPROIC ACID AND CARBAPENEM ANTIBIOTICS IN MONKEYS AND RATSYoshitsugu Nakajima, Minoru Mizobuchi, Masahiro Nakamura, Hidetoshi Takagi, Haruhisa Inagaki, Goro Kominami, Masahiro Koike and Toshiro YamaguchiDrug Metabolism and Disposition December 2004, 32 (12) 1383-1391; DOI: https://doi.org/10.1124/dmd.104.000661
Taskinen, Jyrki
- You have accessASSESSMENT OF CATECHOL INDUCTION AND GLUCURONIDATION IN RAT LIVER MICROSOMESEivor Elovaara, Jouni Mikkola, Leena Luukkanen, Laurence Antonio, Sylvie Fournel-Gigleux, Brian Burchell, Jacques Magdalou and Jyrki TaskinenDrug Metabolism and Disposition December 2004, 32 (12) 1426-1433; DOI: https://doi.org/10.1124/dmd.104.000992
Tateno, Chise
- You have accessEXPRESSION OF HUMAN CYTOCHROMES P450 IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Miki Nakajima, Chise Tateno, Miho Kataoka, Yoshinori Soeno, Toru Horie, Kazuhide Iwasaki, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition December 2004, 32 (12) 1402-1410; DOI: https://doi.org/10.1124/dmd.104.001347
Tezuka, Yasuhiro
- You have accessIDENTIFICATION AND CHARACTERIZATION OF POTENT CYP3A4 INHIBITORS IN SCHISANDRA FRUIT EXTRACTHiroshi Iwata, Yasuhiro Tezuka, Shigetoshi Kadota, Akira Hiratsuka and Tadashi WatabeDrug Metabolism and Disposition December 2004, 32 (12) 1351-1358; DOI: https://doi.org/10.1124/dmd.104.000646
Thummel, Kenneth E.
- You have accessEVIDENCE OF SIGNIFICANT CONTRIBUTION FROM CYP3A5 TO HEPATIC DRUG METABOLISMWeili Huang, Yvonne S. Lin, Donavon J. McConn, Justina C. Calamia, Rheem A. Totah, Nina Isoherranen, Mary Glodowski and Kenneth E. ThummelDrug Metabolism and Disposition December 2004, 32 (12) 1434-1445; DOI: https://doi.org/10.1124/dmd.104.001313
Totah, Rheem A.
- You have accessEVIDENCE OF SIGNIFICANT CONTRIBUTION FROM CYP3A5 TO HEPATIC DRUG METABOLISMWeili Huang, Yvonne S. Lin, Donavon J. McConn, Justina C. Calamia, Rheem A. Totah, Nina Isoherranen, Mary Glodowski and Kenneth E. ThummelDrug Metabolism and Disposition December 2004, 32 (12) 1434-1445; DOI: https://doi.org/10.1124/dmd.104.001313
Trapani, Valentina
- You have accessFLUORINATED 2-(4-AMINO-3-METHYLPHENYL)BENZOTHIAZOLES INDUCE CYP1A1 EXPRESSION, BECOME METABOLIZED, AND BIND TO MACROMOLECULES IN SENSITIVE HUMAN CANCER CELLSEileen Brantley, Valentina Trapani, Michael C. Alley, Curtis D. Hose, Tracey D. Bradshaw, Malcolm F. G. Stevens, Edward A. Sausville and Sherman F. StinsonDrug Metabolism and Disposition December 2004, 32 (12) 1392-1401; DOI: https://doi.org/10.1124/dmd.104.001057
Tu, Yaping
- You have accessIDENTIFICATION OF GLUTATHIONE-DERIVED METABOLITES FROM AN IP RECEPTOR ANTAGONISTWilliam L. Fitch, Pamela W. Berry, Yaping Tu, Ali Tabatabaei, Lee Lowrie, Francisco Lopez-Tapia, Yanzhou Liu, Dov Nitzan, Mohammad R. Masjedizadeh and Aravamuthan VaradarajanDrug Metabolism and Disposition December 2004, 32 (12) 1482-1490; DOI: https://doi.org/10.1124/dmd.104.000471
Tucker, Geoffrey T.
- You have accessPREDICTING THE CLEARANCE OF CYP2C9 SUBSTRATESKaren Rowland Yeo, Eleanor M. Howgate, Geoffrey T. Tucker and Amin Rostami-HodjeganDrug Metabolism and Disposition December 2004, 32 (12) 1522; DOI: https://doi.org/10.1124/dmd.104.001792
Turner, Sharon
- You have accessMETABOLISM AND DISPOSITION OF CALCIMIMETIC AGENT CINACALCET HCL IN HUMANS AND ANIMAL MODELSGondi N. Kumar, Christopher Sproul, Leszek Poppe, Sharon Turner, Mark Gohdes, Hesham Ghoborah, Desmond Padhi and Lorin RoskosDrug Metabolism and Disposition December 2004, 32 (12) 1491-1500; DOI: https://doi.org/10.1124/dmd.104.000604
U
Uesawa, Yoshihiro
- You have accessIDENTIFICATION OF THE RABBIT LIVER UDP-GLUCURONOSYLTRANSFERASE CATALYZING THE GLUCURONIDATION OF 4-ETHOXYPHENYLUREA (DULCIN)Yoshihiro Uesawa, Adam G. Staines, Audrey O'Sullivan, Kiminori Mohri and Brian BurchellDrug Metabolism and Disposition December 2004, 32 (12) 1476-1481; DOI: https://doi.org/10.1124/dmd.104.001206
V
Vanrenterghem, Yves
- You have accessTHE RATE OF GASTRIC EMPTYING DETERMINES THE TIMING BUT NOT THE EXTENT OF ORAL TACROLIMUS ABSORPTION: SIMULTANEOUS MEASUREMENT OF DRUG EXPOSURE AND GASTRIC EMPTYING BY CARBON-14-OCTANOIC ACID BREATH TEST IN STABLE RENAL ALLOGRAFT RECIPIENTSDirk R. J. Kuypers, Kathleen Claes, P. Evenepoel, B. Maes and Yves VanrenterghemDrug Metabolism and Disposition December 2004, 32 (12) 1421-1425; DOI: https://doi.org/10.1124/dmd.104.001503
Varadarajan, Aravamuthan
- You have accessIDENTIFICATION OF GLUTATHIONE-DERIVED METABOLITES FROM AN IP RECEPTOR ANTAGONISTWilliam L. Fitch, Pamela W. Berry, Yaping Tu, Ali Tabatabaei, Lee Lowrie, Francisco Lopez-Tapia, Yanzhou Liu, Dov Nitzan, Mohammad R. Masjedizadeh and Aravamuthan VaradarajanDrug Metabolism and Disposition December 2004, 32 (12) 1482-1490; DOI: https://doi.org/10.1124/dmd.104.000471
Vuppugalla, Ragini
- You have accessSHORT-TERM INHIBITORY EFFECTS OF NITRIC OXIDE ON CYTOCHROME P450-MEDIATED DRUG METABOLISM: TIME DEPENDENCY AND REVERSIBILITY PROFILES IN ISOLATED PERFUSED RAT LIVERSRagini Vuppugalla and Reza MehvarDrug Metabolism and Disposition December 2004, 32 (12) 1446-1454; DOI: https://doi.org/10.1124/dmd.104.001487
W
Walle, Thomas
- You have accessHIGH ABSORPTION BUT VERY LOW BIOAVAILABILITY OF ORAL RESVERATROL IN HUMANSThomas Walle, Faye Hsieh, Mark H. DeLegge, John E. Oatis and U. Kristina WalleDrug Metabolism and Disposition December 2004, 32 (12) 1377-1382; DOI: https://doi.org/10.1124/dmd.104.000885
Walle, U. Kristina
- You have accessHIGH ABSORPTION BUT VERY LOW BIOAVAILABILITY OF ORAL RESVERATROL IN HUMANSThomas Walle, Faye Hsieh, Mark H. DeLegge, John E. Oatis and U. Kristina WalleDrug Metabolism and Disposition December 2004, 32 (12) 1377-1382; DOI: https://doi.org/10.1124/dmd.104.000885
Wang, Jun-Sheng
- You have accessMULTIPLE NIGHT-TIME DOSES OF VALERIAN (Valeriana officinalis) HAD MINIMAL EFFECTS ON CYP3A4 ACTIVITY AND NO EFFECT ON CYP2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, C. Lindsay DeVane, Kenneth D. Chavin, Jun-Sheng Wang, Bryan B. Gibson, Holly A. Gefroh and John S. MarkowitzDrug Metabolism and Disposition December 2004, 32 (12) 1333-1336; DOI: https://doi.org/10.1124/dmd.104.001164
Watabe, Tadashi
- You have accessIDENTIFICATION AND CHARACTERIZATION OF POTENT CYP3A4 INHIBITORS IN SCHISANDRA FRUIT EXTRACTHiroshi Iwata, Yasuhiro Tezuka, Shigetoshi Kadota, Akira Hiratsuka and Tadashi WatabeDrug Metabolism and Disposition December 2004, 32 (12) 1351-1358; DOI: https://doi.org/10.1124/dmd.104.000646
Williams, David E.
- You have accessDIFFERENCES IN FMO2*1 ALLELIC FREQUENCY BETWEEN HISPANICS OF PUERTO RICAN AND MEXICAN DESCENTSharon K. Krueger, Lisbeth K. Siddens, Sarah R. Martin, Zhen Yu, Clifford B. Pereira, Erwin T. Cabacungan, Ronald N. Hines, Kristin G. Ardlie, Judy L. Raucy and David E. WilliamsDrug Metabolism and Disposition December 2004, 32 (12) 1337-1340; DOI: https://doi.org/10.1124/dmd.104.001099
Wong, Harvey
- You have accessTHE CHIMPANZEE (PAN TROGLODYTES) AS A PHARMACOKINETIC MODEL FOR SELECTION OF DRUG CANDIDATES: MODEL CHARACTERIZATION AND APPLICATIONHarvey Wong, Scott J. Grossman, Stephen A. Bai, Sharon Diamond, Matthew R. Wright, James E. Grace, Mingxin Qian, Kan He, Krishnaswamy Yeleswaram and David D. ChristDrug Metabolism and Disposition December 2004, 32 (12) 1359-1369; DOI: https://doi.org/10.1124/dmd.104.000943
Wright, Matthew R.
- You have accessTHE CHIMPANZEE (PAN TROGLODYTES) AS A PHARMACOKINETIC MODEL FOR SELECTION OF DRUG CANDIDATES: MODEL CHARACTERIZATION AND APPLICATIONHarvey Wong, Scott J. Grossman, Stephen A. Bai, Sharon Diamond, Matthew R. Wright, James E. Grace, Mingxin Qian, Kan He, Krishnaswamy Yeleswaram and David D. ChristDrug Metabolism and Disposition December 2004, 32 (12) 1359-1369; DOI: https://doi.org/10.1124/dmd.104.000943
Y
Yamaguchi, Toshiro
- You have accessMECHANISM OF THE DRUG INTERACTION BETWEEN VALPROIC ACID AND CARBAPENEM ANTIBIOTICS IN MONKEYS AND RATSYoshitsugu Nakajima, Minoru Mizobuchi, Masahiro Nakamura, Hidetoshi Takagi, Haruhisa Inagaki, Goro Kominami, Masahiro Koike and Toshiro YamaguchiDrug Metabolism and Disposition December 2004, 32 (12) 1383-1391; DOI: https://doi.org/10.1124/dmd.104.000661
Yeleswaram, Krishnaswamy
- You have accessTHE CHIMPANZEE (PAN TROGLODYTES) AS A PHARMACOKINETIC MODEL FOR SELECTION OF DRUG CANDIDATES: MODEL CHARACTERIZATION AND APPLICATIONHarvey Wong, Scott J. Grossman, Stephen A. Bai, Sharon Diamond, Matthew R. Wright, James E. Grace, Mingxin Qian, Kan He, Krishnaswamy Yeleswaram and David D. ChristDrug Metabolism and Disposition December 2004, 32 (12) 1359-1369; DOI: https://doi.org/10.1124/dmd.104.000943
Yeo, Karen Rowland
- You have accessPREDICTING THE CLEARANCE OF CYP2C9 SUBSTRATESKaren Rowland Yeo, Eleanor M. Howgate, Geoffrey T. Tucker and Amin Rostami-HodjeganDrug Metabolism and Disposition December 2004, 32 (12) 1522; DOI: https://doi.org/10.1124/dmd.104.001792
Yokoi, Tsuyoshi
- You have accessEXPRESSION OF HUMAN CYTOCHROMES P450 IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Miki Nakajima, Chise Tateno, Miho Kataoka, Yoshinori Soeno, Toru Horie, Kazuhide Iwasaki, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition December 2004, 32 (12) 1402-1410; DOI: https://doi.org/10.1124/dmd.104.001347
Yoshizato, Katsutoshi
- You have accessEXPRESSION OF HUMAN CYTOCHROMES P450 IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Miki Nakajima, Chise Tateno, Miho Kataoka, Yoshinori Soeno, Toru Horie, Kazuhide Iwasaki, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition December 2004, 32 (12) 1402-1410; DOI: https://doi.org/10.1124/dmd.104.001347
Yu, Kyung-Sang
- You have accessHAPLOTYPE STRUCTURE AND ALLELE FREQUENCIES OF CYP2B6 IN A KOREAN POPULATIONJoo-Youn Cho, Hyeong-Seok Lim, Jae-Yong Chung, Kyung-Sang Yu, Jung-Ryul Kim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition December 2004, 32 (12) 1341-1344; DOI: https://doi.org/10.1124/dmd.104.001107
Yu, Zhen
- You have accessDIFFERENCES IN FMO2*1 ALLELIC FREQUENCY BETWEEN HISPANICS OF PUERTO RICAN AND MEXICAN DESCENTSharon K. Krueger, Lisbeth K. Siddens, Sarah R. Martin, Zhen Yu, Clifford B. Pereira, Erwin T. Cabacungan, Ronald N. Hines, Kristin G. Ardlie, Judy L. Raucy and David E. WilliamsDrug Metabolism and Disposition December 2004, 32 (12) 1337-1340; DOI: https://doi.org/10.1124/dmd.104.001099
Z
Zheng, Jiang
- You have accessDETECTION OF GLUTATHIONE CONJUGATES DERIVED FROM 4-IPOMEANOL METABOLISM IN BILE OF RATS BY LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYTeresa M. Alvarez-Diez and Jiang ZhengDrug Metabolism and Disposition December 2004, 32 (12) 1345-1350; DOI: https://doi.org/10.1124/dmd.104.000406
Zheng, Xianxian
- You have accessEFFECTS OF AVASIMIBE ON CYTOCHROME P450 2C9 EXPRESSION IN VITRO AND IN VIVOJasminder Sahi, Ralph H. Stern, Mark A. Milad, Kelly A. Rose, Gordon Gibson, Xianxian Zheng, Linda Stilgenbauer, Nalini Sadagopan, Summer Jolley, Darryl Gilbert and Edward L. LeCluyseDrug Metabolism and Disposition December 2004, 32 (12) 1370-1376; DOI: https://doi.org/10.1124/dmd.104.000208