Index by author
September 01, 2004; Volume 32,Issue 9
A
Ahlf, Susan B.
- You have accessKINETIC CHARACTERIZATION OF P-GLYCOPROTEIN-MEDIATED EFFLUX OF RHODAMINE 6G IN THE INTACT RABBIT LUNGDavid L. Roerig, Said H. Audi and Susan B. AhlfDrug Metabolism and Disposition September 2004, 32 (9) 953-958; DOI: https://doi.org/10.1124/dmd.104.000042
Ali, Rabia Y.
- You have accessEFFECT OF PROTOTYPICAL INDUCING AGENTS ON P-GLYCOPROTEIN AND CYP3A EXPRESSION IN MOUSE TISSUESChristopher J. Matheny, Rabia Y. Ali, Xiaodong Yang and Gary M. PollackDrug Metabolism and Disposition September 2004, 32 (9) 1008-1014;
Ali, Shazia Y.
- You have accessALTERED PHARMACOKINETICS OF OMEPRAZOLE IN CYSTIC FIBROSIS KNOCKOUT MICE RELATIVE TO WILD-TYPE MICEMelanie N. Tallman, Shazia Y. Ali and Philip C. SmithDrug Metabolism and Disposition September 2004, 32 (9) 902-905;
Audi, Said H.
- You have accessKINETIC CHARACTERIZATION OF P-GLYCOPROTEIN-MEDIATED EFFLUX OF RHODAMINE 6G IN THE INTACT RABBIT LUNGDavid L. Roerig, Said H. Audi and Susan B. AhlfDrug Metabolism and Disposition September 2004, 32 (9) 953-958; DOI: https://doi.org/10.1124/dmd.104.000042
Awano, Katsuya
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. I. ROLE OF CYTOCHROME P450, METHYLTRANSFERASES, FLAVIN MONOOXYGENASES, AND ESTERASESBindhu V. Karanam, Cornelis E.C.A. Hop, David Q. Liu, Mike Wallace, Dennis Dean, Hiroya Satoh, Masakatsu Komuro, Katsuya Awano and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 1015-1022; DOI: https://doi.org/10.1124/dmd.104.000034
B
Baldwin, R. Michael
- You have accessBIOACTIVATION OF 1,1-DICHLOROETHYLENE TO ITS EPOXIDE BY CYP2E1 AND CYP2F ENZYMESAndrea C. Simmonds, Christopher A. Reilly, R. Michael Baldwin, Burhan I. Ghanayem, Diane L. Lanza, Garold S. Yost, Kathy S. Collins and Poh-Gek ForkertDrug Metabolism and Disposition September 2004, 32 (9) 1032-1039;
Barbuch, Robert J.
- You have accessSELECTIVE REDUCTION OF N-OXIDES TO AMINES: APPLICATION TO DRUG METABOLISMPalaniappan Kulanthaivel, Robert J. Barbuch, Rita S. Davidson, Ping Yi, Gregory A. Rener, Edward L. Mattiuz, Chad E. Hadden, Lawrence A. Goodwin and William J. EhlhardtDrug Metabolism and Disposition September 2004, 32 (9) 966-972;
Bergstrand, S.
- You have accessPHARMACOKINETICS AND METABOLISM OF TESAGLITAZAR, A NOVEL DUAL-ACTING PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST, AFTER A SINGLE ORAL AND INTRAVENOUS DOSE IN HUMANSH. Ericsson, B. Hamrén, S. Bergstrand, M. Elebring, L. Fryklund, M. Heijer and K. P. ÖhmanDrug Metabolism and Disposition September 2004, 32 (9) 923-929;
Bickel, Ulrich
- You have accessEFFECT OF POLY(ETHYLENE IMINE) MOLECULAR WEIGHT AND PEGYLATION ON ORGAN DISTRIBUTION AND PHARMACOKINETICS OF POLYPLEXES WITH OLIGODEOXYNUCLEOTIDES IN MICEDagmar Fischer, Berit Osburg, Holger Petersen, Thomas Kissel and Ulrich BickelDrug Metabolism and Disposition September 2004, 32 (9) 983-992;
Blair, Ian A.
- You have accessKINETICS AND REGULATION OF CYTOCHROME P450-MEDIATED ETOPOSIDE METABOLISMXiaoliang Zhuo, Naiyu Zheng, Carolyn A. Felix and Ian A. BlairDrug Metabolism and Disposition September 2004, 32 (9) 993-1000;
Breyer-Pfaff, Ursula
- You have accessENANTIOSELECTIVITY OF CARBONYL REDUCTION OF 4-METHYLNITROSAMINO-1-(3-PYRIDYL)-1-BUTANONE BY TISSUE FRACTIONS FROM HUMAN AND RAT AND BY ENZYMES ISOLATED FROM HUMAN LIVERUrsula Breyer-Pfaff, Hans-Jörg Martin, Michael Ernst and Edmund MaserDrug Metabolism and Disposition September 2004, 32 (9) 915-922;
C
Chavin, Kenneth D.
- You have accessGREEN TEA (CAMELLIA SINENSIS) EXTRACT DOES NOT ALTER CYTOCHROME P450 3A4 OR 2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, Kenneth D. Chavin, C. Lindsay Devane, Robin M. Taylor, Jun-Sheng Wang, Ying Ruan and John S. MarkowitzDrug Metabolism and Disposition September 2004, 32 (9) 906-908; DOI: https://doi.org/10.1124/dmd.104.000083
Chen, Yung-Hsiang
- You have accessEVALUATION OF A NOVEL IN VITRO CACO-2 HEPATOCYTE HYBRID SYSTEM FOR PREDICTING IN VIVO ORAL BIOAVAILABILITYYau Yi Lau, Yung-Hsiang Chen, Tong-tong Liu, Cheng Li, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition September 2004, 32 (9) 937-942;
Cheng, K.-C.
- You have accessEVALUATION OF A NOVEL IN VITRO CACO-2 HEPATOCYTE HYBRID SYSTEM FOR PREDICTING IN VIVO ORAL BIOAVAILABILITYYau Yi Lau, Yung-Hsiang Chen, Tong-tong Liu, Cheng Li, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition September 2004, 32 (9) 937-942;
Cho, Il Je
- You have accessCERAMIDE, AN APOPTOTIC RHEOSTAT, INHIBITS CCAAT/ENHANCER BINDING PROTEIN-β AND NF-E2-RELATED FACTOR-2 ACTIVATION: THE ROLE IN GLUTATHIONE S-TRANSFERASE A2 GENE REPRESSIONI-Na Park, Il Je Cho and Sang Geon KimDrug Metabolism and Disposition September 2004, 32 (9) 893-897;
Collins, Kathy S.
- You have accessBIOACTIVATION OF 1,1-DICHLOROETHYLENE TO ITS EPOXIDE BY CYP2E1 AND CYP2F ENZYMESAndrea C. Simmonds, Christopher A. Reilly, R. Michael Baldwin, Burhan I. Ghanayem, Diane L. Lanza, Garold S. Yost, Kathy S. Collins and Poh-Gek ForkertDrug Metabolism and Disposition September 2004, 32 (9) 1032-1039;
Cui, Xiaoming
- You have accessEVALUATION OF A NOVEL IN VITRO CACO-2 HEPATOCYTE HYBRID SYSTEM FOR PREDICTING IN VIVO ORAL BIOAVAILABILITYYau Yi Lau, Yung-Hsiang Chen, Tong-tong Liu, Cheng Li, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition September 2004, 32 (9) 937-942;
D
Davidson, Rita S.
- You have accessSELECTIVE REDUCTION OF N-OXIDES TO AMINES: APPLICATION TO DRUG METABOLISMPalaniappan Kulanthaivel, Robert J. Barbuch, Rita S. Davidson, Ping Yi, Gregory A. Rener, Edward L. Mattiuz, Chad E. Hadden, Lawrence A. Goodwin and William J. EhlhardtDrug Metabolism and Disposition September 2004, 32 (9) 966-972;
Dean, Dennis
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. I. ROLE OF CYTOCHROME P450, METHYLTRANSFERASES, FLAVIN MONOOXYGENASES, AND ESTERASESBindhu V. Karanam, Cornelis E.C.A. Hop, David Q. Liu, Mike Wallace, Dennis Dean, Hiroya Satoh, Masakatsu Komuro, Katsuya Awano and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 1015-1022; DOI: https://doi.org/10.1124/dmd.104.000034
de la Torre, Rafael
- You have accessSTEREOCHEMICAL ANALYSIS OF 3,4-METHYLENEDIOXYMETHAMPHETAMINE AND ITS MAIN METABOLITES IN HUMAN SAMPLES INCLUDING THE CATECHOL-TYPE METABOLITE (3,4-DIHYDROXYMETHAMPHETAMINE)Nieves Pizarro, Magí Farré, Mitona Pujadas, Ana Ma͢ Peiró, Pere N Roset, Jesús Joglar and Rafael de la TorreDrug Metabolism and Disposition September 2004, 32 (9) 1001-1007;
Devane, C. Lindsay
- You have accessGREEN TEA (CAMELLIA SINENSIS) EXTRACT DOES NOT ALTER CYTOCHROME P450 3A4 OR 2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, Kenneth D. Chavin, C. Lindsay Devane, Robin M. Taylor, Jun-Sheng Wang, Ying Ruan and John S. MarkowitzDrug Metabolism and Disposition September 2004, 32 (9) 906-908; DOI: https://doi.org/10.1124/dmd.104.000083
Donovan, Jennifer L.
- You have accessGREEN TEA (CAMELLIA SINENSIS) EXTRACT DOES NOT ALTER CYTOCHROME P450 3A4 OR 2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, Kenneth D. Chavin, C. Lindsay Devane, Robin M. Taylor, Jun-Sheng Wang, Ying Ruan and John S. MarkowitzDrug Metabolism and Disposition September 2004, 32 (9) 906-908; DOI: https://doi.org/10.1124/dmd.104.000083
Doss, George A.
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)-PHENYL] METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. II. IDENTIFICATION OF METABOLITES BY LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYDavid Q. Liu, Bindhu V. Karanam, George A. Doss, Rick R. Sidler, Stella H. Vincent and Cornelis E.C.A. HopDrug Metabolism and Disposition September 2004, 32 (9) 1023-1031; DOI: https://doi.org/10.1124/dmd.104.000059
E
Ehlhardt, William J.
- You have accessSELECTIVE REDUCTION OF N-OXIDES TO AMINES: APPLICATION TO DRUG METABOLISMPalaniappan Kulanthaivel, Robert J. Barbuch, Rita S. Davidson, Ping Yi, Gregory A. Rener, Edward L. Mattiuz, Chad E. Hadden, Lawrence A. Goodwin and William J. EhlhardtDrug Metabolism and Disposition September 2004, 32 (9) 966-972;
Elebring, M.
- You have accessPHARMACOKINETICS AND METABOLISM OF TESAGLITAZAR, A NOVEL DUAL-ACTING PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST, AFTER A SINGLE ORAL AND INTRAVENOUS DOSE IN HUMANSH. Ericsson, B. Hamrén, S. Bergstrand, M. Elebring, L. Fryklund, M. Heijer and K. P. ÖhmanDrug Metabolism and Disposition September 2004, 32 (9) 923-929;
Endou, Hitoshi
- You have accessCARRIER-MEDIATED UPTAKE OF H2-RECEPTOR ANTAGONISTS BY THE RAT CHOROID PLEXUS: INVOLVEMENT OF RAT ORGANIC ANION TRANSPORTER 3Yoshinori Nagata, Hiroyuki Kusuhara, Shuichi Hirono, Hitoshi Endou and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 1040-1047;
Ericsson, H.
- You have accessPHARMACOKINETICS AND METABOLISM OF TESAGLITAZAR, A NOVEL DUAL-ACTING PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST, AFTER A SINGLE ORAL AND INTRAVENOUS DOSE IN HUMANSH. Ericsson, B. Hamrén, S. Bergstrand, M. Elebring, L. Fryklund, M. Heijer and K. P. ÖhmanDrug Metabolism and Disposition September 2004, 32 (9) 923-929;
Ernst, Michael
- You have accessENANTIOSELECTIVITY OF CARBONYL REDUCTION OF 4-METHYLNITROSAMINO-1-(3-PYRIDYL)-1-BUTANONE BY TISSUE FRACTIONS FROM HUMAN AND RAT AND BY ENZYMES ISOLATED FROM HUMAN LIVERUrsula Breyer-Pfaff, Hans-Jörg Martin, Michael Ernst and Edmund MaserDrug Metabolism and Disposition September 2004, 32 (9) 915-922;
F
Farré, Magí
- You have accessSTEREOCHEMICAL ANALYSIS OF 3,4-METHYLENEDIOXYMETHAMPHETAMINE AND ITS MAIN METABOLITES IN HUMAN SAMPLES INCLUDING THE CATECHOL-TYPE METABOLITE (3,4-DIHYDROXYMETHAMPHETAMINE)Nieves Pizarro, Magí Farré, Mitona Pujadas, Ana Ma͢ Peiró, Pere N Roset, Jesús Joglar and Rafael de la TorreDrug Metabolism and Disposition September 2004, 32 (9) 1001-1007;
Felix, Carolyn A.
- You have accessKINETICS AND REGULATION OF CYTOCHROME P450-MEDIATED ETOPOSIDE METABOLISMXiaoliang Zhuo, Naiyu Zheng, Carolyn A. Felix and Ian A. BlairDrug Metabolism and Disposition September 2004, 32 (9) 993-1000;
Fischer, Dagmar
- You have accessEFFECT OF POLY(ETHYLENE IMINE) MOLECULAR WEIGHT AND PEGYLATION ON ORGAN DISTRIBUTION AND PHARMACOKINETICS OF POLYPLEXES WITH OLIGODEOXYNUCLEOTIDES IN MICEDagmar Fischer, Berit Osburg, Holger Petersen, Thomas Kissel and Ulrich BickelDrug Metabolism and Disposition September 2004, 32 (9) 983-992;
Flockhart, David A.
- You have accessCYP2B6, CYP3A4, AND CYP2C19 ARE RESPONSIBLE FOR THE IN VITRO N-DEMETHYLATION OF MEPERIDINE IN HUMAN LIVER MICROSOMESJacqueline Ramírez, Federico Innocenti, Erin G. Schuetz, David A. Flockhart, Mary V. Relling, Raymond Santucci and Mark J. RatainDrug Metabolism and Disposition September 2004, 32 (9) 930-936;
Forkert, Poh-Gek
- You have accessBIOACTIVATION OF 1,1-DICHLOROETHYLENE TO ITS EPOXIDE BY CYP2E1 AND CYP2F ENZYMESAndrea C. Simmonds, Christopher A. Reilly, R. Michael Baldwin, Burhan I. Ghanayem, Diane L. Lanza, Garold S. Yost, Kathy S. Collins and Poh-Gek ForkertDrug Metabolism and Disposition September 2004, 32 (9) 1032-1039;
Franklin, Ronald B.
- You have accessDIFFERENCES IN THE PHARMACOKINETICS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONISTS IN GENETICALLY OBESE ZUCKER AND SPRAGUE-DAWLEY RATS: IMPLICATIONS OF DECREASED GLUCURONIDATION IN OBESE ZUCKER RATSMi-Sook Kim, Sui Wang, Zhongzhou Shen, Christopher J. Kochansky, John R. Strauss, Ronald B. Franklin and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 909-914;
Fryklund, L.
- You have accessPHARMACOKINETICS AND METABOLISM OF TESAGLITAZAR, A NOVEL DUAL-ACTING PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST, AFTER A SINGLE ORAL AND INTRAVENOUS DOSE IN HUMANSH. Ericsson, B. Hamrén, S. Bergstrand, M. Elebring, L. Fryklund, M. Heijer and K. P. ÖhmanDrug Metabolism and Disposition September 2004, 32 (9) 923-929;
Fujita, Shoichi
- You have accessSTRAIN DIFFERENCES IN DIAZEPAM METABOLISM AT ITS THREE METABOLIC SITES IN SPRAGUE-DAWLEY, BROWN NORWAY, DARK AGOUTI, AND WISTAR STRAIN RATSKonomu Saito, Noriaki Sakai, Hyung-Sub Kim, Mayumi Ishizuka, Akio Kazusaka and Shoichi FujitaDrug Metabolism and Disposition September 2004, 32 (9) 959-965;
G
Ghanayem, Burhan I.
- You have accessBIOACTIVATION OF 1,1-DICHLOROETHYLENE TO ITS EPOXIDE BY CYP2E1 AND CYP2F ENZYMESAndrea C. Simmonds, Christopher A. Reilly, R. Michael Baldwin, Burhan I. Ghanayem, Diane L. Lanza, Garold S. Yost, Kathy S. Collins and Poh-Gek ForkertDrug Metabolism and Disposition September 2004, 32 (9) 1032-1039;
Goodwin, Lawrence A.
- You have accessSELECTIVE REDUCTION OF N-OXIDES TO AMINES: APPLICATION TO DRUG METABOLISMPalaniappan Kulanthaivel, Robert J. Barbuch, Rita S. Davidson, Ping Yi, Gregory A. Rener, Edward L. Mattiuz, Chad E. Hadden, Lawrence A. Goodwin and William J. EhlhardtDrug Metabolism and Disposition September 2004, 32 (9) 966-972;
H
Hadden, Chad E.
- You have accessSELECTIVE REDUCTION OF N-OXIDES TO AMINES: APPLICATION TO DRUG METABOLISMPalaniappan Kulanthaivel, Robert J. Barbuch, Rita S. Davidson, Ping Yi, Gregory A. Rener, Edward L. Mattiuz, Chad E. Hadden, Lawrence A. Goodwin and William J. EhlhardtDrug Metabolism and Disposition September 2004, 32 (9) 966-972;
Hamrén, B.
- You have accessPHARMACOKINETICS AND METABOLISM OF TESAGLITAZAR, A NOVEL DUAL-ACTING PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST, AFTER A SINGLE ORAL AND INTRAVENOUS DOSE IN HUMANSH. Ericsson, B. Hamrén, S. Bergstrand, M. Elebring, L. Fryklund, M. Heijer and K. P. ÖhmanDrug Metabolism and Disposition September 2004, 32 (9) 923-929;
Heijer, M.
- You have accessPHARMACOKINETICS AND METABOLISM OF TESAGLITAZAR, A NOVEL DUAL-ACTING PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST, AFTER A SINGLE ORAL AND INTRAVENOUS DOSE IN HUMANSH. Ericsson, B. Hamrén, S. Bergstrand, M. Elebring, L. Fryklund, M. Heijer and K. P. ÖhmanDrug Metabolism and Disposition September 2004, 32 (9) 923-929;
Hirono, Shuichi
- You have accessCARRIER-MEDIATED UPTAKE OF H2-RECEPTOR ANTAGONISTS BY THE RAT CHOROID PLEXUS: INVOLVEMENT OF RAT ORGANIC ANION TRANSPORTER 3Yoshinori Nagata, Hiroyuki Kusuhara, Shuichi Hirono, Hitoshi Endou and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 1040-1047;
Hop, Cornelis E.C.A.
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. I. ROLE OF CYTOCHROME P450, METHYLTRANSFERASES, FLAVIN MONOOXYGENASES, AND ESTERASESBindhu V. Karanam, Cornelis E.C.A. Hop, David Q. Liu, Mike Wallace, Dennis Dean, Hiroya Satoh, Masakatsu Komuro, Katsuya Awano and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 1015-1022; DOI: https://doi.org/10.1124/dmd.104.000034
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)-PHENYL] METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. II. IDENTIFICATION OF METABOLITES BY LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYDavid Q. Liu, Bindhu V. Karanam, George A. Doss, Rick R. Sidler, Stella H. Vincent and Cornelis E.C.A. HopDrug Metabolism and Disposition September 2004, 32 (9) 1023-1031; DOI: https://doi.org/10.1124/dmd.104.000059
Houston, J. Brian
- You have accessSUBSTRATE DEPLETION APPROACH FOR DETERMINING IN VITRO METABOLIC CLEARANCE: TIME DEPENDENCIES IN HEPATOCYTE AND MICROSOMAL INCUBATIONSHannah M. Jones and J. Brian HoustonDrug Metabolism and Disposition September 2004, 32 (9) 973-982; DOI: https://doi.org/10.1124/dmd.104.000125
I
Innocenti, Federico
- You have accessCYP2B6, CYP3A4, AND CYP2C19 ARE RESPONSIBLE FOR THE IN VITRO N-DEMETHYLATION OF MEPERIDINE IN HUMAN LIVER MICROSOMESJacqueline Ramírez, Federico Innocenti, Erin G. Schuetz, David A. Flockhart, Mary V. Relling, Raymond Santucci and Mark J. RatainDrug Metabolism and Disposition September 2004, 32 (9) 930-936;
Ishizuka, Mayumi
- You have accessSTRAIN DIFFERENCES IN DIAZEPAM METABOLISM AT ITS THREE METABOLIC SITES IN SPRAGUE-DAWLEY, BROWN NORWAY, DARK AGOUTI, AND WISTAR STRAIN RATSKonomu Saito, Noriaki Sakai, Hyung-Sub Kim, Mayumi Ishizuka, Akio Kazusaka and Shoichi FujitaDrug Metabolism and Disposition September 2004, 32 (9) 959-965;
J
Jinno, Hideto
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
Joglar, Jesús
- You have accessSTEREOCHEMICAL ANALYSIS OF 3,4-METHYLENEDIOXYMETHAMPHETAMINE AND ITS MAIN METABOLITES IN HUMAN SAMPLES INCLUDING THE CATECHOL-TYPE METABOLITE (3,4-DIHYDROXYMETHAMPHETAMINE)Nieves Pizarro, Magí Farré, Mitona Pujadas, Ana Ma͢ Peiró, Pere N Roset, Jesús Joglar and Rafael de la TorreDrug Metabolism and Disposition September 2004, 32 (9) 1001-1007;
Jones, Hannah M.
- You have accessSUBSTRATE DEPLETION APPROACH FOR DETERMINING IN VITRO METABOLIC CLEARANCE: TIME DEPENDENCIES IN HEPATOCYTE AND MICROSOMAL INCUBATIONSHannah M. Jones and J. Brian HoustonDrug Metabolism and Disposition September 2004, 32 (9) 973-982; DOI: https://doi.org/10.1124/dmd.104.000125
Jonker, Johan W.
- You have accessIMPAIRED RENAL EXCRETION OF 6-HYDROXY-5,7-DIMETHYL-2-METHYLAMINO-4-(3-PYRIDYLMETHYL) BENZOTHIAZOLE (E3040) SULFATE IN BREAST CANCER RESISTANCE PROTEIN (BCRP1/ABCG2) KNOCKOUT MICENaomi Mizuno, Michiko Suzuki, Hiroyuki Kusuhara, Hiroshi Suzuki, Kenji Takeuchi, Takuro Niwa, Johan W. Jonker and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 898-901;
K
Kalgutkar, Amit S.
- You have accessIDENTIFICATION OF AN N-METHYL-4-PHENYLPYRIDINIUM-LIKE METABOLITE OF THE ANTIDIARRHEAL AGENT LOPERAMIDE IN HUMAN LIVER MICROSOMES: UNDERLYING REASON(S) FOR THE LACK OF NEUROTOXICITY DESPITE THE BIOACTIVATION EVENTAmit S. Kalgutkar and Hang T. NguyenDrug Metabolism and Disposition September 2004, 32 (9) 943-952;
Kamakura, Shiro
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
Kamatani, Naoyuki
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
Karanam, Bindhu V.
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. I. ROLE OF CYTOCHROME P450, METHYLTRANSFERASES, FLAVIN MONOOXYGENASES, AND ESTERASESBindhu V. Karanam, Cornelis E.C.A. Hop, David Q. Liu, Mike Wallace, Dennis Dean, Hiroya Satoh, Masakatsu Komuro, Katsuya Awano and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 1015-1022; DOI: https://doi.org/10.1124/dmd.104.000034
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)-PHENYL] METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. II. IDENTIFICATION OF METABOLITES BY LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYDavid Q. Liu, Bindhu V. Karanam, George A. Doss, Rick R. Sidler, Stella H. Vincent and Cornelis E.C.A. HopDrug Metabolism and Disposition September 2004, 32 (9) 1023-1031; DOI: https://doi.org/10.1124/dmd.104.000059
Kazusaka, Akio
- You have accessSTRAIN DIFFERENCES IN DIAZEPAM METABOLISM AT ITS THREE METABOLIC SITES IN SPRAGUE-DAWLEY, BROWN NORWAY, DARK AGOUTI, AND WISTAR STRAIN RATSKonomu Saito, Noriaki Sakai, Hyung-Sub Kim, Mayumi Ishizuka, Akio Kazusaka and Shoichi FujitaDrug Metabolism and Disposition September 2004, 32 (9) 959-965;
Kim, Hyung-Sub
- You have accessSTRAIN DIFFERENCES IN DIAZEPAM METABOLISM AT ITS THREE METABOLIC SITES IN SPRAGUE-DAWLEY, BROWN NORWAY, DARK AGOUTI, AND WISTAR STRAIN RATSKonomu Saito, Noriaki Sakai, Hyung-Sub Kim, Mayumi Ishizuka, Akio Kazusaka and Shoichi FujitaDrug Metabolism and Disposition September 2004, 32 (9) 959-965;
Kim, Mi-Sook
- You have accessDIFFERENCES IN THE PHARMACOKINETICS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONISTS IN GENETICALLY OBESE ZUCKER AND SPRAGUE-DAWLEY RATS: IMPLICATIONS OF DECREASED GLUCURONIDATION IN OBESE ZUCKER RATSMi-Sook Kim, Sui Wang, Zhongzhou Shen, Christopher J. Kochansky, John R. Strauss, Ronald B. Franklin and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 909-914;
Kim, Sang Geon
- You have accessCERAMIDE, AN APOPTOTIC RHEOSTAT, INHIBITS CCAAT/ENHANCER BINDING PROTEIN-β AND NF-E2-RELATED FACTOR-2 ACTIVATION: THE ROLE IN GLUTATHIONE S-TRANSFERASE A2 GENE REPRESSIONI-Na Park, Il Je Cho and Sang Geon KimDrug Metabolism and Disposition September 2004, 32 (9) 893-897;
Kissel, Thomas
- You have accessEFFECT OF POLY(ETHYLENE IMINE) MOLECULAR WEIGHT AND PEGYLATION ON ORGAN DISTRIBUTION AND PHARMACOKINETICS OF POLYPLEXES WITH OLIGODEOXYNUCLEOTIDES IN MICEDagmar Fischer, Berit Osburg, Holger Petersen, Thomas Kissel and Ulrich BickelDrug Metabolism and Disposition September 2004, 32 (9) 983-992;
Kitakaze, Masafumi
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
Kochansky, Christopher J.
- You have accessDIFFERENCES IN THE PHARMACOKINETICS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONISTS IN GENETICALLY OBESE ZUCKER AND SPRAGUE-DAWLEY RATS: IMPLICATIONS OF DECREASED GLUCURONIDATION IN OBESE ZUCKER RATSMi-Sook Kim, Sui Wang, Zhongzhou Shen, Christopher J. Kochansky, John R. Strauss, Ronald B. Franklin and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 909-914;
Komamura, Kazuo
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
Komuro, Masakatsu
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. I. ROLE OF CYTOCHROME P450, METHYLTRANSFERASES, FLAVIN MONOOXYGENASES, AND ESTERASESBindhu V. Karanam, Cornelis E.C.A. Hop, David Q. Liu, Mike Wallace, Dennis Dean, Hiroya Satoh, Masakatsu Komuro, Katsuya Awano and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 1015-1022; DOI: https://doi.org/10.1124/dmd.104.000034
Kulanthaivel, Palaniappan
- You have accessSELECTIVE REDUCTION OF N-OXIDES TO AMINES: APPLICATION TO DRUG METABOLISMPalaniappan Kulanthaivel, Robert J. Barbuch, Rita S. Davidson, Ping Yi, Gregory A. Rener, Edward L. Mattiuz, Chad E. Hadden, Lawrence A. Goodwin and William J. EhlhardtDrug Metabolism and Disposition September 2004, 32 (9) 966-972;
Kusuhara, Hiroyuki
- You have accessCARRIER-MEDIATED UPTAKE OF H2-RECEPTOR ANTAGONISTS BY THE RAT CHOROID PLEXUS: INVOLVEMENT OF RAT ORGANIC ANION TRANSPORTER 3Yoshinori Nagata, Hiroyuki Kusuhara, Shuichi Hirono, Hitoshi Endou and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 1040-1047;
- You have accessIMPAIRED RENAL EXCRETION OF 6-HYDROXY-5,7-DIMETHYL-2-METHYLAMINO-4-(3-PYRIDYLMETHYL) BENZOTHIAZOLE (E3040) SULFATE IN BREAST CANCER RESISTANCE PROTEIN (BCRP1/ABCG2) KNOCKOUT MICENaomi Mizuno, Michiko Suzuki, Hiroyuki Kusuhara, Hiroshi Suzuki, Kenji Takeuchi, Takuro Niwa, Johan W. Jonker and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 898-901;
L
Lanza, Diane L.
- You have accessBIOACTIVATION OF 1,1-DICHLOROETHYLENE TO ITS EPOXIDE BY CYP2E1 AND CYP2F ENZYMESAndrea C. Simmonds, Christopher A. Reilly, R. Michael Baldwin, Burhan I. Ghanayem, Diane L. Lanza, Garold S. Yost, Kathy S. Collins and Poh-Gek ForkertDrug Metabolism and Disposition September 2004, 32 (9) 1032-1039;
Lau, Yau Yi
- You have accessEVALUATION OF A NOVEL IN VITRO CACO-2 HEPATOCYTE HYBRID SYSTEM FOR PREDICTING IN VIVO ORAL BIOAVAILABILITYYau Yi Lau, Yung-Hsiang Chen, Tong-tong Liu, Cheng Li, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition September 2004, 32 (9) 937-942;
Li, Cheng
- You have accessEVALUATION OF A NOVEL IN VITRO CACO-2 HEPATOCYTE HYBRID SYSTEM FOR PREDICTING IN VIVO ORAL BIOAVAILABILITYYau Yi Lau, Yung-Hsiang Chen, Tong-tong Liu, Cheng Li, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition September 2004, 32 (9) 937-942;
Liu, David Q.
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. I. ROLE OF CYTOCHROME P450, METHYLTRANSFERASES, FLAVIN MONOOXYGENASES, AND ESTERASESBindhu V. Karanam, Cornelis E.C.A. Hop, David Q. Liu, Mike Wallace, Dennis Dean, Hiroya Satoh, Masakatsu Komuro, Katsuya Awano and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 1015-1022; DOI: https://doi.org/10.1124/dmd.104.000034
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)-PHENYL] METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. II. IDENTIFICATION OF METABOLITES BY LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYDavid Q. Liu, Bindhu V. Karanam, George A. Doss, Rick R. Sidler, Stella H. Vincent and Cornelis E.C.A. HopDrug Metabolism and Disposition September 2004, 32 (9) 1023-1031; DOI: https://doi.org/10.1124/dmd.104.000059
Liu, Tong-tong
- You have accessEVALUATION OF A NOVEL IN VITRO CACO-2 HEPATOCYTE HYBRID SYSTEM FOR PREDICTING IN VIVO ORAL BIOAVAILABILITYYau Yi Lau, Yung-Hsiang Chen, Tong-tong Liu, Cheng Li, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition September 2004, 32 (9) 937-942;
M
Markowitz, John S.
- You have accessGREEN TEA (CAMELLIA SINENSIS) EXTRACT DOES NOT ALTER CYTOCHROME P450 3A4 OR 2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, Kenneth D. Chavin, C. Lindsay Devane, Robin M. Taylor, Jun-Sheng Wang, Ying Ruan and John S. MarkowitzDrug Metabolism and Disposition September 2004, 32 (9) 906-908; DOI: https://doi.org/10.1124/dmd.104.000083
Martin, Hans-Jörg
- You have accessENANTIOSELECTIVITY OF CARBONYL REDUCTION OF 4-METHYLNITROSAMINO-1-(3-PYRIDYL)-1-BUTANONE BY TISSUE FRACTIONS FROM HUMAN AND RAT AND BY ENZYMES ISOLATED FROM HUMAN LIVERUrsula Breyer-Pfaff, Hans-Jörg Martin, Michael Ernst and Edmund MaserDrug Metabolism and Disposition September 2004, 32 (9) 915-922;
Maser, Edmund
- You have accessENANTIOSELECTIVITY OF CARBONYL REDUCTION OF 4-METHYLNITROSAMINO-1-(3-PYRIDYL)-1-BUTANONE BY TISSUE FRACTIONS FROM HUMAN AND RAT AND BY ENZYMES ISOLATED FROM HUMAN LIVERUrsula Breyer-Pfaff, Hans-Jörg Martin, Michael Ernst and Edmund MaserDrug Metabolism and Disposition September 2004, 32 (9) 915-922;
Matheny, Christopher J.
- You have accessEFFECT OF PROTOTYPICAL INDUCING AGENTS ON P-GLYCOPROTEIN AND CYP3A EXPRESSION IN MOUSE TISSUESChristopher J. Matheny, Rabia Y. Ali, Xiaodong Yang and Gary M. PollackDrug Metabolism and Disposition September 2004, 32 (9) 1008-1014;
Mattiuz, Edward L.
- You have accessSELECTIVE REDUCTION OF N-OXIDES TO AMINES: APPLICATION TO DRUG METABOLISMPalaniappan Kulanthaivel, Robert J. Barbuch, Rita S. Davidson, Ping Yi, Gregory A. Rener, Edward L. Mattiuz, Chad E. Hadden, Lawrence A. Goodwin and William J. EhlhardtDrug Metabolism and Disposition September 2004, 32 (9) 966-972;
Mizuno, Naomi
- You have accessIMPAIRED RENAL EXCRETION OF 6-HYDROXY-5,7-DIMETHYL-2-METHYLAMINO-4-(3-PYRIDYLMETHYL) BENZOTHIAZOLE (E3040) SULFATE IN BREAST CANCER RESISTANCE PROTEIN (BCRP1/ABCG2) KNOCKOUT MICENaomi Mizuno, Michiko Suzuki, Hiroyuki Kusuhara, Hiroshi Suzuki, Kenji Takeuchi, Takuro Niwa, Johan W. Jonker and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 898-901;
N
Nagata, Yoshinori
- You have accessCARRIER-MEDIATED UPTAKE OF H2-RECEPTOR ANTAGONISTS BY THE RAT CHOROID PLEXUS: INVOLVEMENT OF RAT ORGANIC ANION TRANSPORTER 3Yoshinori Nagata, Hiroyuki Kusuhara, Shuichi Hirono, Hitoshi Endou and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 1040-1047;
Nguyen, Hang T.
- You have accessIDENTIFICATION OF AN N-METHYL-4-PHENYLPYRIDINIUM-LIKE METABOLITE OF THE ANTIDIARRHEAL AGENT LOPERAMIDE IN HUMAN LIVER MICROSOMES: UNDERLYING REASON(S) FOR THE LACK OF NEUROTOXICITY DESPITE THE BIOACTIVATION EVENTAmit S. Kalgutkar and Hang T. NguyenDrug Metabolism and Disposition September 2004, 32 (9) 943-952;
Niwa, Takuro
- You have accessIMPAIRED RENAL EXCRETION OF 6-HYDROXY-5,7-DIMETHYL-2-METHYLAMINO-4-(3-PYRIDYLMETHYL) BENZOTHIAZOLE (E3040) SULFATE IN BREAST CANCER RESISTANCE PROTEIN (BCRP1/ABCG2) KNOCKOUT MICENaomi Mizuno, Michiko Suzuki, Hiroyuki Kusuhara, Hiroshi Suzuki, Kenji Takeuchi, Takuro Niwa, Johan W. Jonker and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 898-901;
O
Öhman, K. P.
- You have accessPHARMACOKINETICS AND METABOLISM OF TESAGLITAZAR, A NOVEL DUAL-ACTING PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST, AFTER A SINGLE ORAL AND INTRAVENOUS DOSE IN HUMANSH. Ericsson, B. Hamrén, S. Bergstrand, M. Elebring, L. Fryklund, M. Heijer and K. P. ÖhmanDrug Metabolism and Disposition September 2004, 32 (9) 923-929;
Ohno, Akiko
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
Osburg, Berit
- You have accessEFFECT OF POLY(ETHYLENE IMINE) MOLECULAR WEIGHT AND PEGYLATION ON ORGAN DISTRIBUTION AND PHARMACOKINETICS OF POLYPLEXES WITH OLIGODEOXYNUCLEOTIDES IN MICEDagmar Fischer, Berit Osburg, Holger Petersen, Thomas Kissel and Ulrich BickelDrug Metabolism and Disposition September 2004, 32 (9) 983-992;
Ozawa, Shogo
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
P
Park, I-Na
- You have accessCERAMIDE, AN APOPTOTIC RHEOSTAT, INHIBITS CCAAT/ENHANCER BINDING PROTEIN-β AND NF-E2-RELATED FACTOR-2 ACTIVATION: THE ROLE IN GLUTATHIONE S-TRANSFERASE A2 GENE REPRESSIONI-Na Park, Il Je Cho and Sang Geon KimDrug Metabolism and Disposition September 2004, 32 (9) 893-897;
Peiró, Ana Ma͢
- You have accessSTEREOCHEMICAL ANALYSIS OF 3,4-METHYLENEDIOXYMETHAMPHETAMINE AND ITS MAIN METABOLITES IN HUMAN SAMPLES INCLUDING THE CATECHOL-TYPE METABOLITE (3,4-DIHYDROXYMETHAMPHETAMINE)Nieves Pizarro, Magí Farré, Mitona Pujadas, Ana Ma͢ Peiró, Pere N Roset, Jesús Joglar and Rafael de la TorreDrug Metabolism and Disposition September 2004, 32 (9) 1001-1007;
Petersen, Holger
- You have accessEFFECT OF POLY(ETHYLENE IMINE) MOLECULAR WEIGHT AND PEGYLATION ON ORGAN DISTRIBUTION AND PHARMACOKINETICS OF POLYPLEXES WITH OLIGODEOXYNUCLEOTIDES IN MICEDagmar Fischer, Berit Osburg, Holger Petersen, Thomas Kissel and Ulrich BickelDrug Metabolism and Disposition September 2004, 32 (9) 983-992;
Pizarro, Nieves
- You have accessSTEREOCHEMICAL ANALYSIS OF 3,4-METHYLENEDIOXYMETHAMPHETAMINE AND ITS MAIN METABOLITES IN HUMAN SAMPLES INCLUDING THE CATECHOL-TYPE METABOLITE (3,4-DIHYDROXYMETHAMPHETAMINE)Nieves Pizarro, Magí Farré, Mitona Pujadas, Ana Ma͢ Peiró, Pere N Roset, Jesús Joglar and Rafael de la TorreDrug Metabolism and Disposition September 2004, 32 (9) 1001-1007;
Pollack, Gary M.
- You have accessEFFECT OF PROTOTYPICAL INDUCING AGENTS ON P-GLYCOPROTEIN AND CYP3A EXPRESSION IN MOUSE TISSUESChristopher J. Matheny, Rabia Y. Ali, Xiaodong Yang and Gary M. PollackDrug Metabolism and Disposition September 2004, 32 (9) 1008-1014;
Pujadas, Mitona
- You have accessSTEREOCHEMICAL ANALYSIS OF 3,4-METHYLENEDIOXYMETHAMPHETAMINE AND ITS MAIN METABOLITES IN HUMAN SAMPLES INCLUDING THE CATECHOL-TYPE METABOLITE (3,4-DIHYDROXYMETHAMPHETAMINE)Nieves Pizarro, Magí Farré, Mitona Pujadas, Ana Ma͢ Peiró, Pere N Roset, Jesús Joglar and Rafael de la TorreDrug Metabolism and Disposition September 2004, 32 (9) 1001-1007;
R
Ramírez, Jacqueline
- You have accessCYP2B6, CYP3A4, AND CYP2C19 ARE RESPONSIBLE FOR THE IN VITRO N-DEMETHYLATION OF MEPERIDINE IN HUMAN LIVER MICROSOMESJacqueline Ramírez, Federico Innocenti, Erin G. Schuetz, David A. Flockhart, Mary V. Relling, Raymond Santucci and Mark J. RatainDrug Metabolism and Disposition September 2004, 32 (9) 930-936;
Ratain, Mark J.
- You have accessCYP2B6, CYP3A4, AND CYP2C19 ARE RESPONSIBLE FOR THE IN VITRO N-DEMETHYLATION OF MEPERIDINE IN HUMAN LIVER MICROSOMESJacqueline Ramírez, Federico Innocenti, Erin G. Schuetz, David A. Flockhart, Mary V. Relling, Raymond Santucci and Mark J. RatainDrug Metabolism and Disposition September 2004, 32 (9) 930-936;
Reilly, Christopher A.
- You have accessBIOACTIVATION OF 1,1-DICHLOROETHYLENE TO ITS EPOXIDE BY CYP2E1 AND CYP2F ENZYMESAndrea C. Simmonds, Christopher A. Reilly, R. Michael Baldwin, Burhan I. Ghanayem, Diane L. Lanza, Garold S. Yost, Kathy S. Collins and Poh-Gek ForkertDrug Metabolism and Disposition September 2004, 32 (9) 1032-1039;
Relling, Mary V.
- You have accessCYP2B6, CYP3A4, AND CYP2C19 ARE RESPONSIBLE FOR THE IN VITRO N-DEMETHYLATION OF MEPERIDINE IN HUMAN LIVER MICROSOMESJacqueline Ramírez, Federico Innocenti, Erin G. Schuetz, David A. Flockhart, Mary V. Relling, Raymond Santucci and Mark J. RatainDrug Metabolism and Disposition September 2004, 32 (9) 930-936;
Rener, Gregory A.
- You have accessSELECTIVE REDUCTION OF N-OXIDES TO AMINES: APPLICATION TO DRUG METABOLISMPalaniappan Kulanthaivel, Robert J. Barbuch, Rita S. Davidson, Ping Yi, Gregory A. Rener, Edward L. Mattiuz, Chad E. Hadden, Lawrence A. Goodwin and William J. EhlhardtDrug Metabolism and Disposition September 2004, 32 (9) 966-972;
Roerig, David L.
- You have accessKINETIC CHARACTERIZATION OF P-GLYCOPROTEIN-MEDIATED EFFLUX OF RHODAMINE 6G IN THE INTACT RABBIT LUNGDavid L. Roerig, Said H. Audi and Susan B. AhlfDrug Metabolism and Disposition September 2004, 32 (9) 953-958; DOI: https://doi.org/10.1124/dmd.104.000042
Roset, Pere N
- You have accessSTEREOCHEMICAL ANALYSIS OF 3,4-METHYLENEDIOXYMETHAMPHETAMINE AND ITS MAIN METABOLITES IN HUMAN SAMPLES INCLUDING THE CATECHOL-TYPE METABOLITE (3,4-DIHYDROXYMETHAMPHETAMINE)Nieves Pizarro, Magí Farré, Mitona Pujadas, Ana Ma͢ Peiró, Pere N Roset, Jesús Joglar and Rafael de la TorreDrug Metabolism and Disposition September 2004, 32 (9) 1001-1007;
Ruan, Ying
- You have accessGREEN TEA (CAMELLIA SINENSIS) EXTRACT DOES NOT ALTER CYTOCHROME P450 3A4 OR 2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, Kenneth D. Chavin, C. Lindsay Devane, Robin M. Taylor, Jun-Sheng Wang, Ying Ruan and John S. MarkowitzDrug Metabolism and Disposition September 2004, 32 (9) 906-908; DOI: https://doi.org/10.1124/dmd.104.000083
S
Saeki, Mayumi
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
Saito, Konomu
- You have accessSTRAIN DIFFERENCES IN DIAZEPAM METABOLISM AT ITS THREE METABOLIC SITES IN SPRAGUE-DAWLEY, BROWN NORWAY, DARK AGOUTI, AND WISTAR STRAIN RATSKonomu Saito, Noriaki Sakai, Hyung-Sub Kim, Mayumi Ishizuka, Akio Kazusaka and Shoichi FujitaDrug Metabolism and Disposition September 2004, 32 (9) 959-965;
Saito, Yoshiro
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
Sakai, Noriaki
- You have accessSTRAIN DIFFERENCES IN DIAZEPAM METABOLISM AT ITS THREE METABOLIC SITES IN SPRAGUE-DAWLEY, BROWN NORWAY, DARK AGOUTI, AND WISTAR STRAIN RATSKonomu Saito, Noriaki Sakai, Hyung-Sub Kim, Mayumi Ishizuka, Akio Kazusaka and Shoichi FujitaDrug Metabolism and Disposition September 2004, 32 (9) 959-965;
Santucci, Raymond
- You have accessCYP2B6, CYP3A4, AND CYP2C19 ARE RESPONSIBLE FOR THE IN VITRO N-DEMETHYLATION OF MEPERIDINE IN HUMAN LIVER MICROSOMESJacqueline Ramírez, Federico Innocenti, Erin G. Schuetz, David A. Flockhart, Mary V. Relling, Raymond Santucci and Mark J. RatainDrug Metabolism and Disposition September 2004, 32 (9) 930-936;
Satoh, Hiroya
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. I. ROLE OF CYTOCHROME P450, METHYLTRANSFERASES, FLAVIN MONOOXYGENASES, AND ESTERASESBindhu V. Karanam, Cornelis E.C.A. Hop, David Q. Liu, Mike Wallace, Dennis Dean, Hiroya Satoh, Masakatsu Komuro, Katsuya Awano and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 1015-1022; DOI: https://doi.org/10.1124/dmd.104.000034
Sawada, Jun-ichi
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
Schuetz, Erin G.
- You have accessCYP2B6, CYP3A4, AND CYP2C19 ARE RESPONSIBLE FOR THE IN VITRO N-DEMETHYLATION OF MEPERIDINE IN HUMAN LIVER MICROSOMESJacqueline Ramírez, Federico Innocenti, Erin G. Schuetz, David A. Flockhart, Mary V. Relling, Raymond Santucci and Mark J. RatainDrug Metabolism and Disposition September 2004, 32 (9) 930-936;
Shen, Zhongzhou
- You have accessDIFFERENCES IN THE PHARMACOKINETICS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONISTS IN GENETICALLY OBESE ZUCKER AND SPRAGUE-DAWLEY RATS: IMPLICATIONS OF DECREASED GLUCURONIDATION IN OBESE ZUCKER RATSMi-Sook Kim, Sui Wang, Zhongzhou Shen, Christopher J. Kochansky, John R. Strauss, Ronald B. Franklin and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 909-914;
Sidler, Rick R.
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)-PHENYL] METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. II. IDENTIFICATION OF METABOLITES BY LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYDavid Q. Liu, Bindhu V. Karanam, George A. Doss, Rick R. Sidler, Stella H. Vincent and Cornelis E.C.A. HopDrug Metabolism and Disposition September 2004, 32 (9) 1023-1031; DOI: https://doi.org/10.1124/dmd.104.000059
Simmonds, Andrea C.
- You have accessBIOACTIVATION OF 1,1-DICHLOROETHYLENE TO ITS EPOXIDE BY CYP2E1 AND CYP2F ENZYMESAndrea C. Simmonds, Christopher A. Reilly, R. Michael Baldwin, Burhan I. Ghanayem, Diane L. Lanza, Garold S. Yost, Kathy S. Collins and Poh-Gek ForkertDrug Metabolism and Disposition September 2004, 32 (9) 1032-1039;
Smith, Philip C.
- You have accessALTERED PHARMACOKINETICS OF OMEPRAZOLE IN CYSTIC FIBROSIS KNOCKOUT MICE RELATIVE TO WILD-TYPE MICEMelanie N. Tallman, Shazia Y. Ali and Philip C. SmithDrug Metabolism and Disposition September 2004, 32 (9) 902-905;
Strauss, John R.
- You have accessDIFFERENCES IN THE PHARMACOKINETICS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONISTS IN GENETICALLY OBESE ZUCKER AND SPRAGUE-DAWLEY RATS: IMPLICATIONS OF DECREASED GLUCURONIDATION IN OBESE ZUCKER RATSMi-Sook Kim, Sui Wang, Zhongzhou Shen, Christopher J. Kochansky, John R. Strauss, Ronald B. Franklin and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 909-914;
Sugiyama, Yuichi
- You have accessCARRIER-MEDIATED UPTAKE OF H2-RECEPTOR ANTAGONISTS BY THE RAT CHOROID PLEXUS: INVOLVEMENT OF RAT ORGANIC ANION TRANSPORTER 3Yoshinori Nagata, Hiroyuki Kusuhara, Shuichi Hirono, Hitoshi Endou and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 1040-1047;
- You have accessIMPAIRED RENAL EXCRETION OF 6-HYDROXY-5,7-DIMETHYL-2-METHYLAMINO-4-(3-PYRIDYLMETHYL) BENZOTHIAZOLE (E3040) SULFATE IN BREAST CANCER RESISTANCE PROTEIN (BCRP1/ABCG2) KNOCKOUT MICENaomi Mizuno, Michiko Suzuki, Hiroyuki Kusuhara, Hiroshi Suzuki, Kenji Takeuchi, Takuro Niwa, Johan W. Jonker and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 898-901;
Suzuki, Hiroshi
- You have accessIMPAIRED RENAL EXCRETION OF 6-HYDROXY-5,7-DIMETHYL-2-METHYLAMINO-4-(3-PYRIDYLMETHYL) BENZOTHIAZOLE (E3040) SULFATE IN BREAST CANCER RESISTANCE PROTEIN (BCRP1/ABCG2) KNOCKOUT MICENaomi Mizuno, Michiko Suzuki, Hiroyuki Kusuhara, Hiroshi Suzuki, Kenji Takeuchi, Takuro Niwa, Johan W. Jonker and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 898-901;
Suzuki, Michiko
- You have accessIMPAIRED RENAL EXCRETION OF 6-HYDROXY-5,7-DIMETHYL-2-METHYLAMINO-4-(3-PYRIDYLMETHYL) BENZOTHIAZOLE (E3040) SULFATE IN BREAST CANCER RESISTANCE PROTEIN (BCRP1/ABCG2) KNOCKOUT MICENaomi Mizuno, Michiko Suzuki, Hiroyuki Kusuhara, Hiroshi Suzuki, Kenji Takeuchi, Takuro Niwa, Johan W. Jonker and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 898-901;
T
Takeuchi, Kenji
- You have accessIMPAIRED RENAL EXCRETION OF 6-HYDROXY-5,7-DIMETHYL-2-METHYLAMINO-4-(3-PYRIDYLMETHYL) BENZOTHIAZOLE (E3040) SULFATE IN BREAST CANCER RESISTANCE PROTEIN (BCRP1/ABCG2) KNOCKOUT MICENaomi Mizuno, Michiko Suzuki, Hiroyuki Kusuhara, Hiroshi Suzuki, Kenji Takeuchi, Takuro Niwa, Johan W. Jonker and Yuichi SugiyamaDrug Metabolism and Disposition September 2004, 32 (9) 898-901;
Tallman, Melanie N.
- You have accessALTERED PHARMACOKINETICS OF OMEPRAZOLE IN CYSTIC FIBROSIS KNOCKOUT MICE RELATIVE TO WILD-TYPE MICEMelanie N. Tallman, Shazia Y. Ali and Philip C. SmithDrug Metabolism and Disposition September 2004, 32 (9) 902-905;
Tanaka-Kagawa, Toshiko
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
Taylor, Robin M.
- You have accessGREEN TEA (CAMELLIA SINENSIS) EXTRACT DOES NOT ALTER CYTOCHROME P450 3A4 OR 2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, Kenneth D. Chavin, C. Lindsay Devane, Robin M. Taylor, Jun-Sheng Wang, Ying Ruan and John S. MarkowitzDrug Metabolism and Disposition September 2004, 32 (9) 906-908; DOI: https://doi.org/10.1124/dmd.104.000083
U
Ueno, Kazuyuki
- You have accessSINGLE NUCLEOTIDE POLYMORPHISMS AND HAPLOTYPE FREQUENCIES OF UGT2B4 AND UGT2B7 IN A JAPANESE POPULATIONMayumi Saeki, Yoshiro Saito, Hideto Jinno, Toshiko Tanaka-Kagawa, Akiko Ohno, Shogo Ozawa, Kazuyuki Ueno, Shiro Kamakura, Naoyuki Kamatani, Kazuo Komamura, Masafumi Kitakaze and Jun-ichi SawadaDrug Metabolism and Disposition September 2004, 32 (9) 1048-1054;
V
Vincent, Stella H.
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. I. ROLE OF CYTOCHROME P450, METHYLTRANSFERASES, FLAVIN MONOOXYGENASES, AND ESTERASESBindhu V. Karanam, Cornelis E.C.A. Hop, David Q. Liu, Mike Wallace, Dennis Dean, Hiroya Satoh, Masakatsu Komuro, Katsuya Awano and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 1015-1022; DOI: https://doi.org/10.1124/dmd.104.000034
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL)-PHENYL] METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. II. IDENTIFICATION OF METABOLITES BY LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYDavid Q. Liu, Bindhu V. Karanam, George A. Doss, Rick R. Sidler, Stella H. Vincent and Cornelis E.C.A. HopDrug Metabolism and Disposition September 2004, 32 (9) 1023-1031; DOI: https://doi.org/10.1124/dmd.104.000059
- You have accessDIFFERENCES IN THE PHARMACOKINETICS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONISTS IN GENETICALLY OBESE ZUCKER AND SPRAGUE-DAWLEY RATS: IMPLICATIONS OF DECREASED GLUCURONIDATION IN OBESE ZUCKER RATSMi-Sook Kim, Sui Wang, Zhongzhou Shen, Christopher J. Kochansky, John R. Strauss, Ronald B. Franklin and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 909-914;
W
Wallace, Mike
- You have accessIN VITRO METABOLISM OF MK-0767 [(±)-5-[(2,4-DIOXOTHIAZOLIDIN-5-YL)METHYL]-2-METHOXY-N-[[(4-TRIFLUOROMETHYL) PHENYL]METHYL]BENZAMIDE], A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR α/γ AGONIST. I. ROLE OF CYTOCHROME P450, METHYLTRANSFERASES, FLAVIN MONOOXYGENASES, AND ESTERASESBindhu V. Karanam, Cornelis E.C.A. Hop, David Q. Liu, Mike Wallace, Dennis Dean, Hiroya Satoh, Masakatsu Komuro, Katsuya Awano and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 1015-1022; DOI: https://doi.org/10.1124/dmd.104.000034
Wang, Jun-Sheng
- You have accessGREEN TEA (CAMELLIA SINENSIS) EXTRACT DOES NOT ALTER CYTOCHROME P450 3A4 OR 2D6 ACTIVITY IN HEALTHY VOLUNTEERSJennifer L. Donovan, Kenneth D. Chavin, C. Lindsay Devane, Robin M. Taylor, Jun-Sheng Wang, Ying Ruan and John S. MarkowitzDrug Metabolism and Disposition September 2004, 32 (9) 906-908; DOI: https://doi.org/10.1124/dmd.104.000083
Wang, Sui
- You have accessDIFFERENCES IN THE PHARMACOKINETICS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONISTS IN GENETICALLY OBESE ZUCKER AND SPRAGUE-DAWLEY RATS: IMPLICATIONS OF DECREASED GLUCURONIDATION IN OBESE ZUCKER RATSMi-Sook Kim, Sui Wang, Zhongzhou Shen, Christopher J. Kochansky, John R. Strauss, Ronald B. Franklin and Stella H. VincentDrug Metabolism and Disposition September 2004, 32 (9) 909-914;
White, Ronald E.
- You have accessEVALUATION OF A NOVEL IN VITRO CACO-2 HEPATOCYTE HYBRID SYSTEM FOR PREDICTING IN VIVO ORAL BIOAVAILABILITYYau Yi Lau, Yung-Hsiang Chen, Tong-tong Liu, Cheng Li, Xiaoming Cui, Ronald E. White and K.-C. ChengDrug Metabolism and Disposition September 2004, 32 (9) 937-942;
Y
Yang, Xiaodong
- You have accessEFFECT OF PROTOTYPICAL INDUCING AGENTS ON P-GLYCOPROTEIN AND CYP3A EXPRESSION IN MOUSE TISSUESChristopher J. Matheny, Rabia Y. Ali, Xiaodong Yang and Gary M. PollackDrug Metabolism and Disposition September 2004, 32 (9) 1008-1014;
Yi, Ping
- You have accessSELECTIVE REDUCTION OF N-OXIDES TO AMINES: APPLICATION TO DRUG METABOLISMPalaniappan Kulanthaivel, Robert J. Barbuch, Rita S. Davidson, Ping Yi, Gregory A. Rener, Edward L. Mattiuz, Chad E. Hadden, Lawrence A. Goodwin and William J. EhlhardtDrug Metabolism and Disposition September 2004, 32 (9) 966-972;
Yost, Garold S.
- You have accessBIOACTIVATION OF 1,1-DICHLOROETHYLENE TO ITS EPOXIDE BY CYP2E1 AND CYP2F ENZYMESAndrea C. Simmonds, Christopher A. Reilly, R. Michael Baldwin, Burhan I. Ghanayem, Diane L. Lanza, Garold S. Yost, Kathy S. Collins and Poh-Gek ForkertDrug Metabolism and Disposition September 2004, 32 (9) 1032-1039;
Z
Zheng, Naiyu
- You have accessKINETICS AND REGULATION OF CYTOCHROME P450-MEDIATED ETOPOSIDE METABOLISMXiaoliang Zhuo, Naiyu Zheng, Carolyn A. Felix and Ian A. BlairDrug Metabolism and Disposition September 2004, 32 (9) 993-1000;
Zhuo, Xiaoliang
- You have accessKINETICS AND REGULATION OF CYTOCHROME P450-MEDIATED ETOPOSIDE METABOLISMXiaoliang Zhuo, Naiyu Zheng, Carolyn A. Felix and Ian A. BlairDrug Metabolism and Disposition September 2004, 32 (9) 993-1000;