Index by author
October 01, 2005; Volume 33,Issue 10
A
Abdulla, Dalya
- You have accessTHE SIGNAL TRANSDUCTION PATHWAYS INVOLVED IN HEPATIC CYTOCHROME P450 REGULATION IN THE RAT DURING A LIPOPOLYSACCHARIDE-INDUCED MODEL OF CENTRAL NERVOUS SYSTEM INFLAMMATIONDalya Abdulla, Kerry B. Goralski, Elena Garcia Del Busto Cano and Kenneth W. RentonDrug Metabolism and Disposition October 2005, 33 (10) 1521-1531; DOI: https://doi.org/10.1124/dmd.105.004564
Ali, Shazia
- You have accessAN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITYKristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. RitterDrug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663
B
Baldwin, R. Michael
- You have accessPULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. CollinsDrug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
Ben-Am, Monique
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
Bertrand, Marc
- You have accessFUNCTIONAL EXPRESSION OF SINUSOIDAL DRUG TRANSPORTERS IN PRIMARY HUMAN AND RAT HEPATOCYTESEmilie Jigorel, Marc Le Vee, Claire Boursier-Neyret, Marc Bertrand and Olivier FardelDrug Metabolism and Disposition October 2005, 33 (10) 1418-1422; DOI: https://doi.org/10.1124/dmd.105.004762
Bialer, Meir
- You have accessPHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATSEyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir BialerDrug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
Black, Sherry R.
- You have accessPHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITROJames M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. BurkaDrug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
Boursier-Neyret, Claire
- You have accessFUNCTIONAL EXPRESSION OF SINUSOIDAL DRUG TRANSPORTERS IN PRIMARY HUMAN AND RAT HEPATOCYTESEmilie Jigorel, Marc Le Vee, Claire Boursier-Neyret, Marc Bertrand and Olivier FardelDrug Metabolism and Disposition October 2005, 33 (10) 1418-1422; DOI: https://doi.org/10.1124/dmd.105.004762
Britzi, Malka
- You have accessPHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATSEyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir BialerDrug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
Bu, Hai-Zhi
- You have accessA SIMPLE SEQUENTIAL INCUBATION METHOD FOR DECONVOLUTING THE COMPLICATED SEQUENTIAL METABOLISM OF CAPRAVIRINE IN HUMANSHai-Zhi Bu, Ping Kang, Ping Zhao, William F. Pool and Ellen Y. WuDrug Metabolism and Disposition October 2005, 33 (10) 1438-1445; DOI: https://doi.org/10.1124/dmd.105.005413
Burka, Leo T.
- You have accessPHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITROJames M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. BurkaDrug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
C
Chen, Ying
- You have accessEXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSAXiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin DingDrug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
Cheung, Connie
- You have accessHUMAN CYP2D6 AND MOUSE CYP2DS: ORGAN DISTRIBUTION IN A HUMANIZED MOUSE MODELSharon L. Miksys, Connie Cheung, Frank J. Gonzalez and Rachel F. TyndaleDrug Metabolism and Disposition October 2005, 33 (10) 1495-1502; DOI: https://doi.org/10.1124/dmd.105.005488
Churchwell, Mona I.
- You have accessMETABOLISM OF PIGMENT YELLOW 74 BY RAT AND HUMAN MICROSOMAL PROTEINSYanyan Cui, Mona I. Churchwell, Letha H. Couch, Daniel R. Doerge and Paul C. HowardDrug Metabolism and Disposition October 2005, 33 (10) 1459-1465; DOI: https://doi.org/10.1124/dmd.104.003285
Clement, Bernd
- You have accessMETABOLISM OF N-HYDROXYGUANIDINES (N-HYDROXYDEBRISOQUINE) IN HUMAN AND PORCINE HEPATOCYTES: REDUCTION AND FORMATION OF GLUCURONIDESAnja Kristina Froehlich, Ulrich Girreser and Bernd ClementDrug Metabolism and Disposition October 2005, 33 (10) 1532-1537; DOI: https://doi.org/10.1124/dmd.105.004572
Coleman, Donna P.
- You have accessPHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITROJames M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. BurkaDrug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
Collins, Kathy S.
- You have accessPULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. CollinsDrug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
Couch, Letha H.
- You have accessMETABOLISM OF PIGMENT YELLOW 74 BY RAT AND HUMAN MICROSOMAL PROTEINSYanyan Cui, Mona I. Churchwell, Letha H. Couch, Daniel R. Doerge and Paul C. HowardDrug Metabolism and Disposition October 2005, 33 (10) 1459-1465; DOI: https://doi.org/10.1124/dmd.104.003285
Cui, Yanyan
- You have accessMETABOLISM OF PIGMENT YELLOW 74 BY RAT AND HUMAN MICROSOMAL PROTEINSYanyan Cui, Mona I. Churchwell, Letha H. Couch, Daniel R. Doerge and Paul C. HowardDrug Metabolism and Disposition October 2005, 33 (10) 1459-1465; DOI: https://doi.org/10.1124/dmd.104.003285
Cummings, Meredith E.
- You have accessGLUTATHIONE TRAPPING TO MEASURE MICROSOMAL OXIDATION OF FURAN TO CIS-2-BUTENE-1,4-DIALLisa A. Peterson, Meredith E. Cummings, Choua C. Vu and Brock A. MatterDrug Metabolism and Disposition October 2005, 33 (10) 1453-1458; DOI: https://doi.org/10.1124/dmd.105.004432
D
Daidoji, Tomo
- You have accessUDP-GLUCURONOSYLTRANSFERASE ISOFORMS CATALYZING GLUCURONIDATION OF HYDROXY-POLYCHLORINATED BIPHENYLS IN RATTomo Daidoji, Keisuke Gozu, Hidetomo Iwano, Hiroki Inoue and Hiroshi YokotaDrug Metabolism and Disposition October 2005, 33 (10) 1466-1476; DOI: https://doi.org/10.1124/dmd.105.004416
Del Busto Cano, Elena Garcia
- You have accessTHE SIGNAL TRANSDUCTION PATHWAYS INVOLVED IN HEPATIC CYTOCHROME P450 REGULATION IN THE RAT DURING A LIPOPOLYSACCHARIDE-INDUCED MODEL OF CENTRAL NERVOUS SYSTEM INFLAMMATIONDalya Abdulla, Kerry B. Goralski, Elena Garcia Del Busto Cano and Kenneth W. RentonDrug Metabolism and Disposition October 2005, 33 (10) 1521-1531; DOI: https://doi.org/10.1124/dmd.105.004564
Ding, Xinxin
- You have accessEXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSAXiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin DingDrug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
Doerge, Daniel R.
- You have accessMETABOLISM OF PIGMENT YELLOW 74 BY RAT AND HUMAN MICROSOMAL PROTEINSYanyan Cui, Mona I. Churchwell, Letha H. Couch, Daniel R. Doerge and Paul C. HowardDrug Metabolism and Disposition October 2005, 33 (10) 1459-1465; DOI: https://doi.org/10.1124/dmd.104.003285
E
Etheridge, Amy S.
- You have accessPHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITROJames M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. BurkaDrug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
F
Fardel, Olivier
- You have accessFUNCTIONAL EXPRESSION OF SINUSOIDAL DRUG TRANSPORTERS IN PRIMARY HUMAN AND RAT HEPATOCYTESEmilie Jigorel, Marc Le Vee, Claire Boursier-Neyret, Marc Bertrand and Olivier FardelDrug Metabolism and Disposition October 2005, 33 (10) 1418-1422; DOI: https://doi.org/10.1124/dmd.105.004762
Forkert, Poh-Gek
- You have accessPULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. CollinsDrug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
Froehlich, Anja Kristina
- You have accessMETABOLISM OF N-HYDROXYGUANIDINES (N-HYDROXYDEBRISOQUINE) IN HUMAN AND PORCINE HEPATOCYTES: REDUCTION AND FORMATION OF GLUCURONIDESAnja Kristina Froehlich, Ulrich Girreser and Bernd ClementDrug Metabolism and Disposition October 2005, 33 (10) 1532-1537; DOI: https://doi.org/10.1124/dmd.105.004572
Fuse, Kaori
- You have accessCONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANSMaki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622
G
Gibson, Dan
- You have accessPHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATSEyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir BialerDrug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
Girreser, Ulrich
- You have accessMETABOLISM OF N-HYDROXYGUANIDINES (N-HYDROXYDEBRISOQUINE) IN HUMAN AND PORCINE HEPATOCYTES: REDUCTION AND FORMATION OF GLUCURONIDESAnja Kristina Froehlich, Ulrich Girreser and Bernd ClementDrug Metabolism and Disposition October 2005, 33 (10) 1532-1537; DOI: https://doi.org/10.1124/dmd.105.004572
Gonzalez, Frank J.
- You have accessHUMAN CYP2D6 AND MOUSE CYP2DS: ORGAN DISTRIBUTION IN A HUMANIZED MOUSE MODELSharon L. Miksys, Connie Cheung, Frank J. Gonzalez and Rachel F. TyndaleDrug Metabolism and Disposition October 2005, 33 (10) 1495-1502; DOI: https://doi.org/10.1124/dmd.105.005488
Goralski, Kerry B.
- You have accessTHE SIGNAL TRANSDUCTION PATHWAYS INVOLVED IN HEPATIC CYTOCHROME P450 REGULATION IN THE RAT DURING A LIPOPOLYSACCHARIDE-INDUCED MODEL OF CENTRAL NERVOUS SYSTEM INFLAMMATIONDalya Abdulla, Kerry B. Goralski, Elena Garcia Del Busto Cano and Kenneth W. RentonDrug Metabolism and Disposition October 2005, 33 (10) 1521-1531; DOI: https://doi.org/10.1124/dmd.105.004564
Gozu, Keisuke
- You have accessUDP-GLUCURONOSYLTRANSFERASE ISOFORMS CATALYZING GLUCURONIDATION OF HYDROXY-POLYCHLORINATED BIPHENYLS IN RATTomo Daidoji, Keisuke Gozu, Hidetomo Iwano, Hiroki Inoue and Hiroshi YokotaDrug Metabolism and Disposition October 2005, 33 (10) 1466-1476; DOI: https://doi.org/10.1124/dmd.105.004416
Gross, Gerhard
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
Gschwind, Hans-Peter
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
Gu, Jun
- You have accessEXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSAXiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin DingDrug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
H
Hayes, Michael
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
Hoskins, Janelle M.
- You have accessCOMMENT ON “A FRAMESHIFT MUTATION AND ALTERNATE SPLICING IN HUMAN BRAIN GENERATE A FUNCTIONAL FORM OF THE PSEUDOGENE CYTOCHROME P4502D7 THAT DEMETHYLATES CODEINE TO MORPHINE”Janelle M. Hoskins, Sharon Marsh and Howard L. McLeodDrug Metabolism and Disposition October 2005, 33 (10) 1564-1565; DOI: https://doi.org/10.1124/dmd.105.005736
Howard, Paul C.
- You have accessMETABOLISM OF PIGMENT YELLOW 74 BY RAT AND HUMAN MICROSOMAL PROTEINSYanyan Cui, Mona I. Churchwell, Letha H. Couch, Daniel R. Doerge and Paul C. HowardDrug Metabolism and Disposition October 2005, 33 (10) 1459-1465; DOI: https://doi.org/10.1124/dmd.104.003285
I
Inoue, Hiroki
- You have accessUDP-GLUCURONOSYLTRANSFERASE ISOFORMS CATALYZING GLUCURONIDATION OF HYDROXY-POLYCHLORINATED BIPHENYLS IN RATTomo Daidoji, Keisuke Gozu, Hidetomo Iwano, Hiroki Inoue and Hiroshi YokotaDrug Metabolism and Disposition October 2005, 33 (10) 1466-1476; DOI: https://doi.org/10.1124/dmd.105.004416
Iwano, Hidetomo
- You have accessUDP-GLUCURONOSYLTRANSFERASE ISOFORMS CATALYZING GLUCURONIDATION OF HYDROXY-POLYCHLORINATED BIPHENYLS IN RATTomo Daidoji, Keisuke Gozu, Hidetomo Iwano, Hiroki Inoue and Hiroshi YokotaDrug Metabolism and Disposition October 2005, 33 (10) 1466-1476; DOI: https://doi.org/10.1124/dmd.105.004416
J
Jigorel, Emilie
- You have accessFUNCTIONAL EXPRESSION OF SINUSOIDAL DRUG TRANSPORTERS IN PRIMARY HUMAN AND RAT HEPATOCYTESEmilie Jigorel, Marc Le Vee, Claire Boursier-Neyret, Marc Bertrand and Olivier FardelDrug Metabolism and Disposition October 2005, 33 (10) 1418-1422; DOI: https://doi.org/10.1124/dmd.105.004762
K
Kang, Ping
- You have accessA SIMPLE SEQUENTIAL INCUBATION METHOD FOR DECONVOLUTING THE COMPLICATED SEQUENTIAL METABOLISM OF CAPRAVIRINE IN HUMANSHai-Zhi Bu, Ping Kang, Ping Zhao, William F. Pool and Ellen Y. WuDrug Metabolism and Disposition October 2005, 33 (10) 1438-1445; DOI: https://doi.org/10.1124/dmd.105.005413
Kessler, Fay K.
- You have accessAN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITYKristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. RitterDrug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663
Kim, Su-Ryang
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Kogetsu, Hirokuni
- You have accessPHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATSRisa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
Kubo, Takashi
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Kumagai, Yoichi
- You have accessPHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATSRisa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
Kupfer, David
- You have accessOXIDATION OF TAMOXIFEN BY HUMAN FLAVIN-CONTAINING MONOOXYGENASE (FMO) 1 AND FMO3 TO TAMOXIFEN-N-OXIDE AND ITS NOVEL REDUCTION BACK TO TAMOXIFEN BY HUMAN CYTOCHROMES P450 AND HEMOGLOBINPriyanka Parte and David KupferDrug Metabolism and Disposition October 2005, 33 (10) 1446-1452; DOI: https://doi.org/10.1124/dmd.104.000802
Kusuhara, Hiroyuki
- You have accessCONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANSMaki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622
L
Lash, Lawrence H.
- You have accessPULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. CollinsDrug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
Le Vee, Marc
- You have accessFUNCTIONAL EXPRESSION OF SINUSOIDAL DRUG TRANSPORTERS IN PRIMARY HUMAN AND RAT HEPATOCYTESEmilie Jigorel, Marc Le Vee, Claire Boursier-Neyret, Marc Bertrand and Olivier FardelDrug Metabolism and Disposition October 2005, 33 (10) 1418-1422; DOI: https://doi.org/10.1124/dmd.105.004762
Ling, Guoyu
- You have accessEXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSAXiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin DingDrug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
Liu, Dazhi
- You have accessEXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSAXiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin DingDrug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
M
Maeda, Kazuya
- You have accessCONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANSMaki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622
Marsh, Sharon
- You have accessCOMMENT ON “A FRAMESHIFT MUTATION AND ALTERNATE SPLICING IN HUMAN BRAIN GENERATE A FUNCTIONAL FORM OF THE PSEUDOGENE CYTOCHROME P4502D7 THAT DEMETHYLATES CODEINE TO MORPHINE”Janelle M. Hoskins, Sharon Marsh and Howard L. McLeodDrug Metabolism and Disposition October 2005, 33 (10) 1564-1565; DOI: https://doi.org/10.1124/dmd.105.005736
Mathews, James M.
- You have accessPHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITROJames M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. BurkaDrug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
Matsumoto, Kenji
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Matter, Brock A.
- You have accessGLUTATHIONE TRAPPING TO MEASURE MICROSOMAL OXIDATION OF FURAN TO CIS-2-BUTENE-1,4-DIALLisa A. Peterson, Meredith E. Cummings, Choua C. Vu and Brock A. MatterDrug Metabolism and Disposition October 2005, 33 (10) 1453-1458; DOI: https://doi.org/10.1124/dmd.105.004432
McLeod, Howard L.
- You have accessCOMMENT ON “A FRAMESHIFT MUTATION AND ALTERNATE SPLICING IN HUMAN BRAIN GENERATE A FUNCTIONAL FORM OF THE PSEUDOGENE CYTOCHROME P4502D7 THAT DEMETHYLATES CODEINE TO MORPHINE”Janelle M. Hoskins, Sharon Marsh and Howard L. McLeodDrug Metabolism and Disposition October 2005, 33 (10) 1564-1565; DOI: https://doi.org/10.1124/dmd.105.005736
Miksys, Sharon L.
- You have accessHUMAN CYP2D6 AND MOUSE CYP2DS: ORGAN DISTRIBUTION IN A HUMANIZED MOUSE MODELSharon L. Miksys, Connie Cheung, Frank J. Gonzalez and Rachel F. TyndaleDrug Metabolism and Disposition October 2005, 33 (10) 1495-1502; DOI: https://doi.org/10.1124/dmd.105.005488
Miles, Kristini K.
- You have accessAN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITYKristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. RitterDrug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663
Millen, Brandie
- You have accessPULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. CollinsDrug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
Minami, Hironobu
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
N
Nakajima, Toshiharu
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Nasu, Risa
- You have accessPHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATSRisa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
Nishigaki, Ryuichiro
- You have accessCONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANSMaki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622
O
Obach, R. Scott
- You have accessSEEING THROUGH THE MIST: ABUNDANCE VERSUS PERCENTAGE. COMMENTARY ON METABOLITES IN SAFETY TESTINGDennis A. Smith and R. Scott ObachDrug Metabolism and Disposition October 2005, 33 (10) 1409-1417; DOI: https://doi.org/10.1124/dmd.105.005041
Ohno, Yasuo
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Ohtani, Hisakazu
- You have accessPHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATSRisa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
Ohtsu, Atsushi
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Okudaira, Kazuho
- You have accessCONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANSMaki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622
Ozawa, Shogo
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
P
Pai, Harish V.
- You have accessRESPONSE TO COMMENT ON “A FRAMESHIFT MUTATION AND ALTERNATE SPLICING IN HUMAN BRAIN GENERATE A FUNCTIONAL FORM OF THE PSEUDOGENE CYTOCHROME P4502D7 THAT DEMETHYLATES CODEINE TO MORPHINE”Harish V. Pai and Vijayalakshmi RavindranathDrug Metabolism and Disposition October 2005, 33 (10) 1566; DOI: https://doi.org/10.1124/dmd.105.006155
Park, Seonghee
- You have accessTHE BLOOD-BRAIN BARRIER SODIUM-DEPENDENT MULTIVITAMIN TRANSPORTER: A MOLECULAR FUNCTIONAL IN VITRO-IN SITU CORRELATIONSeonghee Park and Patrick J. SinkoDrug Metabolism and Disposition October 2005, 33 (10) 1547-1554; DOI: https://doi.org/10.1124/dmd.105.005231
Parte, Priyanka
- You have accessOXIDATION OF TAMOXIFEN BY HUMAN FLAVIN-CONTAINING MONOOXYGENASE (FMO) 1 AND FMO3 TO TAMOXIFEN-N-OXIDE AND ITS NOVEL REDUCTION BACK TO TAMOXIFEN BY HUMAN CYTOCHROMES P450 AND HEMOGLOBINPriyanka Parte and David KupferDrug Metabolism and Disposition October 2005, 33 (10) 1446-1452; DOI: https://doi.org/10.1124/dmd.104.000802
Patel, Purvi
- You have accessPHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITROJames M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. BurkaDrug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
Peng, Bin
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
Peterson, Lisa A.
- You have accessGLUTATHIONE TRAPPING TO MEASURE MICROSOMAL OXIDATION OF FURAN TO CIS-2-BUTENE-1,4-DIALLisa A. Peterson, Meredith E. Cummings, Choua C. Vu and Brock A. MatterDrug Metabolism and Disposition October 2005, 33 (10) 1453-1458; DOI: https://doi.org/10.1124/dmd.105.004432
Pfaar, Ulrike
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
Pokorny, Rolf
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
Pool, William F.
- You have accessA SIMPLE SEQUENTIAL INCUBATION METHOD FOR DECONVOLUTING THE COMPLICATED SEQUENTIAL METABOLISM OF CAPRAVIRINE IN HUMANSHai-Zhi Bu, Ping Kang, Ping Zhao, William F. Pool and Ellen Y. WuDrug Metabolism and Disposition October 2005, 33 (10) 1438-1445; DOI: https://doi.org/10.1124/dmd.105.005413
Putt, David A.
- You have accessPULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. CollinsDrug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
R
Ravindranath, Vijayalakshmi
- You have accessRESPONSE TO COMMENT ON “A FRAMESHIFT MUTATION AND ALTERNATE SPLICING IN HUMAN BRAIN GENERATE A FUNCTIONAL FORM OF THE PSEUDOGENE CYTOCHROME P4502D7 THAT DEMETHYLATES CODEINE TO MORPHINE”Harish V. Pai and Vijayalakshmi RavindranathDrug Metabolism and Disposition October 2005, 33 (10) 1566; DOI: https://doi.org/10.1124/dmd.105.006155
Renton, Kenneth W.
- You have accessTHE SIGNAL TRANSDUCTION PATHWAYS INVOLVED IN HEPATIC CYTOCHROME P450 REGULATION IN THE RAT DURING A LIPOPOLYSACCHARIDE-INDUCED MODEL OF CENTRAL NERVOUS SYSTEM INFLAMMATIONDalya Abdulla, Kerry B. Goralski, Elena Garcia Del Busto Cano and Kenneth W. RentonDrug Metabolism and Disposition October 2005, 33 (10) 1521-1531; DOI: https://doi.org/10.1124/dmd.105.004564
Ritter, Joseph K.
- You have accessAN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITYKristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. RitterDrug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663
S
Sai, Kimie
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Saijo, Nagahiro
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Saito, Hirohisa
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Saito, Yoshiro
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Sawada, Jun-ichi
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Sawada, Yasufumi
- You have accessPHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATSRisa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
Sayer, Claudia
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
Schilling, Boris
- You have accessEXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSAXiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin DingDrug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
Seiberling, Michael
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
Shimizu, Maki
- You have accessCONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANSMaki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622
Shirao, Kuniaki
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Shultz, Michael A.
- You have accessPULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. CollinsDrug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
Sinko, Patrick J.
- You have accessTHE BLOOD-BRAIN BARRIER SODIUM-DEPENDENT MULTIVITAMIN TRANSPORTER: A MOLECULAR FUNCTIONAL IN VITRO-IN SITU CORRELATIONSeonghee Park and Patrick J. SinkoDrug Metabolism and Disposition October 2005, 33 (10) 1547-1554; DOI: https://doi.org/10.1124/dmd.105.005231
Smith, Dennis A.
- You have accessSEEING THROUGH THE MIST: ABUNDANCE VERSUS PERCENTAGE. COMMENTARY ON METABOLITES IN SAFETY TESTINGDennis A. Smith and R. Scott ObachDrug Metabolism and Disposition October 2005, 33 (10) 1409-1417; DOI: https://doi.org/10.1124/dmd.105.005041
Smith, Philip C.
- You have accessAN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITYKristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. RitterDrug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663
So, James
- You have accessPHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITROJames M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. BurkaDrug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
Sobol, Eyal
- You have accessPHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATSEyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir BialerDrug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
Stern, Stephan T.
- You have accessAN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITYKristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. RitterDrug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663
Su, Ting
- You have accessEXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSAXiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin DingDrug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
Sugiyama, Yuichi
- You have accessCONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANSMaki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622
T
Tsujimoto, Masayuki
- You have accessPHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATSRisa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
Tyndale, Rachel F.
- You have accessHUMAN CYP2D6 AND MOUSE CYP2DS: ORGAN DISTRIBUTION IN A HUMANIZED MOUSE MODELSharon L. Miksys, Connie Cheung, Frank J. Gonzalez and Rachel F. TyndaleDrug Metabolism and Disposition October 2005, 33 (10) 1495-1502; DOI: https://doi.org/10.1124/dmd.105.005488
V
Valentine, John L.
- You have accessPHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITROJames M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. BurkaDrug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
Vu, Choua C.
- You have accessGLUTATHIONE TRAPPING TO MEASURE MICROSOMAL OXIDATION OF FURAN TO CIS-2-BUTENE-1,4-DIALLisa A. Peterson, Meredith E. Cummings, Choua C. Vu and Brock A. MatterDrug Metabolism and Disposition October 2005, 33 (10) 1453-1458; DOI: https://doi.org/10.1124/dmd.105.004432
W
Waldmeier, Felix
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
Weng, Yan
- You have accessEXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSAXiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin DingDrug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
Winkler, Ilan
- You have accessPHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATSEyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir BialerDrug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
Wu, Ellen Y.
- You have accessA SIMPLE SEQUENTIAL INCUBATION METHOD FOR DECONVOLUTING THE COMPLICATED SEQUENTIAL METABOLISM OF CAPRAVIRINE IN HUMANSHai-Zhi Bu, Ping Kang, Ping Zhao, William F. Pool and Ellen Y. WuDrug Metabolism and Disposition October 2005, 33 (10) 1438-1445; DOI: https://doi.org/10.1124/dmd.105.005413
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Yagen, Boris
- You have accessPHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATSEyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir BialerDrug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
Yamamoto, Noboru
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
Yokota, Hiroshi
- You have accessUDP-GLUCURONOSYLTRANSFERASE ISOFORMS CATALYZING GLUCURONIDATION OF HYDROXY-POLYCHLORINATED BIPHENYLS IN RATTomo Daidoji, Keisuke Gozu, Hidetomo Iwano, Hiroki Inoue and Hiroshi YokotaDrug Metabolism and Disposition October 2005, 33 (10) 1466-1476; DOI: https://doi.org/10.1124/dmd.105.004416
Yoshida, Teruhiko
- You have accessFUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi SawadaDrug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
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Zbinden, Peter
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
Zhang, Qing-Yu
- You have accessEXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSAXiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin DingDrug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
Zhang, Xiuling
- You have accessEXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSAXiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin DingDrug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
Zhao, Ping
- You have accessA SIMPLE SEQUENTIAL INCUBATION METHOD FOR DECONVOLUTING THE COMPLICATED SEQUENTIAL METABOLISM OF CAPRAVIRINE IN HUMANSHai-Zhi Bu, Ping Kang, Ping Zhao, William F. Pool and Ellen Y. WuDrug Metabolism and Disposition October 2005, 33 (10) 1438-1445; DOI: https://doi.org/10.1124/dmd.105.005413
Zollinger, Markus
- You have accessMETABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERSHans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard GrossDrug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283