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Drug Metabolism & Disposition

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Index by author

October 01, 2005; Volume 33,Issue 10
  • A
  • B
  • C
  • D
  • E
  • F
  • G
  • H
  • I
  • J
  • K
  • L
  • M
  • N
  • O
  • P
  • Q
  • R
  • S
  • T
  • U
  • V
  • W
  • X
  • Y
  • Z

A

  1. Abdulla, Dalya

    1. You have access
      THE SIGNAL TRANSDUCTION PATHWAYS INVOLVED IN HEPATIC CYTOCHROME P450 REGULATION IN THE RAT DURING A LIPOPOLYSACCHARIDE-INDUCED MODEL OF CENTRAL NERVOUS SYSTEM INFLAMMATION
      Dalya Abdulla, Kerry B. Goralski, Elena Garcia Del Busto Cano and Kenneth W. Renton
      Drug Metabolism and Disposition October 2005, 33 (10) 1521-1531; DOI: https://doi.org/10.1124/dmd.105.004564
  2. Ali, Shazia

    1. You have access
      AN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITY
      Kristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. Ritter
      Drug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663

B

  1. Baldwin, R. Michael

    1. You have access
      PULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1
      Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. Collins
      Drug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
  2. Ben-Am, Monique

    1. You have access
      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
  3. Bertrand, Marc

    1. You have access
      FUNCTIONAL EXPRESSION OF SINUSOIDAL DRUG TRANSPORTERS IN PRIMARY HUMAN AND RAT HEPATOCYTES
      Emilie Jigorel, Marc Le Vee, Claire Boursier-Neyret, Marc Bertrand and Olivier Fardel
      Drug Metabolism and Disposition October 2005, 33 (10) 1418-1422; DOI: https://doi.org/10.1124/dmd.105.004762
  4. Bialer, Meir

    1. You have access
      PHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATS
      Eyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir Bialer
      Drug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
  5. Black, Sherry R.

    1. You have access
      PHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITRO
      James M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. Burka
      Drug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
  6. Boursier-Neyret, Claire

    1. You have access
      FUNCTIONAL EXPRESSION OF SINUSOIDAL DRUG TRANSPORTERS IN PRIMARY HUMAN AND RAT HEPATOCYTES
      Emilie Jigorel, Marc Le Vee, Claire Boursier-Neyret, Marc Bertrand and Olivier Fardel
      Drug Metabolism and Disposition October 2005, 33 (10) 1418-1422; DOI: https://doi.org/10.1124/dmd.105.004762
  7. Britzi, Malka

    1. You have access
      PHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATS
      Eyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir Bialer
      Drug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
  8. Bu, Hai-Zhi

    1. You have access
      A SIMPLE SEQUENTIAL INCUBATION METHOD FOR DECONVOLUTING THE COMPLICATED SEQUENTIAL METABOLISM OF CAPRAVIRINE IN HUMANS
      Hai-Zhi Bu, Ping Kang, Ping Zhao, William F. Pool and Ellen Y. Wu
      Drug Metabolism and Disposition October 2005, 33 (10) 1438-1445; DOI: https://doi.org/10.1124/dmd.105.005413
  9. Burka, Leo T.

    1. You have access
      PHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITRO
      James M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. Burka
      Drug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317

C

  1. Chen, Ying

    1. You have access
      EXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSA
      Xiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin Ding
      Drug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
  2. Cheung, Connie

    1. You have access
      HUMAN CYP2D6 AND MOUSE CYP2DS: ORGAN DISTRIBUTION IN A HUMANIZED MOUSE MODEL
      Sharon L. Miksys, Connie Cheung, Frank J. Gonzalez and Rachel F. Tyndale
      Drug Metabolism and Disposition October 2005, 33 (10) 1495-1502; DOI: https://doi.org/10.1124/dmd.105.005488
  3. Churchwell, Mona I.

    1. You have access
      METABOLISM OF PIGMENT YELLOW 74 BY RAT AND HUMAN MICROSOMAL PROTEINS
      Yanyan Cui, Mona I. Churchwell, Letha H. Couch, Daniel R. Doerge and Paul C. Howard
      Drug Metabolism and Disposition October 2005, 33 (10) 1459-1465; DOI: https://doi.org/10.1124/dmd.104.003285
  4. Clement, Bernd

    1. You have access
      METABOLISM OF N-HYDROXYGUANIDINES (N-HYDROXYDEBRISOQUINE) IN HUMAN AND PORCINE HEPATOCYTES: REDUCTION AND FORMATION OF GLUCURONIDES
      Anja Kristina Froehlich, Ulrich Girreser and Bernd Clement
      Drug Metabolism and Disposition October 2005, 33 (10) 1532-1537; DOI: https://doi.org/10.1124/dmd.105.004572
  5. Coleman, Donna P.

    1. You have access
      PHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITRO
      James M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. Burka
      Drug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
  6. Collins, Kathy S.

    1. You have access
      PULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1
      Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. Collins
      Drug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
  7. Couch, Letha H.

    1. You have access
      METABOLISM OF PIGMENT YELLOW 74 BY RAT AND HUMAN MICROSOMAL PROTEINS
      Yanyan Cui, Mona I. Churchwell, Letha H. Couch, Daniel R. Doerge and Paul C. Howard
      Drug Metabolism and Disposition October 2005, 33 (10) 1459-1465; DOI: https://doi.org/10.1124/dmd.104.003285
  8. Cui, Yanyan

    1. You have access
      METABOLISM OF PIGMENT YELLOW 74 BY RAT AND HUMAN MICROSOMAL PROTEINS
      Yanyan Cui, Mona I. Churchwell, Letha H. Couch, Daniel R. Doerge and Paul C. Howard
      Drug Metabolism and Disposition October 2005, 33 (10) 1459-1465; DOI: https://doi.org/10.1124/dmd.104.003285
  9. Cummings, Meredith E.

    1. You have access
      GLUTATHIONE TRAPPING TO MEASURE MICROSOMAL OXIDATION OF FURAN TO CIS-2-BUTENE-1,4-DIAL
      Lisa A. Peterson, Meredith E. Cummings, Choua C. Vu and Brock A. Matter
      Drug Metabolism and Disposition October 2005, 33 (10) 1453-1458; DOI: https://doi.org/10.1124/dmd.105.004432

D

  1. Daidoji, Tomo

    1. You have access
      UDP-GLUCURONOSYLTRANSFERASE ISOFORMS CATALYZING GLUCURONIDATION OF HYDROXY-POLYCHLORINATED BIPHENYLS IN RAT
      Tomo Daidoji, Keisuke Gozu, Hidetomo Iwano, Hiroki Inoue and Hiroshi Yokota
      Drug Metabolism and Disposition October 2005, 33 (10) 1466-1476; DOI: https://doi.org/10.1124/dmd.105.004416
  2. Del Busto Cano, Elena Garcia

    1. You have access
      THE SIGNAL TRANSDUCTION PATHWAYS INVOLVED IN HEPATIC CYTOCHROME P450 REGULATION IN THE RAT DURING A LIPOPOLYSACCHARIDE-INDUCED MODEL OF CENTRAL NERVOUS SYSTEM INFLAMMATION
      Dalya Abdulla, Kerry B. Goralski, Elena Garcia Del Busto Cano and Kenneth W. Renton
      Drug Metabolism and Disposition October 2005, 33 (10) 1521-1531; DOI: https://doi.org/10.1124/dmd.105.004564
  3. Ding, Xinxin

    1. You have access
      EXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSA
      Xiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin Ding
      Drug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
  4. Doerge, Daniel R.

    1. You have access
      METABOLISM OF PIGMENT YELLOW 74 BY RAT AND HUMAN MICROSOMAL PROTEINS
      Yanyan Cui, Mona I. Churchwell, Letha H. Couch, Daniel R. Doerge and Paul C. Howard
      Drug Metabolism and Disposition October 2005, 33 (10) 1459-1465; DOI: https://doi.org/10.1124/dmd.104.003285

E

  1. Etheridge, Amy S.

    1. You have access
      PHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITRO
      James M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. Burka
      Drug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317

F

  1. Fardel, Olivier

    1. You have access
      FUNCTIONAL EXPRESSION OF SINUSOIDAL DRUG TRANSPORTERS IN PRIMARY HUMAN AND RAT HEPATOCYTES
      Emilie Jigorel, Marc Le Vee, Claire Boursier-Neyret, Marc Bertrand and Olivier Fardel
      Drug Metabolism and Disposition October 2005, 33 (10) 1418-1422; DOI: https://doi.org/10.1124/dmd.105.004762
  2. Forkert, Poh-Gek

    1. You have access
      PULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1
      Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. Collins
      Drug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
  3. Froehlich, Anja Kristina

    1. You have access
      METABOLISM OF N-HYDROXYGUANIDINES (N-HYDROXYDEBRISOQUINE) IN HUMAN AND PORCINE HEPATOCYTES: REDUCTION AND FORMATION OF GLUCURONIDES
      Anja Kristina Froehlich, Ulrich Girreser and Bernd Clement
      Drug Metabolism and Disposition October 2005, 33 (10) 1532-1537; DOI: https://doi.org/10.1124/dmd.105.004572
  4. Fuse, Kaori

    1. You have access
      CONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANS
      Maki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi Sugiyama
      Drug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622

G

  1. Gibson, Dan

    1. You have access
      PHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATS
      Eyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir Bialer
      Drug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
  2. Girreser, Ulrich

    1. You have access
      METABOLISM OF N-HYDROXYGUANIDINES (N-HYDROXYDEBRISOQUINE) IN HUMAN AND PORCINE HEPATOCYTES: REDUCTION AND FORMATION OF GLUCURONIDES
      Anja Kristina Froehlich, Ulrich Girreser and Bernd Clement
      Drug Metabolism and Disposition October 2005, 33 (10) 1532-1537; DOI: https://doi.org/10.1124/dmd.105.004572
  3. Gonzalez, Frank J.

    1. You have access
      HUMAN CYP2D6 AND MOUSE CYP2DS: ORGAN DISTRIBUTION IN A HUMANIZED MOUSE MODEL
      Sharon L. Miksys, Connie Cheung, Frank J. Gonzalez and Rachel F. Tyndale
      Drug Metabolism and Disposition October 2005, 33 (10) 1495-1502; DOI: https://doi.org/10.1124/dmd.105.005488
  4. Goralski, Kerry B.

    1. You have access
      THE SIGNAL TRANSDUCTION PATHWAYS INVOLVED IN HEPATIC CYTOCHROME P450 REGULATION IN THE RAT DURING A LIPOPOLYSACCHARIDE-INDUCED MODEL OF CENTRAL NERVOUS SYSTEM INFLAMMATION
      Dalya Abdulla, Kerry B. Goralski, Elena Garcia Del Busto Cano and Kenneth W. Renton
      Drug Metabolism and Disposition October 2005, 33 (10) 1521-1531; DOI: https://doi.org/10.1124/dmd.105.004564
  5. Gozu, Keisuke

    1. You have access
      UDP-GLUCURONOSYLTRANSFERASE ISOFORMS CATALYZING GLUCURONIDATION OF HYDROXY-POLYCHLORINATED BIPHENYLS IN RAT
      Tomo Daidoji, Keisuke Gozu, Hidetomo Iwano, Hiroki Inoue and Hiroshi Yokota
      Drug Metabolism and Disposition October 2005, 33 (10) 1466-1476; DOI: https://doi.org/10.1124/dmd.105.004416
  6. Gross, Gerhard

    1. You have access
      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
  7. Gschwind, Hans-Peter

    1. You have access
      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
  8. Gu, Jun

    1. You have access
      EXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSA
      Xiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin Ding
      Drug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769

H

  1. Hayes, Michael

    1. You have access
      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
  2. Hoskins, Janelle M.

    1. You have access
      COMMENT ON “A FRAMESHIFT MUTATION AND ALTERNATE SPLICING IN HUMAN BRAIN GENERATE A FUNCTIONAL FORM OF THE PSEUDOGENE CYTOCHROME P4502D7 THAT DEMETHYLATES CODEINE TO MORPHINE”
      Janelle M. Hoskins, Sharon Marsh and Howard L. McLeod
      Drug Metabolism and Disposition October 2005, 33 (10) 1564-1565; DOI: https://doi.org/10.1124/dmd.105.005736
  3. Howard, Paul C.

    1. You have access
      METABOLISM OF PIGMENT YELLOW 74 BY RAT AND HUMAN MICROSOMAL PROTEINS
      Yanyan Cui, Mona I. Churchwell, Letha H. Couch, Daniel R. Doerge and Paul C. Howard
      Drug Metabolism and Disposition October 2005, 33 (10) 1459-1465; DOI: https://doi.org/10.1124/dmd.104.003285

I

  1. Inoue, Hiroki

    1. You have access
      UDP-GLUCURONOSYLTRANSFERASE ISOFORMS CATALYZING GLUCURONIDATION OF HYDROXY-POLYCHLORINATED BIPHENYLS IN RAT
      Tomo Daidoji, Keisuke Gozu, Hidetomo Iwano, Hiroki Inoue and Hiroshi Yokota
      Drug Metabolism and Disposition October 2005, 33 (10) 1466-1476; DOI: https://doi.org/10.1124/dmd.105.004416
  2. Iwano, Hidetomo

    1. You have access
      UDP-GLUCURONOSYLTRANSFERASE ISOFORMS CATALYZING GLUCURONIDATION OF HYDROXY-POLYCHLORINATED BIPHENYLS IN RAT
      Tomo Daidoji, Keisuke Gozu, Hidetomo Iwano, Hiroki Inoue and Hiroshi Yokota
      Drug Metabolism and Disposition October 2005, 33 (10) 1466-1476; DOI: https://doi.org/10.1124/dmd.105.004416

J

  1. Jigorel, Emilie

    1. You have access
      FUNCTIONAL EXPRESSION OF SINUSOIDAL DRUG TRANSPORTERS IN PRIMARY HUMAN AND RAT HEPATOCYTES
      Emilie Jigorel, Marc Le Vee, Claire Boursier-Neyret, Marc Bertrand and Olivier Fardel
      Drug Metabolism and Disposition October 2005, 33 (10) 1418-1422; DOI: https://doi.org/10.1124/dmd.105.004762

K

  1. Kang, Ping

    1. You have access
      A SIMPLE SEQUENTIAL INCUBATION METHOD FOR DECONVOLUTING THE COMPLICATED SEQUENTIAL METABOLISM OF CAPRAVIRINE IN HUMANS
      Hai-Zhi Bu, Ping Kang, Ping Zhao, William F. Pool and Ellen Y. Wu
      Drug Metabolism and Disposition October 2005, 33 (10) 1438-1445; DOI: https://doi.org/10.1124/dmd.105.005413
  2. Kessler, Fay K.

    1. You have access
      AN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITY
      Kristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. Ritter
      Drug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663
  3. Kim, Su-Ryang

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  4. Kogetsu, Hirokuni

    1. You have access
      PHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATS
      Risa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
  5. Kubo, Takashi

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  6. Kumagai, Yoichi

    1. You have access
      PHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATS
      Risa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
  7. Kupfer, David

    1. You have access
      OXIDATION OF TAMOXIFEN BY HUMAN FLAVIN-CONTAINING MONOOXYGENASE (FMO) 1 AND FMO3 TO TAMOXIFEN-N-OXIDE AND ITS NOVEL REDUCTION BACK TO TAMOXIFEN BY HUMAN CYTOCHROMES P450 AND HEMOGLOBIN
      Priyanka Parte and David Kupfer
      Drug Metabolism and Disposition October 2005, 33 (10) 1446-1452; DOI: https://doi.org/10.1124/dmd.104.000802
  8. Kusuhara, Hiroyuki

    1. You have access
      CONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANS
      Maki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi Sugiyama
      Drug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622

L

  1. Lash, Lawrence H.

    1. You have access
      PULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1
      Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. Collins
      Drug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
  2. Le Vee, Marc

    1. You have access
      FUNCTIONAL EXPRESSION OF SINUSOIDAL DRUG TRANSPORTERS IN PRIMARY HUMAN AND RAT HEPATOCYTES
      Emilie Jigorel, Marc Le Vee, Claire Boursier-Neyret, Marc Bertrand and Olivier Fardel
      Drug Metabolism and Disposition October 2005, 33 (10) 1418-1422; DOI: https://doi.org/10.1124/dmd.105.004762
  3. Ling, Guoyu

    1. You have access
      EXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSA
      Xiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin Ding
      Drug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
  4. Liu, Dazhi

    1. You have access
      EXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSA
      Xiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin Ding
      Drug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769

M

  1. Maeda, Kazuya

    1. You have access
      CONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANS
      Maki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi Sugiyama
      Drug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622
  2. Marsh, Sharon

    1. You have access
      COMMENT ON “A FRAMESHIFT MUTATION AND ALTERNATE SPLICING IN HUMAN BRAIN GENERATE A FUNCTIONAL FORM OF THE PSEUDOGENE CYTOCHROME P4502D7 THAT DEMETHYLATES CODEINE TO MORPHINE”
      Janelle M. Hoskins, Sharon Marsh and Howard L. McLeod
      Drug Metabolism and Disposition October 2005, 33 (10) 1564-1565; DOI: https://doi.org/10.1124/dmd.105.005736
  3. Mathews, James M.

    1. You have access
      PHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITRO
      James M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. Burka
      Drug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
  4. Matsumoto, Kenji

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  5. Matter, Brock A.

    1. You have access
      GLUTATHIONE TRAPPING TO MEASURE MICROSOMAL OXIDATION OF FURAN TO CIS-2-BUTENE-1,4-DIAL
      Lisa A. Peterson, Meredith E. Cummings, Choua C. Vu and Brock A. Matter
      Drug Metabolism and Disposition October 2005, 33 (10) 1453-1458; DOI: https://doi.org/10.1124/dmd.105.004432
  6. McLeod, Howard L.

    1. You have access
      COMMENT ON “A FRAMESHIFT MUTATION AND ALTERNATE SPLICING IN HUMAN BRAIN GENERATE A FUNCTIONAL FORM OF THE PSEUDOGENE CYTOCHROME P4502D7 THAT DEMETHYLATES CODEINE TO MORPHINE”
      Janelle M. Hoskins, Sharon Marsh and Howard L. McLeod
      Drug Metabolism and Disposition October 2005, 33 (10) 1564-1565; DOI: https://doi.org/10.1124/dmd.105.005736
  7. Miksys, Sharon L.

    1. You have access
      HUMAN CYP2D6 AND MOUSE CYP2DS: ORGAN DISTRIBUTION IN A HUMANIZED MOUSE MODEL
      Sharon L. Miksys, Connie Cheung, Frank J. Gonzalez and Rachel F. Tyndale
      Drug Metabolism and Disposition October 2005, 33 (10) 1495-1502; DOI: https://doi.org/10.1124/dmd.105.005488
  8. Miles, Kristini K.

    1. You have access
      AN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITY
      Kristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. Ritter
      Drug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663
  9. Millen, Brandie

    1. You have access
      PULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1
      Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. Collins
      Drug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
  10. Minami, Hironobu

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587

N

  1. Nakajima, Toshiharu

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  2. Nasu, Risa

    1. You have access
      PHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATS
      Risa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
  3. Nishigaki, Ryuichiro

    1. You have access
      CONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANS
      Maki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi Sugiyama
      Drug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622

O

  1. Obach, R. Scott

    1. You have access
      SEEING THROUGH THE MIST: ABUNDANCE VERSUS PERCENTAGE. COMMENTARY ON METABOLITES IN SAFETY TESTING
      Dennis A. Smith and R. Scott Obach
      Drug Metabolism and Disposition October 2005, 33 (10) 1409-1417; DOI: https://doi.org/10.1124/dmd.105.005041
  2. Ohno, Yasuo

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  3. Ohtani, Hisakazu

    1. You have access
      PHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATS
      Risa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
  4. Ohtsu, Atsushi

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  5. Okudaira, Kazuho

    1. You have access
      CONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANS
      Maki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi Sugiyama
      Drug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622
  6. Ozawa, Shogo

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587

P

  1. Pai, Harish V.

    1. You have access
      RESPONSE TO COMMENT ON “A FRAMESHIFT MUTATION AND ALTERNATE SPLICING IN HUMAN BRAIN GENERATE A FUNCTIONAL FORM OF THE PSEUDOGENE CYTOCHROME P4502D7 THAT DEMETHYLATES CODEINE TO MORPHINE”
      Harish V. Pai and Vijayalakshmi Ravindranath
      Drug Metabolism and Disposition October 2005, 33 (10) 1566; DOI: https://doi.org/10.1124/dmd.105.006155
  2. Park, Seonghee

    1. You have access
      THE BLOOD-BRAIN BARRIER SODIUM-DEPENDENT MULTIVITAMIN TRANSPORTER: A MOLECULAR FUNCTIONAL IN VITRO-IN SITU CORRELATION
      Seonghee Park and Patrick J. Sinko
      Drug Metabolism and Disposition October 2005, 33 (10) 1547-1554; DOI: https://doi.org/10.1124/dmd.105.005231
  3. Parte, Priyanka

    1. You have access
      OXIDATION OF TAMOXIFEN BY HUMAN FLAVIN-CONTAINING MONOOXYGENASE (FMO) 1 AND FMO3 TO TAMOXIFEN-N-OXIDE AND ITS NOVEL REDUCTION BACK TO TAMOXIFEN BY HUMAN CYTOCHROMES P450 AND HEMOGLOBIN
      Priyanka Parte and David Kupfer
      Drug Metabolism and Disposition October 2005, 33 (10) 1446-1452; DOI: https://doi.org/10.1124/dmd.104.000802
  4. Patel, Purvi

    1. You have access
      PHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITRO
      James M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. Burka
      Drug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
  5. Peng, Bin

    1. You have access
      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
  6. Peterson, Lisa A.

    1. You have access
      GLUTATHIONE TRAPPING TO MEASURE MICROSOMAL OXIDATION OF FURAN TO CIS-2-BUTENE-1,4-DIAL
      Lisa A. Peterson, Meredith E. Cummings, Choua C. Vu and Brock A. Matter
      Drug Metabolism and Disposition October 2005, 33 (10) 1453-1458; DOI: https://doi.org/10.1124/dmd.105.004432
  7. Pfaar, Ulrike

    1. You have access
      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
  8. Pokorny, Rolf

    1. You have access
      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
  9. Pool, William F.

    1. You have access
      A SIMPLE SEQUENTIAL INCUBATION METHOD FOR DECONVOLUTING THE COMPLICATED SEQUENTIAL METABOLISM OF CAPRAVIRINE IN HUMANS
      Hai-Zhi Bu, Ping Kang, Ping Zhao, William F. Pool and Ellen Y. Wu
      Drug Metabolism and Disposition October 2005, 33 (10) 1438-1445; DOI: https://doi.org/10.1124/dmd.105.005413
  10. Putt, David A.

    1. You have access
      PULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1
      Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. Collins
      Drug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074

R

  1. Ravindranath, Vijayalakshmi

    1. You have access
      RESPONSE TO COMMENT ON “A FRAMESHIFT MUTATION AND ALTERNATE SPLICING IN HUMAN BRAIN GENERATE A FUNCTIONAL FORM OF THE PSEUDOGENE CYTOCHROME P4502D7 THAT DEMETHYLATES CODEINE TO MORPHINE”
      Harish V. Pai and Vijayalakshmi Ravindranath
      Drug Metabolism and Disposition October 2005, 33 (10) 1566; DOI: https://doi.org/10.1124/dmd.105.006155
  2. Renton, Kenneth W.

    1. You have access
      THE SIGNAL TRANSDUCTION PATHWAYS INVOLVED IN HEPATIC CYTOCHROME P450 REGULATION IN THE RAT DURING A LIPOPOLYSACCHARIDE-INDUCED MODEL OF CENTRAL NERVOUS SYSTEM INFLAMMATION
      Dalya Abdulla, Kerry B. Goralski, Elena Garcia Del Busto Cano and Kenneth W. Renton
      Drug Metabolism and Disposition October 2005, 33 (10) 1521-1531; DOI: https://doi.org/10.1124/dmd.105.004564
  3. Ritter, Joseph K.

    1. You have access
      AN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITY
      Kristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. Ritter
      Drug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663

S

  1. Sai, Kimie

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  2. Saijo, Nagahiro

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  3. Saito, Hirohisa

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  4. Saito, Yoshiro

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  5. Sawada, Jun-ichi

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  6. Sawada, Yasufumi

    1. You have access
      PHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATS
      Risa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
  7. Sayer, Claudia

    1. You have access
      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
  8. Schilling, Boris

    1. You have access
      EXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSA
      Xiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin Ding
      Drug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
  9. Seiberling, Michael

    1. You have access
      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
  10. Shimizu, Maki

    1. You have access
      CONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANS
      Maki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi Sugiyama
      Drug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622
  11. Shirao, Kuniaki

    1. You have access
      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  12. Shultz, Michael A.

    1. You have access
      PULMONARY BIOACTIVATION OF TRICHLOROETHYLENE TO CHLORAL HYDRATE: RELATIVE CONTRIBUTIONS OF CYP2E1, CYP2F, AND CYP2B1
      Poh-Gek Forkert, R. Michael Baldwin, Brandie Millen, Lawrence H. Lash, David A. Putt, Michael A. Shultz and Kathy S. Collins
      Drug Metabolism and Disposition October 2005, 33 (10) 1429-1437; DOI: https://doi.org/10.1124/dmd.105.005074
  13. Sinko, Patrick J.

    1. You have access
      THE BLOOD-BRAIN BARRIER SODIUM-DEPENDENT MULTIVITAMIN TRANSPORTER: A MOLECULAR FUNCTIONAL IN VITRO-IN SITU CORRELATION
      Seonghee Park and Patrick J. Sinko
      Drug Metabolism and Disposition October 2005, 33 (10) 1547-1554; DOI: https://doi.org/10.1124/dmd.105.005231
  14. Smith, Dennis A.

    1. You have access
      SEEING THROUGH THE MIST: ABUNDANCE VERSUS PERCENTAGE. COMMENTARY ON METABOLITES IN SAFETY TESTING
      Dennis A. Smith and R. Scott Obach
      Drug Metabolism and Disposition October 2005, 33 (10) 1409-1417; DOI: https://doi.org/10.1124/dmd.105.005041
  15. Smith, Philip C.

    1. You have access
      AN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITY
      Kristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. Ritter
      Drug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663
  16. So, James

    1. You have access
      PHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITRO
      James M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. Burka
      Drug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
  17. Sobol, Eyal

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      PHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATS
      Eyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir Bialer
      Drug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
  18. Stern, Stephan T.

    1. You have access
      AN INVESTIGATION OF HUMAN AND RAT LIVER MICROSOMAL MYCOPHENOLIC ACID GLUCURONIDATION: EVIDENCE FOR A PRINCIPAL ROLE OF UGT1A ENZYMES AND SPECIES DIFFERENCES IN UGT1A SPECIFICITY
      Kristini K. Miles, Stephan T. Stern, Philip C. Smith, Fay K. Kessler, Shazia Ali and Joseph K. Ritter
      Drug Metabolism and Disposition October 2005, 33 (10) 1513-1520; DOI: https://doi.org/10.1124/dmd.105.004663
  19. Su, Ting

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      EXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSA
      Xiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin Ding
      Drug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
  20. Sugiyama, Yuichi

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      CONTRIBUTION OF OATP (ORGANIC ANION-TRANSPORTING POLYPEPTIDE) FAMILY TRANSPORTERS TO THE HEPATIC UPTAKE OF FEXOFENADINE IN HUMANS
      Maki Shimizu, Kaori Fuse, Kazuho Okudaira, Ryuichiro Nishigaki, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi Sugiyama
      Drug Metabolism and Disposition October 2005, 33 (10) 1477-1481; DOI: https://doi.org/10.1124/dmd.105.004622

T

  1. Tsujimoto, Masayuki

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      PHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL FOR PRALMORELIN HYDROCHLORIDE IN RATS
      Risa Nasu, Yoichi Kumagai, Hirokuni Kogetsu, Masayuki Tsujimoto, Hisakazu Ohtani and Yasufumi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1488-1494; DOI: https://doi.org/10.1124/dmd.104.001040
  2. Tyndale, Rachel F.

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      HUMAN CYP2D6 AND MOUSE CYP2DS: ORGAN DISTRIBUTION IN A HUMANIZED MOUSE MODEL
      Sharon L. Miksys, Connie Cheung, Frank J. Gonzalez and Rachel F. Tyndale
      Drug Metabolism and Disposition October 2005, 33 (10) 1495-1502; DOI: https://doi.org/10.1124/dmd.105.005488

V

  1. Valentine, John L.

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      PHARMACOKINETICS AND DISPOSITION OF THE KAVALACTONE KAWAIN: INTERACTION WITH KAVA EXTRACT AND KAVALACTONES IN VIVO AND IN VITRO
      James M. Mathews, Amy S. Etheridge, John L. Valentine, Sherry R. Black, Donna P. Coleman, Purvi Patel, James So and Leo T. Burka
      Drug Metabolism and Disposition October 2005, 33 (10) 1555-1563; DOI: https://doi.org/10.1124/dmd.105.004317
  2. Vu, Choua C.

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      GLUTATHIONE TRAPPING TO MEASURE MICROSOMAL OXIDATION OF FURAN TO CIS-2-BUTENE-1,4-DIAL
      Lisa A. Peterson, Meredith E. Cummings, Choua C. Vu and Brock A. Matter
      Drug Metabolism and Disposition October 2005, 33 (10) 1453-1458; DOI: https://doi.org/10.1124/dmd.105.004432

W

  1. Waldmeier, Felix

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      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
  2. Weng, Yan

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      EXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSA
      Xiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin Ding
      Drug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
  3. Winkler, Ilan

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      PHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATS
      Eyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir Bialer
      Drug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
  4. Wu, Ellen Y.

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      A SIMPLE SEQUENTIAL INCUBATION METHOD FOR DECONVOLUTING THE COMPLICATED SEQUENTIAL METABOLISM OF CAPRAVIRINE IN HUMANS
      Hai-Zhi Bu, Ping Kang, Ping Zhao, William F. Pool and Ellen Y. Wu
      Drug Metabolism and Disposition October 2005, 33 (10) 1438-1445; DOI: https://doi.org/10.1124/dmd.105.005413

Y

  1. Yagen, Boris

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      PHARMACOKINETICS AND METABOLISM OF A NEW POTENT ANTIEPILEPTIC DRUG, 2,2,3,3-TETRAMETHYCYCLOPROPANECARBONYLUREA, IN RATS
      Eyal Sobol, Boris Yagen, Ilan Winkler, Malka Britzi, Dan Gibson and Meir Bialer
      Drug Metabolism and Disposition October 2005, 33 (10) 1538-1546; DOI: https://doi.org/10.1124/dmd.105.005637
  2. Yamamoto, Noboru

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      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587
  3. Yokota, Hiroshi

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      UDP-GLUCURONOSYLTRANSFERASE ISOFORMS CATALYZING GLUCURONIDATION OF HYDROXY-POLYCHLORINATED BIPHENYLS IN RAT
      Tomo Daidoji, Keisuke Gozu, Hidetomo Iwano, Hiroki Inoue and Hiroshi Yokota
      Drug Metabolism and Disposition October 2005, 33 (10) 1466-1476; DOI: https://doi.org/10.1124/dmd.105.004416
  4. Yoshida, Teruhiko

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      FUNCTIONAL CHARACTERIZATION OF THREE NATURALLY OCCURRING SINGLE NUCLEOTIDE POLYMORPHISMS IN THE CES2 GENE ENCODING CARBOXYLESTERASE 2 (HCE-2)
      Takashi Kubo, Su-Ryang Kim, Kimie Sai, Yoshiro Saito, Toshiharu Nakajima, Kenji Matsumoto, Hirohisa Saito, Kuniaki Shirao, Noboru Yamamoto, Hironobu Minami, Atsushi Ohtsu, Teruhiko Yoshida, Nagahiro Saijo, Yasuo Ohno, Shogo Ozawa and Jun-ichi Sawada
      Drug Metabolism and Disposition October 2005, 33 (10) 1482-1487; DOI: https://doi.org/10.1124/dmd.105.005587

Z

  1. Zbinden, Peter

    1. You have access
      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
  2. Zhang, Qing-Yu

    1. You have access
      EXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSA
      Xiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin Ding
      Drug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
  3. Zhang, Xiuling

    1. You have access
      EXPRESSION OF CYTOCHROME P450 AND OTHER BIOTRANSFORMATION GENES IN FETAL AND ADULT HUMAN NASAL MUCOSA
      Xiuling Zhang, Qing-Yu Zhang, Dazhi Liu, Ting Su, Yan Weng, Guoyu Ling, Ying Chen, Jun Gu, Boris Schilling and Xinxin Ding
      Drug Metabolism and Disposition October 2005, 33 (10) 1423-1428; DOI: https://doi.org/10.1124/dmd.105.005769
  4. Zhao, Ping

    1. You have access
      A SIMPLE SEQUENTIAL INCUBATION METHOD FOR DECONVOLUTING THE COMPLICATED SEQUENTIAL METABOLISM OF CAPRAVIRINE IN HUMANS
      Hai-Zhi Bu, Ping Kang, Ping Zhao, William F. Pool and Ellen Y. Wu
      Drug Metabolism and Disposition October 2005, 33 (10) 1438-1445; DOI: https://doi.org/10.1124/dmd.105.005413
  5. Zollinger, Markus

    1. You have access
      METABOLISM AND DISPOSITION OF IMATINIB MESYLATE IN HEALTHY VOLUNTEERS
      Hans-Peter Gschwind, Ulrike Pfaar, Felix Waldmeier, Markus Zollinger, Claudia Sayer, Peter Zbinden, Michael Hayes, Rolf Pokorny, Michael Seiberling, Monique Ben-Am, Bin Peng and Gerhard Gross
      Drug Metabolism and Disposition October 2005, 33 (10) 1503-1512; DOI: https://doi.org/10.1124/dmd.105.004283
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Drug Metabolism and Disposition: 33 (10)
Drug Metabolism and Disposition
Vol. 33, Issue 10
1 Oct 2005
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  • Cytochrome P450 inhibitors. Evaluation of specificities in the in vitrometabolism of therapeutic agents by human liver microsomes.
  • Prediction of Human Clearance of Twenty-Nine Drugs from Hepatic Microsomal Intrinsic Clearance Data: An Examination of In Vitro Half-Life Approach and Nonspecific Binding to Microsomes
  • DRUG-DRUG INTERACTIONS FOR UDP-GLUCURONOSYLTRANSFERASE SUBSTRATES: A PHARMACOKINETIC EXPLANATION FOR TYPICALLY OBSERVED LOW EXPOSURE (AUCI/AUC) RATIOS
  • In Vitro-In Vivo Scaling of CYP Kinetic Data Not Consistent with the Classical Michaelis-Menten Model
  • THE HUMAN INTESTINAL CYTOCHROME P450 “PIE”
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